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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[(2S,5S)-5-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazolidin-2-yl]-N,N-dimethylaniline —— C22H27N5O2S
4-[(2S,5S)-5-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazolidin-2-yl]-N,N-dimethylaniline
—— [2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] (E)-3-thiophen-3-ylprop-2-enoate —— C22H23N3O3S
[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] (E)-3-thiophen-3-ylprop-2-enoate
—— 1-[2-(5-methyl-1,3-thiazol-2-yl)propan-2-yl]-3-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)propyl]urea —— C17H27N5OS
1-[2-(5-methyl-1,3-thiazol-2-yl)propan-2-yl]-3-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)propyl]urea
—— (4S)-6-amino-3-(4-ethoxyphenyl)-4-(3-hydroxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C21H18N4O3
(4S)-6-amino-3-(4-ethoxyphenyl)-4-(3-hydroxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— N,N-dimethyl-4-[(2R,5S)-5-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]aniline —— C22H28N5OS+
N,N-dimethyl-4-[(2R,5S)-5-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]aniline
—— [2-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl] (E)-3-thiophen-3-ylprop-2-enoate —— C20H19N3O4S
[2-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl] (E)-3-thiophen-3-ylprop-2-enoate
—— [2-[[(2S)-3-methylbutan-2-yl]amino]-2-oxoethyl] 3,5-dimethyl-1,2-oxazole-4-carboxylate —— C13H20N2O4
[2-[[(2S)-3-methylbutan-2-yl]amino]-2-oxoethyl] 3,5-dimethyl-1,2-oxazole-4-carboxylate
—— (2S)-N-[4-(cyanomethyl)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide —— C23H23N5O
(2S)-N-[4-(cyanomethyl)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide
—— N-[(R)-(4-chlorophenyl)-cyanomethyl]-4-(2-methyl-1,3-thiazol-4-yl)butanamide —— C16H16ClN3OS
N-[(R)-(4-chlorophenyl)-cyanomethyl]-4-(2-methyl-1,3-thiazol-4-yl)butanamide
—— 4-[(2S,5R)-5-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]-N,N-dimethylaniline —— C22H28N5OS+
4-[(2S,5R)-5-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]-N,N-dimethylaniline
—— (2S)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)-N-(3-prop-2-enoxyphenyl)pyrrolidine-1-carboxamide —— C24H26N4O2
(2S)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)-N-(3-prop-2-enoxyphenyl)pyrrolidine-1-carboxamide
—— (2S)-N-[4-(cyclopropanecarbonylamino)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide —— C25H27N5O2
(2S)-N-[4-(cyclopropanecarbonylamino)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide
—— N-tert-butyl-2-[[4-(furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C20H24N4O2S
N-tert-butyl-2-[[4-(furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2R)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)-N-(3-prop-2-enoxyphenyl)pyrrolidine-1-carboxamide —— C24H26N4O2
(2R)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)-N-(3-prop-2-enoxyphenyl)pyrrolidine-1-carboxamide
—— 4-[(2S,5S)-5-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-2-yl]-N,N-dimethylaniline —— C22H27N5OS
4-[(2S,5S)-5-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-2-yl]-N,N-dimethylaniline
—— (2R)-N-[4-(cyclopropanecarbonylamino)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide —— C25H27N5O2
(2R)-N-[4-(cyclopropanecarbonylamino)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide
—— N,N-dimethyl-4-[(2S,5R)-5-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-2-yl]aniline —— C23H27N5OS
N,N-dimethyl-4-[(2S,5R)-5-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-2-yl]aniline
—— N,N-dimethyl-4-[(2S,5S)-5-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]aniline —— C23H28N5OS+
N,N-dimethyl-4-[(2S,5S)-5-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]aniline
—— N,N-dimethyl-4-[(2S,5R)-5-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]aniline —— C23H28N5OS+
N,N-dimethyl-4-[(2S,5R)-5-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazolidin-3-ium-2-yl]aniline
—— N-[(S)-(4-chlorophenyl)-cyanomethyl]-4-(2-methyl-1,3-thiazol-4-yl)butanamide —— C16H16ClN3OS
N-[(S)-(4-chlorophenyl)-cyanomethyl]-4-(2-methyl-1,3-thiazol-4-yl)butanamide
—— 5-(3-chloro-4-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide —— C11H9ClFN3O
5-(3-chloro-4-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
—— (2R)-3-(cyclopropylmethyl)-2-[4-(1,2,4-triazol-1-yl)phenyl]-1,3-diazaspiro[4.4]nonan-4-one —— C19H23N5O
(2R)-3-(cyclopropylmethyl)-2-[4-(1,2,4-triazol-1-yl)phenyl]-1,3-diazaspiro[4.4]nonan-4-one
—— 1-cyclopropyl-3-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-1-propan-2-ylurea —— C15H23N3OS
1-cyclopropyl-3-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-1-propan-2-ylurea
—— 1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2S,3S)-2-propan-2-yloxolan-3-yl]methyl]urea —— C15H25N3O2S
1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2S,3S)-2-propan-2-yloxolan-3-yl]methyl]urea
