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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(2,6-difluorophenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H24F2N4O
6-[(2,6-difluorophenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-2,3-dihydroimidazo[1,2-c]quinazolin-5-one —— C18H22N4O2
6-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-2,3-dihydroimidazo[1,2-c]quinazolin-5-one
—— 6-(2,4-Dimethoxybenzoyl)-2-(4-methylphenyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H23N3O4
6-(2,4-Dimethoxybenzoyl)-2-(4-methylphenyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1R,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C24H30FN3O4
6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1R,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— 6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C24H30FN3O4
6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— 6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C24H30FN3O4
6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— 6-methylheptyl (3S)-1,1-dioxothiolane-3-sulfonate —— C12H24O5S2
6-methylheptyl (3S)-1,1-dioxothiolane-3-sulfonate
—— 6-Chloro-2-(3,4-dichlorophenyl)quinoline-4-carboxylic acid —— C16H8Cl3NO2
6-Chloro-2-(3,4-dichlorophenyl)quinoline-4-carboxylic acid
—— 6-nitro-4-oxo-N-(pyridin-4-ylmethylideneamino)-3H-quinazoline-2-carboxamide —— C15H10N6O4
6-nitro-4-oxo-N-(pyridin-4-ylmethylideneamino)-3H-quinazoline-2-carboxamide
—— 6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C24H30FN3O4
6-(3-fluoro-4-methoxyphenyl)-2-[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— 6-[[1-(2,5-Dichlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H16Cl2N6OS
6-[[1-(2,5-Dichlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-Tert-butyl-2-(2-chlorophenyl)quinoline-4-carboxylic acid —— C20H18ClNO2
6-Tert-butyl-2-(2-chlorophenyl)quinoline-4-carboxylic acid
—— 6-[(3S,4R)-4-(4-methoxyphenyl)-1-[(3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one —— C24H30N4O4
6-[(3S,4R)-4-(4-methoxyphenyl)-1-[(3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one
—— 6-ethyl-6-methyl-4-(4-methylpiperidin-1-yl)-2-(methylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine —— C19H27N3OS2
6-ethyl-6-methyl-4-(4-methylpiperidin-1-yl)-2-(methylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine
—— 6-(4-Bromophenyl)sulfonyl-2-methyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C14H14BrN3O3S
6-(4-Bromophenyl)sulfonyl-2-methyl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[(2S)-2-phenylpropyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one —— C26H31N3O3
6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[(2S)-2-phenylpropyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl (3R)-3-acetamido-3-thiophen-2-ylpropanoate —— C21H21NO5S
(6,7-dimethyl-2-oxochromen-4-yl)methyl (3R)-3-acetamido-3-thiophen-2-ylpropanoate
—— 6-methylheptyl (3R)-1,1-dioxothiolane-3-sulfonate —— C12H24O5S2
6-methylheptyl (3R)-1,1-dioxothiolane-3-sulfonate
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (3R)-3-acetamido-3-thiophen-2-ylpropanoate —— C18H18N2O7S
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (3R)-3-acetamido-3-thiophen-2-ylpropanoate
—— 6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[[(3R)-oxolan-3-yl]methyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one —— C22H29N3O4
6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[[(3R)-oxolan-3-yl]methyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one
—— 6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[[(3S)-oxolan-3-yl]methyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one —— C22H29N3O4
6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[[(3S)-oxolan-3-yl]methyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(1-methyl-6-oxopyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H25N5O3
6-ethyl-5-methyl-2-[(2R)-1-(1-methyl-6-oxopyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[(2R)-2-phenylpropyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one —— C26H31N3O3
6-[(3S,4R)-4-(3,4-dimethoxyphenyl)-1-[(2R)-2-phenylpropyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[3-(1,2-oxazol-5-yl)propanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H25N5O3
6-ethyl-5-methyl-2-[(2R)-1-[3-(1,2-oxazol-5-yl)propanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H22N6O2S
6-ethyl-5-methyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[(3S)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H26N4O3
6-ethyl-5-methyl-2-[(2S)-1-[(3S)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23N5O2
6-ethyl-5-methyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-fluoro-5-methyl-2-[(2S)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H21FN6O3
6-fluoro-5-methyl-2-[(2S)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H22N6O2S
6-ethyl-5-methyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H26N4O3
6-ethyl-5-methyl-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23N5O2
6-ethyl-5-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N6O2
6-ethyl-5-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(1,3-thiazole-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H21N5O2S
6-ethyl-5-methyl-2-[(2S)-1-(1,3-thiazole-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H31N5O3
6-ethyl-5-methyl-2-[(2R)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-fluoro-5-methyl-2-[(2R)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H21FN6O3
6-fluoro-5-methyl-2-[(2R)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(1-methyl-6-oxopyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H25N5O3
6-ethyl-5-methyl-2-[(2S)-1-(1-methyl-6-oxopyridine-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H24N6O2
6-ethyl-5-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(1-methylsulfonylpiperidine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H31N5O4S
6-ethyl-5-methyl-2-[(2R)-1-(1-methylsulfonylpiperidine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H24N6O2
6-ethyl-5-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-fluoro-5-methyl-2-[(2R)-1-[2-(4-methylsulfonylphenyl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23FN4O4S
6-fluoro-5-methyl-2-[(2R)-1-[2-(4-methylsulfonylphenyl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H24N6O3
6-ethyl-5-methyl-2-[(2S)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[(3S)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H26N4O3
6-ethyl-5-methyl-2-[(2R)-1-[(3S)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23N5O2
6-ethyl-5-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H24N6O3
6-ethyl-5-methyl-2-[(2R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N6O2
6-ethyl-5-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[2-(3,5-ditert-butyl-4-hydroxyphenyl)ethenyl]-5-nitro-1H-pyrimidine-2,4-dione —— C20H25N3O5
6-[2-(3,5-ditert-butyl-4-hydroxyphenyl)ethenyl]-5-nitro-1H-pyrimidine-2,4-dione
—— 6-ethyl-5-methyl-2-[(2R)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H23N5O3
6-ethyl-5-methyl-2-[(2R)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N6O3
6-ethyl-5-methyl-2-[(2S)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H23N5O3
6-ethyl-5-methyl-2-[(2S)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[(3R)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H26N4O3
6-ethyl-5-methyl-2-[(2S)-1-[(3R)-oxolane-3-carbonyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one