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—— (6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[[3-(4-fluorophenyl)phenyl]methyl]-4-methyl-1,4-diazepan-5-one —— C26H29FN4O
(6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[[3-(4-fluorophenyl)phenyl]methyl]-4-methyl-1,4-diazepan-5-one
—— 6-[(1-Benzylindol-3-yl)methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H24N6O3S
6-[(1-Benzylindol-3-yl)methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O
(6S)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[3-methoxy-4-(propan-2-yloxy)phenyl]-4-methyl-N-phenyl-2-sulfanyl-1,6-dihydropyrimidine-5-carboxamide —— C22H25N3O3S
6-[3-methoxy-4-(propan-2-yloxy)phenyl]-4-methyl-N-phenyl-2-sulfanyl-1,6-dihydropyrimidine-5-carboxamide
—— 6-[[2,5-Dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H20N6OS
6-[[2,5-Dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O
(6R)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-methyl-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-methyl-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O
(6R)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-methyl-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6R)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-methyl-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(4-benzhydrylpiperazin-1-yl)methyl]-2,3-dihydro-1H-inden-5-ol —— C27H30N2O
6-[(4-benzhydrylpiperazin-1-yl)methyl]-2,3-dihydro-1H-inden-5-ol
—— (6S)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O
(6S)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O
(6S)-4-ethyl-1-[(2-ethylpyrimidin-5-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-Methoxy-1-(4-methoxyphenyl)-7-phenylmethoxy-1,2,3,4-tetrahydroisoquinoline —— C24H25NO3
6-Methoxy-1-(4-methoxyphenyl)-7-phenylmethoxy-1,2,3,4-tetrahydroisoquinoline
—— 6,7-Dibromo-3-oxabicyclo[3.2.0]heptane-2,4-dione —— C6H4Br2O3
6,7-Dibromo-3-oxabicyclo[3.2.0]heptane-2,4-dione
—— 6-(cyclopropanecarbonyl)-2-[(3R)-1-[(4-ethylphenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H32N4O2
6-(cyclopropanecarbonyl)-2-[(3R)-1-[(4-ethylphenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethyl-2-[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]-1H-pyrimidin-4-one —— C14H23N3O
6-ethyl-2-[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]-1H-pyrimidin-4-one
—— 6-Amino-5-[2-[[5-(4-methoxyphenyl)-4-propan-2-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1,3-dimethylpyrimidine-2,4-dione —— C20H24N6O4S
6-Amino-5-[2-[[5-(4-methoxyphenyl)-4-propan-2-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-imino-11-methyl-2-oxo-7-(1-phenylethyl)-N-propan-2-yl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C24H25N5O2
6-imino-11-methyl-2-oxo-7-(1-phenylethyl)-N-propan-2-yl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-(cyclopropanecarbonyl)-2-[(3S)-1-[(4-ethylphenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H32N4O2
6-(cyclopropanecarbonyl)-2-[(3S)-1-[(4-ethylphenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3S)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C20H23N5OS
6-[(3S)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— 6-[2-(4-hydroxy-3-iodo-5-methoxyphenyl)ethenyl]-5-nitro-1H-pyrimidine-2,4-dione —— C13H10IN3O6
6-[2-(4-hydroxy-3-iodo-5-methoxyphenyl)ethenyl]-5-nitro-1H-pyrimidine-2,4-dione
—— 6-ethoxy-1-(4-iodophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C19H19IN2O
6-ethoxy-1-(4-iodophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-ethyl-2-[(3S)-1-(1-ethylsulfonylpiperidine-4-carbonyl)piperidin-3-yl]-1H-pyrimidin-4-one —— C19H30N4O4S
6-ethyl-2-[(3S)-1-(1-ethylsulfonylpiperidine-4-carbonyl)piperidin-3-yl]-1H-pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[(2R)-1-(5-ethyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H33N5O3
6-(cyclohexylmethyl)-2-[(2R)-1-(5-ethyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethyl-2-[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]-1H-pyrimidin-4-one —— C14H23N3O
6-ethyl-2-[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]-1H-pyrimidin-4-one
—— 6-ethyl-2-[(3R)-1-(1-ethylsulfonylpiperidine-4-carbonyl)piperidin-3-yl]-1H-pyrimidin-4-one —— C19H30N4O4S
