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—— 6-[(S)-(1-tert-butyltetrazol-5-yl)-[4-(4-methoxyphenyl)piperazin-1-yl]methyl]quinoline —— C26H31N7O
6-[(S)-(1-tert-butyltetrazol-5-yl)-[4-(4-methoxyphenyl)piperazin-1-yl]methyl]quinoline
—— 6-[(R)-azepan-1-yl-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]quinoline —— C22H30N6
6-[(R)-azepan-1-yl-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]quinoline
—— 6-(azepane-1-carbonyl)-3-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C23H32N4O3S
6-(azepane-1-carbonyl)-3-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— 6-(4-benzylpiperidine-1-carbonyl)-5-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C28H34N4O3S
6-(4-benzylpiperidine-1-carbonyl)-5-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-chloro-N-[(2S)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]-2H-chromene-3-carboxamide —— C19H15ClN2O4
6-chloro-N-[(2S)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]-2H-chromene-3-carboxamide
—— 6-[(2-chlorophenyl)methyl]-5-methyl-3-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C27H28ClN5O2
6-[(2-chlorophenyl)methyl]-5-methyl-3-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C27H33N5O4S
6-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-chloro-N-[(2R)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]-2H-chromene-3-carboxamide —— C19H15ClN2O4
6-chloro-N-[(2R)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]-2H-chromene-3-carboxamide
—— 6-methoxy-3-[[[(1R)-2-methyl-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C29H32N6O2S
6-methoxy-3-[[[(1R)-2-methyl-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C27H33N3O6S
6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methylbutyl)-4-oxo-1H-quinoline-3-carboxamide —— C22H31N3O4S
6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methylbutyl)-4-oxo-1H-quinoline-3-carboxamide
—— 6-[2-cyanoethyl(methyl)sulfamoyl]-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C24H26N4O6S
6-[2-cyanoethyl(methyl)sulfamoyl]-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C27H33N5O4S
6-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-[2-cyanoethyl(methyl)sulfamoyl]-N-(furan-2-ylmethyl)-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C24H26N4O6S
6-[2-cyanoethyl(methyl)sulfamoyl]-N-(furan-2-ylmethyl)-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C27H33N3O6S
6-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C27H33N3O6S
6-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(furan-2-ylmethyl)-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[(2-chlorophenyl)methyl]-5-methyl-3-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C27H28ClN5O2
6-[(2-chlorophenyl)methyl]-5-methyl-3-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6,7-dimethyl-3-[[[(1S)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C28H37N7O
6,7-dimethyl-3-[[[(1S)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methoxypropyl)-4-oxo-1H-quinoline-3-carboxamide —— C21H29N3O5S
6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methoxypropyl)-4-oxo-1H-quinoline-3-carboxamide
—— 6-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methylbutyl)-4-oxo-1H-quinoline-3-carboxamide —— C22H31N3O4S
6-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methylbutyl)-4-oxo-1H-quinoline-3-carboxamide
—— 6-[(4-fluorophenyl)-methylsulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C22H22FN3O5S
6-[(4-fluorophenyl)-methylsulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-methyl-3-[5-methyl-3-[[(2R)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C23H24N4O2
6-methyl-3-[5-methyl-3-[[(2R)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 6-[2-[[4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one —— C23H21N5O4S
6-[2-[[4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one
—— 6-[(4-fluorophenyl)-methylsulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C22H22FN3O5S
6-[(4-fluorophenyl)-methylsulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[ethyl-(4-fluorophenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H24FN3O5S
6-[ethyl-(4-fluorophenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[ethyl-(4-fluorophenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H24FN3O5S
6-[ethyl-(4-fluorophenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— [6-[(4-Fluorophenyl)methylamino]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C17H18FN3O
[6-[(4-Fluorophenyl)methylamino]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— (6-(3-Chlorophenylamino)pyridin-3-yl)(piperidin-1-yl)methanone —— C17H18ClN3O
(6-(3-Chlorophenylamino)pyridin-3-yl)(piperidin-1-yl)methanone
