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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-1-[2-(2,6-dimethylphenoxy)acetyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6R)-1-[2-(2,6-dimethylphenoxy)acetyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[2-(2,6-dimethylphenoxy)acetyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6S)-1-[2-(2,6-dimethylphenoxy)acetyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C25H31N5O
6-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[(2-Methoxy-3-methylphenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H21N5O2
6-[(2-Methoxy-3-methylphenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[[4-[(4-Fluorophenyl)methoxy]-3-iodo-5-methoxyphenyl]methylidene]-5-imino-3-phenyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C27H19FIN3O3S
6-[[4-[(4-Fluorophenyl)methoxy]-3-iodo-5-methoxyphenyl]methylidene]-5-imino-3-phenyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6R)-1-(2-methoxy-3-methylbenzoyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H27N3O3
(6R)-1-(2-methoxy-3-methylbenzoyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C23H24N4O2
(6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6R)-1-[3-(3-methoxy-1,2-oxazol-5-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O4
(6R)-1-[3-(3-methoxy-1,2-oxazol-5-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-Tert-butyl-2-[[4-(dimethylamino)phenyl]methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile —— C22H27N3S
6-Tert-butyl-2-[[4-(dimethylamino)phenyl]methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile
—— 6-[5-[[2-(Carboxymethoxy)phenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C18H19NO6S2
6-[5-[[2-(Carboxymethoxy)phenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— (6S)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)acetyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6S)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)acetyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-[(2-methoxy-3-methylphenyl)methyl]-2-[(2S)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C22H30N4O
6-[(2-methoxy-3-methylphenyl)methyl]-2-[(2S)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one —— C24H27N3O3
(6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one
—— (6S)-1-(3-methoxypropanoyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H28N2O3
(6S)-1-(3-methoxypropanoyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-[3-(2,6-dimethylanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C21H23N5O4
6-[3-(2,6-dimethylanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6'-[4-(2-hydroxyethoxy)phenyl]-1',2-dioxo-3',4'-diphenyl-N-prop-2-enylspiro[1H-indole-3,7'-4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine]-8'-carboxamide —— C38H35N3O6
6'-[4-(2-hydroxyethoxy)phenyl]-1',2-dioxo-3',4'-diphenyl-N-prop-2-enylspiro[1H-indole-3,7'-4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine]-8'-carboxamide
—— (6S)-1-[3-(3-methoxy-1,2-oxazol-5-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O4
(6S)-1-[3-(3-methoxy-1,2-oxazol-5-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one —— C24H27N3O3
(6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one
—— (6R)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)acetyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6R)-1-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)acetyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6R)-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-(2-methoxyacetyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C22H26N2O3
(6R)-1-(2-methoxyacetyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one —— C26H30N4O2
(6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one
—— (6S)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H31N3O3
(6S)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C23H24N4O2
(6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one —— C24H27N3O3
(6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one
—— (6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one —— C26H27N3O2
(6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one
—— (6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C25H25N3O2
(6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-(2-methoxyacetyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C22H26N2O3
(6S)-1-(2-methoxyacetyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H31N3O3
(6R)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclobutanecarbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C24H28N2O2
(6S)-1-(cyclobutanecarbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclobutanecarbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C24H28N2O2
(6R)-1-(cyclobutanecarbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one —— C26H30N4O2
(6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one
—— (6S)-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6S)-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one —— C24H27N3O3
(6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one
—— (6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one —— C26H30N4O2
(6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one —— C26H27N3O2
(6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one
—— (6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one —— C26H30N4O2
(6R)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-1,4-diazepan-5-one
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C27H36N4O2
6-(4-methylcyclohexyl)-2-[(2R)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(3-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H30N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(3-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-acetyl-2-[(2S)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-acetyl-2-[(2S)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-acetyl-2-[(2R)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-acetyl-2-[(2R)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[2-(3-methylphenyl)acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C22H23N3O2
6-[1-[2-(3-methylphenyl)acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[2-(3-methylphenyl)acetyl]-1,4-diazepan-5-one —— C28H30N2O3
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[2-(3-methylphenyl)acetyl]-1,4-diazepan-5-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(3-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H30N4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(3-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Amino-4-(4-fluorophenyl)-3-(pyridin-2-yl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C18H12FN5O
6-Amino-4-(4-fluorophenyl)-3-(pyridin-2-yl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[2-(3-methylphenyl)acetyl]-1,4-diazepan-5-one —— C28H30N2O3
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[2-(3-methylphenyl)acetyl]-1,4-diazepan-5-one
—— 6-methyl-2-[(3R)-1-[2-(3-methylphenyl)acetyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O2
6-methyl-2-[(3R)-1-[2-(3-methylphenyl)acetyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-2-[(3S)-1-[2-(3-methylphenyl)acetyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O2
6-methyl-2-[(3S)-1-[2-(3-methylphenyl)acetyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Amino-5-[2-[1-(2-ethoxyphenyl)tetrazol-5-yl]sulfanylacetyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H19N7O4S
6-Amino-5-[2-[1-(2-ethoxyphenyl)tetrazol-5-yl]sulfanylacetyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-methyl-N-[(2R)-1-[(3R)-3-(2-methylsulfonylacetyl)piperidin-1-yl]-1-oxopropan-2-yl]-1H-indole-2-carboxamide —— C21H27N3O5S
6-methyl-N-[(2R)-1-[(3R)-3-(2-methylsulfonylacetyl)piperidin-1-yl]-1-oxopropan-2-yl]-1H-indole-2-carboxamide