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—— 6-bromo-5,6,8-trimethyl-5H-benzo[7]annulen-7-one —— C14H15BrO
6-bromo-5,6,8-trimethyl-5H-benzo[7]annulen-7-one
—— (6S)-1-benzyl-6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H29N3O
(6S)-1-benzyl-6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-(1-benzoylpiperidin-4-yl)-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H27FN2O2
(6S)-6-(1-benzoylpiperidin-4-yl)-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— 6-chloro-N-cyclohexyl-2-(thiophen-3-yl)imidazo[1,2-a]pyridin-3-amine —— C17H18ClN3S
6-chloro-N-cyclohexyl-2-(thiophen-3-yl)imidazo[1,2-a]pyridin-3-amine
—— (6R)-1-benzyl-6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C23H28N4O2
(6R)-1-benzyl-6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(4-fluorophenyl)methyl]-6-[1-(1-methyl-6-oxopyridazine-3-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H27FN4O3
(6R)-1-[(4-fluorophenyl)methyl]-6-[1-(1-methyl-6-oxopyridazine-3-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-benzyl-6-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H29N3O
(6S)-1-benzyl-6-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-[6-(4-hydroxy-3-methoxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-8-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid —— C34H36N2O8
6-[6-(4-hydroxy-3-methoxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-8-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid
—— 6-(5-chloro-2-hydroxyphenyl)-2-cyclohexyl-8-(4-methylanilino)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C39H38ClN3O5
6-(5-chloro-2-hydroxyphenyl)-2-cyclohexyl-8-(4-methylanilino)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6R)-1-benzyl-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C23H30N2O2
(6R)-1-benzyl-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[3-(4-fluorophenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C21H24FN3O2
(6R)-1-[3-(4-fluorophenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6R)-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C23H29FN2O2
(6R)-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— 6-(5-chloro-2-hydroxyphenyl)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-(4-chlorophenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H31Cl3N4O5S
6-(5-chloro-2-hydroxyphenyl)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-(4-chlorophenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6S)-1-benzyl-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C23H30N2O2
(6S)-1-benzyl-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-(1-benzylpiperidin-4-yl)-1-methyl-5,6-dihydro-2H-azepin-7-one —— C19H26N2O
(6R)-6-(1-benzylpiperidin-4-yl)-1-methyl-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-benzyl-6-[1-(cyclopentanecarbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H32N2O2
(6R)-1-benzyl-6-[1-(cyclopentanecarbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[3-(4-methoxyphenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C22H27N3O3
(6S)-1-[3-(4-methoxyphenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6R)-1-benzyl-6-(1-benzylpiperidin-4-yl)-5,6-dihydro-2H-azepin-7-one —— C25H30N2O
(6R)-1-benzyl-6-(1-benzylpiperidin-4-yl)-5,6-dihydro-2H-azepin-7-one
—— 6-[[1-(4-Ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C22H22N4O2S
6-[[1-(4-Ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6S)-1-[3-(4-fluorophenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C21H24FN3O2
(6S)-1-[3-(4-fluorophenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— 6-[(2R)-pyrrolidin-2-yl]-2H-pyrazolo[3,4-b]pyridin-3-amine —— C10H13N5
6-[(2R)-pyrrolidin-2-yl]-2H-pyrazolo[3,4-b]pyridin-3-amine
—— (6R)-6-(1-acetylpiperidin-4-yl)-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C20H25FN2O2
(6R)-6-(1-acetylpiperidin-4-yl)-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-(1-acetylpiperidin-4-yl)-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C20H25FN2O2
(6S)-6-(1-acetylpiperidin-4-yl)-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-(1-acetylpiperidin-4-yl)-1-benzyl-5,6-dihydro-2H-azepin-7-one —— C20H26N2O2
(6S)-6-(1-acetylpiperidin-4-yl)-1-benzyl-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[(4-fluorophenyl)methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one —— C19H25FN2O
