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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-Amino-4-[4-[(2-chloro-6-fluorophenyl)methoxy]phenyl]-3-(trifluoromethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C21H13ClF4N4O2
6-Amino-4-[4-[(2-chloro-6-fluorophenyl)methoxy]phenyl]-3-(trifluoromethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C25H28N4O2
(6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2S
(6S)-1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(1-methylimidazole-4-carbonyl)-1,4-diazepan-5-one —— C26H30N4O3
(6R)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(1-methylimidazole-4-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-benzoyl-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C28H30N2O3
(6S)-1-benzoyl-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(3-pyrazol-1-ylpropanoyl)-1,4-diazepan-5-one —— C26H30N4O2
(6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(3-pyrazol-1-ylpropanoyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[3-[(2R)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one —— C28H36N2O3
(6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[3-[(2R)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2S)-2-(5-methylpyrazol-1-yl)propanoyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H32N4O2
(6R)-4-ethyl-1-[(2S)-2-(5-methylpyrazol-1-yl)propanoyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(5-oxo-1,2-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one —— C24H27N5O3
(6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(5-oxo-1,2-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(4-methylthiadiazole-5-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H24N4O2S2
(6R)-4-ethyl-1-(4-methylthiadiazole-5-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3,3-dimethylbutanoyl)-4-ethyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H33N3O2
(6S)-1-(3,3-dimethylbutanoyl)-4-ethyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(pyridine-2-carbonyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N4O2
(6S)-4-ethyl-1-(pyridine-2-carbonyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H32N2O3S
(6S)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopropylmethyl)-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H29N3O
(6S)-1-(cyclopropylmethyl)-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[(4-phenylphenyl)methyl]-1-(3-pyridin-4-ylpropanoyl)-1,4-diazepan-5-one —— C28H31N3O2
(6S)-4-ethyl-6-[(4-phenylphenyl)methyl]-1-(3-pyridin-4-ylpropanoyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one —— C26H30N4O2
(6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1-methylimidazole-4-carbonyl)-1,4-diazepan-5-one —— C25H27FN4O2
(6S)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1-methylimidazole-4-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H25N5O3
(6R)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H28FN3O3
(6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one —— C24H27N5O3
(6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(6-oxo-1H-pyridazine-3-carbonyl)-1,4-diazepan-5-one —— C26H28N4O3
(6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(6-oxo-1H-pyridazine-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H30N4O2
(6S)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one —— C25H27FN4O2
(6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H34N2O3
(6S)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(6-oxo-1H-pyridazine-3-carbonyl)-1,4-diazepan-5-one —— C25H25FN4O3
(6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(6-oxo-1H-pyridazine-3-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1-methylimidazole-2-carbonyl)-1,4-diazepan-5-one —— C25H27FN4O2
(6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1-methylimidazole-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2
(6R)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(1R)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N3O2
(6R)-1-[(1R)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O3
(6R)-4-ethyl-1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H34N2O3
(6S)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-bromo-N-(2-fluorophenyl)-2-imino-2H-chromene-3-carboxamide —— C16H10BrFN2O2
6-bromo-N-(2-fluorophenyl)-2-imino-2H-chromene-3-carboxamide
—— (6R)-4-ethyl-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6R)-4-ethyl-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(1R)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N3O2
(6S)-1-[(1R)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2R)-2-piperidin-1-ylpropanoyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H36N4O2
(6R)-4-ethyl-1-[(2R)-2-piperidin-1-ylpropanoyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H34N2O3
(6R)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one —— C28H36N2O3
(6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2S)-2-piperidin-1-ylpropanoyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H36N4O2
(6R)-4-ethyl-1-[(2S)-2-piperidin-1-ylpropanoyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O3
(6S)-4-ethyl-1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(1S)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N3O2
(6S)-1-[(1S)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2
(6S)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C24H25FN4O2
(6S)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C24H25FN4O2
(6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one —— C24H27N5O3
(6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6S)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H25N5O3
(6S)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-Amino-4-(2-chloro-6-fluorophenyl)-1,3-dimethyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C15H12ClFN4O
6-Amino-4-(2-chloro-6-fluorophenyl)-1,3-dimethyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (6S)-4-ethyl-6-[(4-phenylphenyl)methyl]-1-(2-pyrazol-1-ylacetyl)-1,4-diazepan-5-one —— C25H28N4O2
(6S)-4-ethyl-6-[(4-phenylphenyl)methyl]-1-(2-pyrazol-1-ylacetyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H34N2O3
(6R)-4-ethyl-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H27N5O2
(6R)-4-ethyl-1-(2-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H28FN3O3
(6S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one