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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R)-3-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]propan-1-one —— C21H24FN5O2
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R)-3-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]propan-1-one
—— 1-[(2R)-1-methoxypropan-2-yl]-2-methyl-3-[2-(1-phenylpyrazol-4-yl)ethyl]guanidine —— C17H25N5O
1-[(2R)-1-methoxypropan-2-yl]-2-methyl-3-[2-(1-phenylpyrazol-4-yl)ethyl]guanidine
—— (2R)-N-[4-(3-amino-4-cyanopyrazol-1-yl)phenyl]oxolane-2-carboxamide —— C15H15N5O2
(2R)-N-[4-(3-amino-4-cyanopyrazol-1-yl)phenyl]oxolane-2-carboxamide
—— [(2R)-2-[(2-chloro-6-fluorophenyl)methyl]pyrrolidin-1-yl]-(1,3-dimethylpyrazol-4-yl)methanone —— C17H19ClFN3O
[(2R)-2-[(2-chloro-6-fluorophenyl)methyl]pyrrolidin-1-yl]-(1,3-dimethylpyrazol-4-yl)methanone
—— 5-[(3S)-oxolan-3-yl]-3-(propan-2-yloxymethyl)-1,2,4-oxadiazole —— C10H16N2O3
5-[(3S)-oxolan-3-yl]-3-(propan-2-yloxymethyl)-1,2,4-oxadiazole
—— ethyl 5-methyl-1-[4-[(7R)-5-oxo-7-(trifluoromethyl)-1,4-diazepane-1-carbonyl]phenyl]pyrazole-4-carboxylate —— C20H21F3N4O4
ethyl 5-methyl-1-[4-[(7R)-5-oxo-7-(trifluoromethyl)-1,4-diazepane-1-carbonyl]phenyl]pyrazole-4-carboxylate
—— N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2S)-oxolan-2-yl]methoxy]acetamide —— C16H27N3O3
N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2S)-oxolan-2-yl]methoxy]acetamide
—— [2-[(2,5-Diphenylpyrazol-3-yl)amino]-2-oxoethyl] 2-fluorobenzoate —— C24H18FN3O3
[2-[(2,5-Diphenylpyrazol-3-yl)amino]-2-oxoethyl] 2-fluorobenzoate
—— ethyl 5-methyl-1-[4-[(7S)-5-oxo-7-(trifluoromethyl)-1,4-diazepane-1-carbonyl]phenyl]pyrazole-4-carboxylate —— C20H21F3N4O4
ethyl 5-methyl-1-[4-[(7S)-5-oxo-7-(trifluoromethyl)-1,4-diazepane-1-carbonyl]phenyl]pyrazole-4-carboxylate
—— (3R)-N-[3-(1H-pyrazol-5-yl)phenyl]-2,3-dihydro-1-benzofuran-3-carboxamide —— C18H15N3O2
(3R)-N-[3-(1H-pyrazol-5-yl)phenyl]-2,3-dihydro-1-benzofuran-3-carboxamide
—— N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2R)-oxolan-2-yl]methoxy]acetamide —— C16H27N3O3
N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2R)-oxolan-2-yl]methoxy]acetamide
—— N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2S)-oxolan-2-yl]methoxy]acetamide —— C16H27N3O3
N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2S)-oxolan-2-yl]methoxy]acetamide
—— (3S)-N-[3-(1H-pyrazol-5-yl)phenyl]-2,3-dihydro-1-benzofuran-3-carboxamide —— C18H15N3O2
(3S)-N-[3-(1H-pyrazol-5-yl)phenyl]-2,3-dihydro-1-benzofuran-3-carboxamide
—— 2-[2-(4-fluorophenyl)-1,3-oxazol-4-yl]-N-methylacetamide —— C12H11FN2O2
2-[2-(4-fluorophenyl)-1,3-oxazol-4-yl]-N-methylacetamide
—— [(2S)-2-[(2-chloro-6-fluorophenyl)methyl]pyrrolidin-1-yl]-(1,3-dimethylpyrazol-4-yl)methanone —— C17H19ClFN3O
[(2S)-2-[(2-chloro-6-fluorophenyl)methyl]pyrrolidin-1-yl]-(1,3-dimethylpyrazol-4-yl)methanone
—— N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2R)-oxolan-2-yl]methoxy]acetamide —— C16H27N3O3
N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-[[(2R)-oxolan-2-yl]methoxy]acetamide
—— (2S)-N-[4-(3-amino-4-cyanopyrazol-1-yl)phenyl]oxolane-2-carboxamide —— C15H15N5O2
(2S)-N-[4-(3-amino-4-cyanopyrazol-1-yl)phenyl]oxolane-2-carboxamide
—— (6R)-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one —— C14H18N2O2S
(6R)-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one
—— 2-[[4,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]imidazol-2-yl]sulfanylmethyl]-5-propan-2-yl-1,3-oxazole —— C17H25N3O2S
2-[[4,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]imidazol-2-yl]sulfanylmethyl]-5-propan-2-yl-1,3-oxazole
—— 2-[(1R,2S)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide —— C16H21N3O3S
2-[(1R,2S)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide
—— 2-[[4,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]imidazol-2-yl]sulfanylmethyl]-5-propan-2-yl-1,3-oxazole —— C17H25N3O2S
2-[[4,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]imidazol-2-yl]sulfanylmethyl]-5-propan-2-yl-1,3-oxazole
—— [(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (E)-3-(furan-2-yl)prop-2-enoate —— C21H21N3O5
[(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (E)-3-(furan-2-yl)prop-2-enoate
—— (3S)-N-[2-(1-phenylpyrazol-3-yl)ethyl]-2,3-dihydro-1-benzofuran-3-carboxamide —— C20H19N3O2
(3S)-N-[2-(1-phenylpyrazol-3-yl)ethyl]-2,3-dihydro-1-benzofuran-3-carboxamide
—— [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 3-(trifluoromethyl)benzoate —— C21H18F3N3O3
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 3-(trifluoromethyl)benzoate
—— 2-[(1S,2R)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide —— C16H21N3O3S