(6S)-6-[1-[(4-fluorophenyl)methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[3-(4-methoxyphenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C22H27N3O3
(6R)-1-[3-(4-methoxyphenyl)propanoyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-6-[1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H28F2N2O2
(6S)-6-[1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-benzyl-6-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H29N3O
(6R)-1-benzyl-6-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C23H29FN2O2
(6S)-6-[1-(cyclobutanecarbonyl)piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-4-methyl-1-(2-phenylacetyl)-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C20H23N3O2
(6S)-4-methyl-1-(2-phenylacetyl)-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— 6-[[(2R)-2-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoxaline —— C24H23F2N5O
6-[[(2R)-2-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoxaline
—— (6R)-1-benzyl-6-[1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C28H31N3O2
(6R)-1-benzyl-6-[1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-Chloro-N-[5-ethyl-4-(thiophen-2-YL)-1,3-thiazol-2-YL]-2-oxo-2H-chromene-3-carboxamide —— C19H13ClN2O3S2
6-Chloro-N-[5-ethyl-4-(thiophen-2-YL)-1,3-thiazol-2-YL]-2-oxo-2H-chromene-3-carboxamide
—— (6R)-6-(1-acetylpiperidin-4-yl)-1-benzyl-5,6-dihydro-2H-azepin-7-one —— C20H26N2O2
(6R)-6-(1-acetylpiperidin-4-yl)-1-benzyl-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[2-(4-fluorophenyl)acetyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C20H22FN3O2
(6R)-1-[2-(4-fluorophenyl)acetyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-1-[2-(4-fluorophenoxy)acetyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C20H22FN3O3
(6S)-1-[2-(4-fluorophenoxy)acetyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6R)-6-[1-[(4-fluorophenyl)methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one —— C19H25FN2O
(6R)-6-[1-[(4-fluorophenyl)methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one
—— 6-[[1-(4-Ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C22H22N4O2S
6-[[1-(4-Ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6R)-1-benzyl-6-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C22H26N4O2
(6R)-1-benzyl-6-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-benzyl-6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H29N3O
(6R)-1-benzyl-6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(4-fluorophenyl)methyl]-6-[1-(1-methyl-6-oxopyridazine-3-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H27FN4O3
(6S)-1-[(4-fluorophenyl)methyl]-6-[1-(1-methyl-6-oxopyridazine-3-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-benzyl-6-[1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C28H31N3O2
(6S)-1-benzyl-6-[1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(4-fluorophenyl)methyl]-6-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H28FN3O
(6R)-1-[(4-fluorophenyl)methyl]-6-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-benzyl-6-(1-benzylpiperidin-4-yl)-5,6-dihydro-2H-azepin-7-one —— C25H30N2O
(6S)-1-benzyl-6-(1-benzylpiperidin-4-yl)-5,6-dihydro-2H-azepin-7-one
—— 6-[(2S)-pyrrolidin-2-yl]-2H-pyrazolo[3,4-b]pyridin-3-amine —— C10H13N5
6-[(2S)-pyrrolidin-2-yl]-2H-pyrazolo[3,4-b]pyridin-3-amine
—— (6R)-6-[1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H28F2N2O2
(6R)-6-[1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— 6((Dimethylamino)ME)-7-HO-2,8-dimethyl-3-(1-PH-1H-pyrazol-4-YL)-4H-chromen-4-one —— C23H23N3O3
6((Dimethylamino)ME)-7-HO-2,8-dimethyl-3-(1-PH-1H-pyrazol-4-YL)-4H-chromen-4-one
—— (6R)-1-[2-(4-fluorophenoxy)acetyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C20H22FN3O3
(6R)-1-[2-(4-fluorophenoxy)acetyl]-4-methyl-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-4-methyl-1-(3-phenylpropanoyl)-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C21H25N3O2
(6S)-4-methyl-1-(3-phenylpropanoyl)-6-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-1-[(4-fluorophenyl)methyl]-6-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C22H25FN4O2
(6S)-1-[(4-fluorophenyl)methyl]-6-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one