—— 6-ethoxy-3-[(S)-[(3S)-3-methylpiperidin-1-yl]-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C27H32N6O2
6-ethoxy-3-[(S)-[(3S)-3-methylpiperidin-1-yl]-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-[(S)-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-(1-cyclopentyltetrazol-5-yl)methyl]quinoline —— C23H29N7
6-[(S)-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-(1-cyclopentyltetrazol-5-yl)methyl]quinoline
—— 6-benzyl-5-[(2S)-2-ethylpiperidine-1-carbonyl]-10-methyl-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one —— C26H28N4O2
6-benzyl-5-[(2S)-2-ethylpiperidine-1-carbonyl]-10-methyl-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one
—— 6-benzyl-5-[(2S)-2-ethylpiperidine-1-carbonyl]-12-methyl-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one —— C26H28N4O2
6-benzyl-5-[(2S)-2-ethylpiperidine-1-carbonyl]-12-methyl-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one
—— 6-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-(2-phenylethyl)-[1,3]dioxolo[4,5-g]quinazolin-8-one —— C26H29N3O4S
6-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-(2-phenylethyl)-[1,3]dioxolo[4,5-g]quinazolin-8-one
—— 6-ethoxy-3-[(S)-[1-(furan-2-ylmethyl)tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-1H-quinolin-2-one —— C24H28N6O3
6-ethoxy-3-[(S)-[1-(furan-2-ylmethyl)tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-1H-quinolin-2-one
—— 6-methyl-2-[1-[4-[(3S)-3-methylpiperidin-1-yl]sulfonylphenyl]sulfonylpiperidin-4-yl]-1H-benzimidazole —— C25H32N4O4S2
6-methyl-2-[1-[4-[(3S)-3-methylpiperidin-1-yl]sulfonylphenyl]sulfonylpiperidin-4-yl]-1H-benzimidazole
—— 6-[(R)-(1-benzyltetrazol-5-yl)-(4-cyclohexylpiperazin-1-yl)methyl]quinoline —— C28H33N7
6-[(R)-(1-benzyltetrazol-5-yl)-(4-cyclohexylpiperazin-1-yl)methyl]quinoline
—— 6-[(4-fluorophenyl)methylamino]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C18H20FN3O2
6-[(4-fluorophenyl)methylamino]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— 6-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-(2-phenylethyl)-[1,3]dioxolo[4,5-g]quinazolin-8-one —— C26H29N3O4S
6-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-(2-phenylethyl)-[1,3]dioxolo[4,5-g]quinazolin-8-one
—— 6-[2-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]-N-(4-methoxyphenyl)hexanamide —— C25H32N4O4S2
6-[2-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]-N-(4-methoxyphenyl)hexanamide
—— (6-Ethyl-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-p-tolyl-amine —— C15H17N5
(6-Ethyl-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-p-tolyl-amine
—— 6-[2-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]-N-[(4-methylphenyl)methyl]hexanamide —— C26H34N4O3S2
6-[2-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]-N-[(4-methylphenyl)methyl]hexanamide
—— 6-[2-[(2R)-1-(2,6-diethylanilino)-1-oxobutan-2-yl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]hexanoic acid —— C26H33N3O4S2
6-[2-[(2R)-1-(2,6-diethylanilino)-1-oxobutan-2-yl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]hexanoic acid
—— 6-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-(2-phenylethyl)-[1,3]dioxolo[4,5-g]quinazolin-8-one —— C26H29N3O4S
6-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-(2-phenylethyl)-[1,3]dioxolo[4,5-g]quinazolin-8-one
—— 6-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-[(4-methoxyphenyl)methyl]-[1,3]dioxolo[4,5-g]quinazolin-8-one —— C26H29N3O5S
6-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-[(4-methoxyphenyl)methyl]-[1,3]dioxolo[4,5-g]quinazolin-8-one
—— (6R,9R)-5-acetyl-9-(3,4-dimethoxyphenyl)-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C27H26N2O5
(6R,9R)-5-acetyl-9-(3,4-dimethoxyphenyl)-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[2-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]-N-(4-methoxyphenyl)hexanamide —— C25H32N4O4S2
6-[2-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]-N-(4-methoxyphenyl)hexanamide
—— 6-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-[(4-methoxyphenyl)methyl]-[1,3]dioxolo[4,5-g]quinazolin-8-one —— C26H29N3O5S
6-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-[(4-methoxyphenyl)methyl]-[1,3]dioxolo[4,5-g]quinazolin-8-one
—— (6S,9R)-6-(4-fluorophenyl)-9-(4-methoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H22F4N2O3
(6S,9R)-6-(4-fluorophenyl)-9-(4-methoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]hexanamide —— C30H39N3O3S
6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]hexanamide
—— 6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]hexanamide —— C30H39N3O3S
6-[2-[(4-tert-butylphenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]hexanamide