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—— 6-[cyclohexyl(methyl)sulfamoyl]-1-ethyl-N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide —— C29H44N4O4S
6-[cyclohexyl(methyl)sulfamoyl]-1-ethyl-N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide
—— 6-[cyclohexyl(methyl)sulfamoyl]-1-methyl-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide —— C27H40N4O4S
6-[cyclohexyl(methyl)sulfamoyl]-1-methyl-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide
—— 6-[(3-methoxyphenyl)sulfamoyl]-4-oxo-N-[(1R)-1-phenylethyl]-1H-quinoline-3-carboxamide —— C25H23N3O5S
6-[(3-methoxyphenyl)sulfamoyl]-4-oxo-N-[(1R)-1-phenylethyl]-1H-quinoline-3-carboxamide
—— 6-[(3-methoxyphenyl)sulfamoyl]-4-oxo-N-[(1S)-1-phenylethyl]-1H-quinoline-3-carboxamide —— C25H23N3O5S
6-[(3-methoxyphenyl)sulfamoyl]-4-oxo-N-[(1S)-1-phenylethyl]-1H-quinoline-3-carboxamide
—— 6-methoxy-1-[(4-methoxyphenyl)methyl]-3-[[[(2R)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid —— C28H30N2O4
6-methoxy-1-[(4-methoxyphenyl)methyl]-3-[[[(2R)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid
—— (6R,9S)-6-(3-fluorophenyl)-9-(4-methoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H22F4N2O3
(6R,9S)-6-(3-fluorophenyl)-9-(4-methoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[1-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(2-chlorophenyl)methyl]hexanamide —— C25H31ClN4O4S
6-[1-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(2-chlorophenyl)methyl]hexanamide
—— 6-[1-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-phenylhexanamide —— C24H30N4O4S
6-[1-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-phenylhexanamide
—— 6-ethyl-3-[(S)-[4-(2-fluorophenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C28H32FN7O2
6-ethyl-3-[(S)-[4-(2-fluorophenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (6S)-9,9-dimethyl-5-(3-methylbutanoyl)-6-pyridin-3-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H29N3O2
(6S)-9,9-dimethyl-5-(3-methylbutanoyl)-6-pyridin-3-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-ethyl-3-[(S)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H28N6O3
6-ethyl-3-[(S)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(S)-[4-(4-methoxyphenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C29H35N7O3
6-ethyl-3-[(S)-[4-(4-methoxyphenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-[1-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(4-fluorophenyl)methyl]hexanamide —— C28H35FN4O4S
6-[1-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(4-fluorophenyl)methyl]hexanamide
—— 6-methoxy-3-[(R)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one —— C22H28N6O3
6-methoxy-3-[(R)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one
—— 6-methoxy-3-[(S)-[4-(2-methoxyphenyl)piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C28H33N7O4
6-methoxy-3-[(S)-[4-(2-methoxyphenyl)piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (6S,9S)-2-chloro-6-(3-methoxyphenyl)-9-phenyl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H23ClN2O2
(6S,9S)-2-chloro-6-(3-methoxyphenyl)-9-phenyl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-ethyl-3-[(S)-(4-methylpiperidin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6-ethyl-3-[(S)-(4-methylpiperidin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-[1-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(2-chlorophenyl)methyl]hexanamide —— C25H31ClN4O4S
6-[1-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(2-chlorophenyl)methyl]hexanamide
—— 6-ethyl-3-[(S)-[(3R)-3-methylpiperidin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6-ethyl-3-[(S)-[(3R)-3-methylpiperidin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(R)-[4-(2-fluorophenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C28H32FN7O2
6-ethyl-3-[(R)-[4-(2-fluorophenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,8-dimethyl-3-[(R)-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C27H30N6O2
6,8-dimethyl-3-[(R)-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-methyl-3-[(S)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one —— C22H28N6O2
6-methyl-3-[(S)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one
—— 6-methyl-3-[(S)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-1H-quinolin-2-one —— C21H26N6O2
6-methyl-3-[(S)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-1H-quinolin-2-one
—— (6S)-6-(1H-indol-3-yl)-9,9-dimethyl-5-propanoyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H27N3O2
(6S)-6-(1H-indol-3-yl)-9,9-dimethyl-5-propanoyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6,7-dimethoxy-4-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-2-(2-methylpropyl)isoquinolin-1-one —— C28H35N3O4
