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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(3S)-1-[2-(3-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C21H20FN3O2
6-[(3S)-1-[2-(3-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-cyclohexyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-cyclohexyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25FN4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-chlorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H21ClN4
6-[(3-chlorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(cyclohexylmethyl)-2-[(2S)-1-(3-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-(cyclohexylmethyl)-2-[(2S)-1-(3-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(3-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27FN4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(3-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-cyclohexyl-2-[(3S)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H29FN4O2
6-cyclohexyl-2-[(3S)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(3-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27FN4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(3-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-1-[2-(3-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C21H20FN3O2
6-[(3R)-1-[2-(3-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-cyclopentyl-2-[(3R)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H27FN4O2
6-cyclopentyl-2-[(3R)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[(3-chlorophenyl)methyl]piperidin-4-yl]-5H-pyrrolo[2,3-b]pyrazine —— C18H19ClN4
6-[1-[(3-chlorophenyl)methyl]piperidin-4-yl]-5H-pyrrolo[2,3-b]pyrazine
—— 6-(cyclohexylmethyl)-2-[(2R)-1-(3-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-(cyclohexylmethyl)-2-[(2R)-1-(3-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-chlorophenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H23ClN4
6-[(3-chlorophenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(Azepan-1-ylsulfonyl)-2-(4-ethylphenyl)quinoline-4-carboxylic acid —— C24H26N2O4S
6-(Azepan-1-ylsulfonyl)-2-(4-ethylphenyl)quinoline-4-carboxylic acid
—— 6-[(3-chlorophenyl)methyl]-2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H23ClN4
6-[(3-chlorophenyl)methyl]-2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(cyclohexanecarbonyl)-2-[(2R)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N6O3
6-(cyclohexanecarbonyl)-2-[(2R)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H22Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H22Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(3R)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-Tert-butyl-2-(6-methoxy-1-benzofuran-2-yl)quinoline-4-carboxylic acid —— C23H21NO4
6-Tert-butyl-2-(6-methoxy-1-benzofuran-2-yl)quinoline-4-carboxylic acid
—— 6-[(3,4-Difluorophenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H15F2N5O
6-[(3,4-Difluorophenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C20H19F2N5O
6-[(3R)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(3R)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H26F2N4O2
6-(cyclopropanecarbonyl)-2-[(3R)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-chloro-3-fluorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20ClFN4
6-[(4-chloro-3-fluorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(4-chloro-3-fluorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20ClFN4
6-[(4-chloro-3-fluorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(3-chlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H21ClN4
6-[(3-chlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(cyclopropanecarbonyl)-2-[(3S)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H26F2N4O2
6-(cyclopropanecarbonyl)-2-[(3S)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H22Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(3S)-piperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-methyl-4-(2-methylphenyl)-2-oxo-N-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide —— C20H18F3N3O2
6-methyl-4-(2-methylphenyl)-2-oxo-N-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
—— 6-cyclopentyl-2-[(3R)-1-[2-(2,5-difluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28F2N4O2
6-cyclopentyl-2-[(3R)-1-[2-(2,5-difluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(3S)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H26F2N4O2
6-(cyclopropanecarbonyl)-2-[(3S)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(3-Morpholin-4-ylpropyl)-4,13,16-trioxa-2,6-diazatetracyclo[8.8.0.03,8.012,17]octadeca-1,3(8),9,11,17-pentaen-5-one —— C20H23N3O5
6-(3-Morpholin-4-ylpropyl)-4,13,16-trioxa-2,6-diazatetracyclo[8.8.0.03,8.012,17]octadeca-1,3(8),9,11,17-pentaen-5-one
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(2-cyclohexylacetyl)-2-[(2R)-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N6O3
6-(2-cyclohexylacetyl)-2-[(2R)-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-Morpholin-4-ylethyl)-4,13,15-trioxa-2,6-diazatetracyclo[8.7.0.03,8.012,16]heptadeca-1,3(8),9,11,16-pentaen-5-one —— C18H19N3O5
6-(2-Morpholin-4-ylethyl)-4,13,15-trioxa-2,6-diazatetracyclo[8.7.0.03,8.012,16]heptadeca-1,3(8),9,11,16-pentaen-5-one
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H22Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H24F2N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-8-[(2,6-dichlorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one —— C17H15Cl2N3O
(6R)-8-[(2,6-dichlorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H24F2N4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2,3-dichlorophenyl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(2,3-dichlorophenyl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(2-Phenylmethoxyphenyl)-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline —— C24H23NO3
6-(2-Phenylmethoxyphenyl)-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline
—— 6-(2-cyclohexylacetyl)-2-[(2S)-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N6O3
6-(2-cyclohexylacetyl)-2-[(2S)-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2,3-dichlorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(2,3-dichlorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(3S)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C20H19F2N5O
6-[(3S)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— (6S)-8-[(2-chloro-6-fluorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one —— C17H15ClFN3O
(6S)-8-[(2-chloro-6-fluorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one
—— 6-(cyclohexanecarbonyl)-2-[(2S)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N6O3
6-(cyclohexanecarbonyl)-2-[(2S)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-8-[(2,6-dichlorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one —— C17H15Cl2N3O
(6S)-8-[(2,6-dichlorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one
—— 6-[(3R)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C20H19F2N5O
6-[(3R)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-[(2,3-dichlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(2,3-dichlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(cyclopropanecarbonyl)-2-[(3R)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H26F2N4O2
6-(cyclopropanecarbonyl)-2-[(3R)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one