—— (4S)-6-amino-4-(2-chloro-6-fluorophenyl)-3-(3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C20H14ClFN4O2
(4S)-6-amino-4-(2-chloro-6-fluorophenyl)-3-(3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (2S)-3-(cyclopropylmethyl)-2-[4-(1,2,4-triazol-1-yl)phenyl]-1,3-diazaspiro[4.4]nonan-4-one —— C19H23N5O
(2S)-3-(cyclopropylmethyl)-2-[4-(1,2,4-triazol-1-yl)phenyl]-1,3-diazaspiro[4.4]nonan-4-one
—— [2-[[3,5-Dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 3,5-dimethyl-1,2-oxazole-4-carboxylate —— C20H22N4O4
[2-[[3,5-Dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 3,5-dimethyl-1,2-oxazole-4-carboxylate
—— 1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2S,3R)-2-propan-2-yloxolan-3-yl]methyl]urea —— C15H25N3O2S
1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2S,3R)-2-propan-2-yloxolan-3-yl]methyl]urea
—— 1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2R,3S)-2-propan-2-yloxolan-3-yl]methyl]urea —— C15H25N3O2S
1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2R,3S)-2-propan-2-yloxolan-3-yl]methyl]urea
—— 1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2R,3R)-2-propan-2-yloxolan-3-yl]methyl]urea —— C15H25N3O2S
1-[(5-ethyl-1,3-thiazol-2-yl)methyl]-3-[[(2R,3R)-2-propan-2-yloxolan-3-yl]methyl]urea
—— (2S)-2-cyclopentyl-N-[(3R,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]propanamide —— C19H31N3OS
(2S)-2-cyclopentyl-N-[(3R,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]propanamide
—— (2S)-3-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylpropane-1,2-diol —— C14H17FN2O3S
(2S)-3-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylpropane-1,2-diol
—— 4-[(2S)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine —— C20H21N7
4-[(2S)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine
—— (2R)-3-[[1-(4-fluorophenyl)pyrazol-3-yl]methylsulfanyl]propane-1,2-diol —— C13H15FN2O2S
(2R)-3-[[1-(4-fluorophenyl)pyrazol-3-yl]methylsulfanyl]propane-1,2-diol
—— (2S)-3-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylpropane-1,2-diol —— C10H18N2O3S
(2S)-3-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylpropane-1,2-diol
—— 6-[(2R)-2-(1H-imidazol-2-yl)piperidin-1-yl]-3-phenyl-[1,2,4]triazolo[4,3-b]pyridazine —— C19H19N7
6-[(2R)-2-(1H-imidazol-2-yl)piperidin-1-yl]-3-phenyl-[1,2,4]triazolo[4,3-b]pyridazine
—— (2S)-2-cyclopentyl-N-[(3R,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]propanamide —— C19H31N3OS
(2S)-2-cyclopentyl-N-[(3R,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]propanamide
—— 4-[(2R)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine —— C20H21N7
4-[(2R)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]-1-phenylpyrazolo[3,4-d]pyrimidine
—— 6-[(2S)-2-(1H-imidazol-2-yl)piperidin-1-yl]-3-phenyl-[1,2,4]triazolo[4,3-b]pyridazine —— C19H19N7
6-[(2S)-2-(1H-imidazol-2-yl)piperidin-1-yl]-3-phenyl-[1,2,4]triazolo[4,3-b]pyridazine
—— 4-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyridin-2-amine —— C18H17N7O
4-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyridin-2-amine
—— N-[(S)-cyano-(1-phenylpyrazol-4-yl)methyl]-3-cyclobutylpropanamide —— C18H20N4O
N-[(S)-cyano-(1-phenylpyrazol-4-yl)methyl]-3-cyclobutylpropanamide
—— (2R)-3-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylpropane-1,2-diol —— C14H17FN2O3S
(2R)-3-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanylpropane-1,2-diol
—— (3R)-3-[[ethyl(methyl)amino]methyl]-N-[[3-(1,2,4-triazol-1-yl)phenyl]methyl]pyrrolidine-1-carboxamide —— C18H26N6O
(3R)-3-[[ethyl(methyl)amino]methyl]-N-[[3-(1,2,4-triazol-1-yl)phenyl]methyl]pyrrolidine-1-carboxamide
—— 1-methyl-3-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1-[[(3R)-oxolan-3-yl]methyl]urea —— C15H23N3O2S
1-methyl-3-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1-[[(3R)-oxolan-3-yl]methyl]urea
—— 1-(4-tert-butyl-1,3-thiazol-5-yl)-3-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea —— C13H20N6OS
1-(4-tert-butyl-1,3-thiazol-5-yl)-3-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea
—— 1-methyl-3-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1-[[(3S)-oxolan-3-yl]methyl]urea —— C15H23N3O2S
1-methyl-3-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1-[[(3S)-oxolan-3-yl]methyl]urea
—— N-[(R)-cyano-(1-phenylpyrazol-4-yl)methyl]-3-cyclobutylpropanamide —— C18H20N4O
N-[(R)-cyano-(1-phenylpyrazol-4-yl)methyl]-3-cyclobutylpropanamide
—— (2R)-1-[[3-(3,5-dichlorophenyl)-1,2,4-oxadiazol-5-yl]amino]-3-methoxypropan-2-ol —— C12H13Cl2N3O3
(2R)-1-[[3-(3,5-dichlorophenyl)-1,2,4-oxadiazol-5-yl]amino]-3-methoxypropan-2-ol
—— 1-methyl-3-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1-[[(3R)-oxolan-3-yl]methyl]urea —— C15H23N3O2S
1-methyl-3-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-1-[[(3R)-oxolan-3-yl]methyl]urea
—— 3-methyl-N-[(2S)-4-methylpentan-2-yl]sulfonyl-5-propyl-1,2-oxazole-4-carboxamide —— C14H24N2O4S
3-methyl-N-[(2S)-4-methylpentan-2-yl]sulfonyl-5-propyl-1,2-oxazole-4-carboxamide