6,7-dimethoxy-4-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-2-(2-methylpropyl)isoquinolin-1-one
—— 6-Nitro-3-(4-phenylpiperazine-1-carbonyl)chromen-2-one —— C20H17N3O5
6-Nitro-3-(4-phenylpiperazine-1-carbonyl)chromen-2-one
—— 6-methyl-3-[(S)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C21H26N6O3
6-methyl-3-[(S)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethoxy-4-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-2-(2-methylpropyl)isoquinolin-1-one —— C28H35N3O4
6,7-dimethoxy-4-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-2-(2-methylpropyl)isoquinolin-1-one
—— (6R)-6-tert-butyl-N-(furan-2-ylmethyl)-2-[(2-methylbenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C26H30N2O3S
(6R)-6-tert-butyl-N-(furan-2-ylmethyl)-2-[(2-methylbenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-3-ethyl-N-(4-fluorophenyl)-2-(2-methoxyphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C20H20FN3O3S
(6R)-3-ethyl-N-(4-fluorophenyl)-2-(2-methoxyphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-chloro-N-[(2,4-dichlorophenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C16H11Cl3N4O
6-chloro-N-[(2,4-dichlorophenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— 6-methoxy-1-[(4-methoxyphenyl)methyl]-3-[[[(2S)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid —— C28H30N2O4
6-methoxy-1-[(4-methoxyphenyl)methyl]-3-[[[(2S)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid
—— 6,7-dimethyl-2-[(5-phenyl-1H-pyrazol-4-yl)methylidene]-[1,3]thiazolo[3,2-a]benzimidazol-1-one —— C21H16N4OS
6,7-dimethyl-2-[(5-phenyl-1H-pyrazol-4-yl)methylidene]-[1,3]thiazolo[3,2-a]benzimidazol-1-one
—— (6R,9R)-6-(3,4-dimethoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H24N2O3S
(6R,9R)-6-(3,4-dimethoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-9-(3,4-dimethoxyphenyl)-6-[3-(trifluoromethyl)phenyl]-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H25F3N2O3
(6R,9S)-9-(3,4-dimethoxyphenyl)-6-[3-(trifluoromethyl)phenyl]-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-methoxy-3-(4-methylphenyl)sulfanyl-N-[(2R)-2-phenylpropyl]-1H-indole-2-carboxamide —— C26H26N2O2S
6-methoxy-3-(4-methylphenyl)sulfanyl-N-[(2R)-2-phenylpropyl]-1H-indole-2-carboxamide
—— 6-[(4-ethoxyphenyl)-methylsulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C24H27N3O6S
6-[(4-ethoxyphenyl)-methylsulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[methyl-(2-methylphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O5S
6-[methyl-(2-methylphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— (6R)-2-[(4-bromophenyl)methylideneamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile —— C17H15BrN2S
(6R)-2-[(4-bromophenyl)methylideneamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile
—— 6-[(4-ethoxyphenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O6S
6-[(4-ethoxyphenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— (6S)-2-(4-methoxyphenyl)imino-N-methyl-4-oxo-3-(2-phenylethyl)-1,3-thiazinane-6-carboxamide —— C21H23N3O3S
(6S)-2-(4-methoxyphenyl)imino-N-methyl-4-oxo-3-(2-phenylethyl)-1,3-thiazinane-6-carboxamide
—— 6-[(4-ethylphenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O5S
6-[(4-ethylphenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[(4-ethoxyphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O6S
6-[(4-ethoxyphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[(4-ethylphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O5S
6-[(4-ethylphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6-[(2-ethylphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O5S
6-[(2-ethylphenyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— (6S)-N-(5-chloro-2-methoxyphenyl)-6-methyl-2-(pyridin-3-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H24ClN3O2S
(6S)-N-(5-chloro-2-methoxyphenyl)-6-methyl-2-(pyridin-3-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[methyl-(2-methylphenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O5S
6-[methyl-(2-methylphenyl)sulfamoyl]-4-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— (6R)-3-[2-(4-methoxyphenyl)ethyl]-2-(4-methoxyphenyl)imino-N-methyl-4-oxo-1,3-thiazinane-6-carboxamide —— C22H25N3O4S
(6R)-3-[2-(4-methoxyphenyl)ethyl]-2-(4-methoxyphenyl)imino-N-methyl-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-Bromo-2-ethyl-3-methylquinoline-4-carboxylic acid —— C13H12BrNO2
6-Bromo-2-ethyl-3-methylquinoline-4-carboxylic acid
—— (6S,9R)-6-(5-methylfuran-2-yl)-9-phenyl-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C27H26N2O3
(6S,9R)-6-(5-methylfuran-2-yl)-9-phenyl-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one