2-[(1S,2R)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide
—— 2-[(1S,2S)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide —— C16H21N3O3S
2-[(1S,2S)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide
—— N-[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]-2-[[(2R)-oxolan-2-yl]methylsulfanyl]acetamide —— C16H24N2O2S2
N-[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]-2-[[(2R)-oxolan-2-yl]methylsulfanyl]acetamide
—— 2-[(1R,3S)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide —— C15H22F3N3O2
2-[(1R,3S)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide
—— 5-(hydroxymethyl)-2-methyl-4-[[3-(tetrazol-1-yl)anilino]methylidene]pyridin-3-one —— C15H14N6O2
5-(hydroxymethyl)-2-methyl-4-[[3-(tetrazol-1-yl)anilino]methylidene]pyridin-3-one
—— 2-[(1S,3S)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide —— C15H22F3N3O2
2-[(1S,3S)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide
—— (6S)-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one —— C14H18N2O2S
(6S)-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one
—— (3R)-N-[2-(1-phenylpyrazol-3-yl)ethyl]-2,3-dihydro-1-benzofuran-3-carboxamide —— C20H19N3O2
(3R)-N-[2-(1-phenylpyrazol-3-yl)ethyl]-2,3-dihydro-1-benzofuran-3-carboxamide
—— 5-(hydroxymethyl)-2-methyl-4-[[4-(tetrazol-1-yl)anilino]methylidene]pyridin-3-one —— C15H14N6O2
5-(hydroxymethyl)-2-methyl-4-[[4-(tetrazol-1-yl)anilino]methylidene]pyridin-3-one
—— 2-[(1R,2R)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide —— C16H21N3O3S
2-[(1R,2R)-2-methylcyclohexyl]oxy-N-[(5-thiophen-3-yl-1,2,4-oxadiazol-3-yl)methyl]acetamide
—— 2-[(1R,3R)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide —— C15H22F3N3O2
2-[(1R,3R)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide
—— 2-[(1S,3R)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide —— C15H22F3N3O2
2-[(1S,3R)-3-methylcyclohexyl]oxy-N-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]acetamide
—— [(2R)-2-cyano-3-(furan-2-yl)propyl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate —— C15H17N3O4
[(2R)-2-cyano-3-(furan-2-yl)propyl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate
—— [(3S)-thian-3-yl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate —— C12H18N2O3S
[(3S)-thian-3-yl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate
—— [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 5-methylthiophene-2-carboxylate —— C19H19N3O3S
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 5-methylthiophene-2-carboxylate
—— [(3R)-thian-3-yl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate —— C12H18N2O3S
[(3R)-thian-3-yl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate
—— 1-[3-(3-methylpyrazol-1-yl)phenyl]-3-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea —— C16H19N7O
1-[3-(3-methylpyrazol-1-yl)phenyl]-3-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea
—— 1-[3-(3-methylpyrazol-1-yl)phenyl]-3-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea —— C16H19N7O
1-[3-(3-methylpyrazol-1-yl)phenyl]-3-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea
—— N-[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]-2-[[(2S)-oxolan-2-yl]methylsulfanyl]acetamide —— C16H24N2O2S2
N-[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]-2-[[(2S)-oxolan-2-yl]methylsulfanyl]acetamide
—— [(2S)-2-cyano-3-(furan-2-yl)propyl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate —— C15H17N3O4
[(2S)-2-cyano-3-(furan-2-yl)propyl] 5-methoxy-1,3-dimethylpyrazole-4-carboxylate
—— N-[(R)-cyclohexyl(pyridin-3-yl)methyl]-5-methyl-1H-pyrazole-4-carboxamide —— C17H22N4O
N-[(R)-cyclohexyl(pyridin-3-yl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
—— N-[(R)-(2,5-difluorophenyl)-pyridin-4-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide —— C17H14F2N4O
N-[(R)-(2,5-difluorophenyl)-pyridin-4-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide
—— N-[(S)-(4-fluorophenyl)-pyridin-2-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide —— C17H15FN4O
N-[(S)-(4-fluorophenyl)-pyridin-2-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide
—— N-[(1S)-2-(diethylamino)-1-phenylethyl]-5-methyl-1H-pyrazole-4-carboxamide —— C17H24N4O
N-[(1S)-2-(diethylamino)-1-phenylethyl]-5-methyl-1H-pyrazole-4-carboxamide
—— N-[(S)-(2,5-difluorophenyl)-pyridin-4-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide —— C17H14F2N4O
N-[(S)-(2,5-difluorophenyl)-pyridin-4-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide
—— N-[(S)-(4-chlorophenyl)-pyridin-2-ylmethyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide —— C18H17ClN4O
N-[(S)-(4-chlorophenyl)-pyridin-2-ylmethyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide