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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-ethyl-5-methyl-2-[(2S)-1-[2-(1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H21N7O2
6-ethyl-5-methyl-2-[(2S)-1-[2-(1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H29N5O3
6-ethyl-5-methyl-2-[(2R)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H29N5O3
6-ethyl-5-methyl-2-[(2S)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23N5O2
6-ethyl-5-methyl-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[(2R)-2-(1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H23N7O2
6-ethyl-5-methyl-2-[(2S)-1-[(2R)-2-(1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(2S)-2-(4-ethoxyphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O4
6-[(2S)-2-(4-ethoxyphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-bromophenyl)-3-phenyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazine —— C17H12BrN3S
6-(4-bromophenyl)-3-phenyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazine
—— 6-Amino-4-(5-bromo-2-fluorophenyl)-3-methyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C14H10BrFN4O
6-Amino-4-(5-bromo-2-fluorophenyl)-3-methyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-Bromo-3-[(2-methoxyphenyl)carbamoyl]-2-methylquinoline-4-carboxylic acid —— C19H15BrN2O4
6-Bromo-3-[(2-methoxyphenyl)carbamoyl]-2-methylquinoline-4-carboxylic acid
—— (6-Chloropyridin-3-yl)-[4-hydroxy-4-(pyrrolo[2,3-c]pyridin-1-ylmethyl)piperidin-1-yl]methanone —— C19H19ClN4O2
(6-Chloropyridin-3-yl)-[4-hydroxy-4-(pyrrolo[2,3-c]pyridin-1-ylmethyl)piperidin-1-yl]methanone
—— 6-[2-(3-Methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H19N5O2
6-[2-(3-Methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(2-Methoxy-4-methylphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O4
6-[2-(2-Methoxy-4-methylphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Azepan-1-yl)-5-nitro-2-(pyrrolidin-1-yl)pyrimidin-4-amine —— C14H22N6O2
6-(Azepan-1-yl)-5-nitro-2-(pyrrolidin-1-yl)pyrimidin-4-amine
—— 6-[2-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]ethenyl]-5-nitro-1H-pyrimidine-2,4-dione —— C19H18N4O4
6-[2-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]ethenyl]-5-nitro-1H-pyrimidine-2,4-dione
—— 6-[[4-[2-(2,6-Dimethylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H24N4O3S
6-[[4-[2-(2,6-Dimethylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(2R)-2-(4-ethoxyphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O4
6-[(2R)-2-(4-ethoxyphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6,7-dimethoxy-2-[[1-(6-methoxypyridin-3-yl)pyrrol-2-yl]methyl]-3,4-dihydro-1H-isoquinoline —— C22H25N3O3
6,7-dimethoxy-2-[[1-(6-methoxypyridin-3-yl)pyrrol-2-yl]methyl]-3,4-dihydro-1H-isoquinoline
—— 6-amino-N-[2-(2,4-dichlorophenyl)ethyl]-N-[(3,4-dimethoxyphenyl)methyl]hexanamide —— C23H30Cl2N2O3
6-amino-N-[2-(2,4-dichlorophenyl)ethyl]-N-[(3,4-dimethoxyphenyl)methyl]hexanamide
—— 6-[(2,5-Dimethoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C13H11N3O3S
6-[(2,5-Dimethoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-[2-(4-Methylphenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O2
6-[2-(4-Methylphenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(2-Ethoxy-4-methylphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O4
6-[2-(2-Ethoxy-4-methylphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(4-Methoxyphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H19N5O4
6-[2-(4-Methoxyphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3S)-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-3-yl]quinoline-3-carboxamide —— C21H23FN4O3
6-fluoro-2-[(3S)-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-[2-(2-Fluorophenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H16FN5O3
6-[2-(2-Fluorophenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2S)-2-(4-methylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O3
6-[(2S)-2-(4-methylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(2-Fluorophenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H16FN5O2
6-[2-(2-Fluorophenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3R)-1-(5-methylthiophene-3-carbonyl)piperidin-3-yl]quinoline-3-carboxamide —— C21H20FN3O2S
6-fluoro-2-[(3R)-1-(5-methylthiophene-3-carbonyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-[4-(2-Fluorophenoxy)butanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H20FN5O3
6-[4-(2-Fluorophenoxy)butanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(4-Methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H19N5O2
6-[2-(4-Methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2R)-2-(4-methylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O3
6-[(2R)-2-(4-methylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(2-Methyl-1,3-thiazol-4-yl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C17H16N6O2S
6-[2-(2-Methyl-1,3-thiazol-4-yl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3S)-1-[2-(4-methylpyrazol-1-yl)acetyl]piperidin-3-yl]quinoline-3-carboxamide —— C21H22FN5O2
6-fluoro-2-[(3S)-1-[2-(4-methylpyrazol-1-yl)acetyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-[2-(4-Methoxyphenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O3
6-[2-(4-Methoxyphenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3S)-1-[3-(pyridine-3-carbonylamino)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C24H24FN5O3
6-fluoro-2-[(3S)-1-[3-(pyridine-3-carbonylamino)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-[2-(4-Methoxy-3-methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O3
6-[2-(4-Methoxy-3-methylphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3S)-1-(2-pyridin-3-yloxyacetyl)piperidin-3-yl]quinoline-3-carboxamide —— C22H21FN4O3
6-fluoro-2-[(3S)-1-(2-pyridin-3-yloxyacetyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3S)-1-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]piperidin-3-yl]quinoline-3-carboxamide —— C23H26FN5O2
6-fluoro-2-[(3S)-1-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-[2-[[(2R)-oxan-2-yl]methoxy]acetyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H23N5O4
6-[2-[[(2R)-oxan-2-yl]methoxy]acetyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3R)-1-(3-pyridin-3-ylpropanoyl)piperidin-3-yl]quinoline-3-carboxamide —— C23H23FN4O2
6-fluoro-2-[(3R)-1-(3-pyridin-3-ylpropanoyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-[2-(4-Ethoxyphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O3
6-[2-(4-Ethoxyphenyl)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(2-Methoxyphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H19N5O4
6-[2-(2-Methoxyphenoxy)acetyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2R)-2-(3,5-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2R)-2-(3,5-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2S)-2-(3,5-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2S)-2-(3,5-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3S)-1-[2-(4-methylphenyl)acetyl]piperidin-3-yl]quinoline-3-carboxamide —— C24H24FN3O2
6-fluoro-2-[(3S)-1-[2-(4-methylphenyl)acetyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-[[3-Chloro-4-[(2-chlorophenyl)methoxy]-5-ethoxyphenyl]methylidene]-2-cyclohexyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H26Cl2N4O3S
6-[[3-Chloro-4-[(2-chlorophenyl)methoxy]-5-ethoxyphenyl]methylidene]-2-cyclohexyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-fluoro-2-[(3S)-1-[(2R)-2-(4-methylphenoxy)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C25H26FN3O3
6-fluoro-2-[(3S)-1-[(2R)-2-(4-methylphenoxy)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3S)-1-[3-(4-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C22H24FN5O2
6-fluoro-2-[(3S)-1-[3-(4-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3R)-1-[3-(pyridine-3-carbonylamino)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C24H24FN5O3
6-fluoro-2-[(3R)-1-[3-(pyridine-3-carbonylamino)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3R)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]quinoline-3-carboxamide —— C20H20FN5O2
6-fluoro-2-[(3R)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3S)-1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]quinoline-3-carboxamide —— C21H20FN5O2
6-fluoro-2-[(3S)-1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]quinoline-3-carboxamide