6-ethyl-2-[(3R)-1-(1-ethylsulfonylpiperidine-4-carbonyl)piperidin-3-yl]-1H-pyrimidin-4-one
—— 6-Chloro-2-propan-2-ylquinoline-4-carboxylic acid —— C13H12ClNO2
6-Chloro-2-propan-2-ylquinoline-4-carboxylic acid
—— 6-ethyl-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-1H-pyrimidin-4-one —— C13H19N3O3
6-ethyl-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-1H-pyrimidin-4-one
—— 6-ethyl-2-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-1H-pyrimidin-4-one —— C18H23N3O4S
6-ethyl-2-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-1H-pyrimidin-4-one
—— 6-Chloro-8-fluoro-2-(3-fluoro-4-methoxyphenyl)quinoline-4-carboxylic acid —— C17H10ClF2NO3
6-Chloro-8-fluoro-2-(3-fluoro-4-methoxyphenyl)quinoline-4-carboxylic acid
—— 6-phenylmethoxy-1-(4-propan-2-ylphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C27H28N2O
6-phenylmethoxy-1-(4-propan-2-ylphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-ethyl-2-[(3S)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-1H-pyrimidin-4-one —— C18H23N3O4S
6-ethyl-2-[(3S)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-1H-pyrimidin-4-one
—— 6,8-Dichloro-2-(4-propan-2-ylphenyl)quinoline-4-carboxylic acid —— C19H15Cl2NO2
6,8-Dichloro-2-(4-propan-2-ylphenyl)quinoline-4-carboxylic acid
—— 6-Bromo-2-(5-bromo-1-benzofuran-2-yl)quinoline-4-carboxylic acid —— C18H9Br2NO3
6-Bromo-2-(5-bromo-1-benzofuran-2-yl)quinoline-4-carboxylic acid
—— 6,8-dimethyl-1-(2-nitrophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C19H19N3O2
6,8-dimethyl-1-(2-nitrophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-Ethyl-3-(1-piperidin-1-ylsulfonylpiperidin-4-yl)-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C19H25F3N4O3S
6-Ethyl-3-(1-piperidin-1-ylsulfonylpiperidin-4-yl)-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-ethyl-3-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
6-ethyl-3-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-Ethyl-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
6-Ethyl-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-ethyl-3-[(3R)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C21H23F3N4O
6-ethyl-3-[(3R)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-Ethyl-3-[1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C21H23F3N4O
6-Ethyl-3-[1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-Ethyl-3-(1-propan-2-ylsulfonylpiperidin-4-yl)-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C17H22F3N3O3S
6-Ethyl-3-(1-propan-2-ylsulfonylpiperidin-4-yl)-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— (6S)-1-(4-ethylthiadiazole-5-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C24H26N4O2S
(6S)-1-(4-ethylthiadiazole-5-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-Ethyl-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
6-Ethyl-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-[(1-Benzyl-2,5-dimethylindol-3-yl)methylidene]-5-imino-3-phenyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C30H24N4OS
6-[(1-Benzyl-2,5-dimethylindol-3-yl)methylidene]-5-imino-3-phenyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6S)-4-ethyl-1-(4-ethylthiadiazole-5-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2S
(6S)-4-ethyl-1-(4-ethylthiadiazole-5-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-ethyl-3-[3-(2-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methyl-1H-pyridin-2-one —— C21H21FN4O3
6-ethyl-3-[3-(2-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methyl-1H-pyridin-2-one
—— (6S)-4-ethyl-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H31N3O3
(6S)-4-ethyl-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-ethyl-3-[(3S)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C21H23F3N4O
6-ethyl-3-[(3S)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-ethyl-5-methyl-3-[(3S)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H23F3N4O3
6-ethyl-5-methyl-3-[(3S)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (6R)-1-(4-ethylthiadiazole-5-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C24H26N4O2S
(6R)-1-(4-ethylthiadiazole-5-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one