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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-1-(5-methylpyrazine-2-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2S
(6S)-1-(5-methylpyrazine-2-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N6O3
(6R)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(5-methylpyrazine-2-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2S
(6R)-1-(5-methylpyrazine-2-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1-methylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6S)-1-(1-methylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(cyclobutanecarbonyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H31N3O2
(6R)-1-(cyclobutanecarbonyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6S)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-5-one —— C24H27N5O2
(6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H28N4O3
(6R)-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(1-methylimidazole-2-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-1-(1-methylimidazole-2-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C28H36N2O3
(6S)-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O
(6R)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(1-methylimidazole-4-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-1-(1-methylimidazole-4-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyrazine-2-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H26N4O2S
(6S)-4-propyl-1-(pyrazine-2-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one —— C28H36N2O3
(6S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(1-methylimidazole-4-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-1-(1-methylimidazole-4-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(4-methylphenyl)phenyl]methyl]-4-propyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C26H30N4O2
(6R)-6-[[2-(4-methylphenyl)phenyl]methyl]-4-propyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O
(6R)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-acetyl-6-[[3-(2-fluorophenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one —— C23H27FN2O2
(6S)-1-acetyl-6-[[3-(2-fluorophenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(pyridin-3-ylmethyl)-1,4-diazepan-5-one —— C28H33N3O2
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2S
(6S)-4-propyl-1-(2-pyridin-3-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1-methylimidazole-2-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6S)-1-(1-methylimidazole-2-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(3-fluorobenzoyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H28FN3O2
(6S)-1-(3-fluorobenzoyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O3
(6R)-1-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N5O
(6R)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C25H29N5O2
(6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-1-(5-methyl-1H-pyrazole-4-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-1-(5-methyl-1H-pyrazole-4-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6R)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-propanoyl-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H29N3O2
(6R)-1-propanoyl-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C28H33N3O2
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6R)-1-(1-methylimidazole-4-carbonyl)-6-[[3-(3-methylphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one —— C27H32N4O2
(6R)-1-(1-methylimidazole-4-carbonyl)-6-[[3-(3-methylphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6R)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C27H33N3O3
(6R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6S)-4-propyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1-methylpyrazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6S)-1-(1-methylpyrazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C24H27N5O3
(6R)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N3O3S
(6R)-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(6-methylpyridin-2-yl)methyl]-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H32N4O
(6R)-1-[(6-methylpyridin-2-yl)methyl]-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1H-imidazol-2-ylmethyl)-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N5O
(6S)-1-(1H-imidazol-2-ylmethyl)-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[3-(2-fluorophenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one —— C26H29FN4O2
(6R)-6-[[3-(2-fluorophenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one