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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-N-[3-(5-ethyl-1H-1,2,4-triazol-3-yl)phenyl]-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C19H24N6O3
(5S)-N-[3-(5-ethyl-1H-1,2,4-triazol-3-yl)phenyl]-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— (4R)-4-(hydroxymethyl)-3-[[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1,3-oxazolidin-2-one —— C16H18N2O5
(4R)-4-(hydroxymethyl)-3-[[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1,3-oxazolidin-2-one
—— [4-(3,5-Dimethyl-1-phenylpyrazole-4-carbonyl)piperazin-1-yl]-phenylmethanone —— C23H24N4O2
[4-(3,5-Dimethyl-1-phenylpyrazole-4-carbonyl)piperazin-1-yl]-phenylmethanone
—— 1,3-dimethyl-N-[(3R)-1-oxaspiro[4.5]decan-3-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine —— C15H22N4OS
1,3-dimethyl-N-[(3R)-1-oxaspiro[4.5]decan-3-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine
—— (2S)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]azetidine-2-carboxylic acid —— C15H15N3O3
(2S)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]azetidine-2-carboxylic acid
—— (2R)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]azetidine-2-carboxylic acid —— C15H15N3O3
(2R)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]azetidine-2-carboxylic acid
—— (3S)-N-[(3-methyl-2-methylsulfanylimidazol-4-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide —— C17H21N5O2S
(3S)-N-[(3-methyl-2-methylsulfanylimidazol-4-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
—— 1-tert-butyl-5-[(2R)-1-pyrazol-1-ylpropan-2-yl]-3-(thiophen-2-ylmethyl)-1,2,4-triazole —— C17H23N5S
1-tert-butyl-5-[(2R)-1-pyrazol-1-ylpropan-2-yl]-3-(thiophen-2-ylmethyl)-1,2,4-triazole
—— 3-[(3S)-3-(1-butylimidazol-2-yl)piperidin-1-yl]-5-phenyl-1,2,4-oxadiazole —— C20H25N5O
3-[(3S)-3-(1-butylimidazol-2-yl)piperidin-1-yl]-5-phenyl-1,2,4-oxadiazole
—— (3R)-N-[(3-methyl-2-methylsulfanylimidazol-4-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide —— C17H21N5O2S
(3R)-N-[(3-methyl-2-methylsulfanylimidazol-4-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
—— (2R)-2-(pyrrolidin-1-ylmethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide —— C18H25N7O
(2R)-2-(pyrrolidin-1-ylmethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide
—— 1-tert-butyl-5-[(2S)-1-pyrazol-1-ylpropan-2-yl]-3-(thiophen-2-ylmethyl)-1,2,4-triazole —— C17H23N5S
1-tert-butyl-5-[(2S)-1-pyrazol-1-ylpropan-2-yl]-3-(thiophen-2-ylmethyl)-1,2,4-triazole
—— (2R)-N-[3-(tetrazol-1-yl)phenyl]-2-(2-thiophen-2-ylethyl)piperidine-1-carboxamide —— C19H22N6OS
(2R)-N-[3-(tetrazol-1-yl)phenyl]-2-(2-thiophen-2-ylethyl)piperidine-1-carboxamide
—— N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-[(2S)-2-methyl-5-oxopyrrolidin-1-yl]acetamide —— C20H26N4O2
N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-[(2S)-2-methyl-5-oxopyrrolidin-1-yl]acetamide
—— (2S)-2-(pyrrolidin-1-ylmethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide —— C18H25N7O
(2S)-2-(pyrrolidin-1-ylmethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide
—— 3-[(3R)-3-(1-butylimidazol-2-yl)piperidin-1-yl]-5-phenyl-1,2,4-oxadiazole —— C20H25N5O
3-[(3R)-3-(1-butylimidazol-2-yl)piperidin-1-yl]-5-phenyl-1,2,4-oxadiazole
—— 1-[(2R)-oxolane-2-carbonyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide —— C20H24N4O3
1-[(2R)-oxolane-2-carbonyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
—— N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-[(2R)-2-methyl-5-oxopyrrolidin-1-yl]acetamide —— C20H26N4O2
N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-[(2R)-2-methyl-5-oxopyrrolidin-1-yl]acetamide
—— 2-[2-[(3S)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl]imidazol-1-yl]acetamide —— C15H21N5O2
2-[2-[(3S)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl]imidazol-1-yl]acetamide
—— 2-[2-[(3R)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl]imidazol-1-yl]acetamide —— C15H21N5O2
2-[2-[(3R)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl]imidazol-1-yl]acetamide
—— N-[(2S)-2-(N-methylanilino)propyl]-2-(2-phenylimidazol-1-yl)acetamide —— C21H24N4O
N-[(2S)-2-(N-methylanilino)propyl]-2-(2-phenylimidazol-1-yl)acetamide
—— N-[(1R)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-(2-phenylimidazol-1-yl)acetamide —— C17H20N6O
N-[(1R)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-(2-phenylimidazol-1-yl)acetamide
—— N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-(2-phenylimidazol-1-yl)acetamide —— C17H20N6O
N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-(2-phenylimidazol-1-yl)acetamide
—— (2S)-N-[3-(tetrazol-1-yl)phenyl]-2-(2-thiophen-2-ylethyl)piperidine-1-carboxamide —— C19H22N6OS
(2S)-N-[3-(tetrazol-1-yl)phenyl]-2-(2-thiophen-2-ylethyl)piperidine-1-carboxamide
—— 1-[(2S)-oxolane-2-carbonyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide —— C20H24N4O3
1-[(2S)-oxolane-2-carbonyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
—— N-[(2R)-2-(N-methylanilino)propyl]-2-(2-phenylimidazol-1-yl)acetamide —— C21H24N4O
N-[(2R)-2-(N-methylanilino)propyl]-2-(2-phenylimidazol-1-yl)acetamide
—— [(3S)-2-oxooxolan-3-yl] 3-(2-methylphenyl)-1-phenylpyrazole-4-carboxylate —— C21H18N2O4
[(3S)-2-oxooxolan-3-yl] 3-(2-methylphenyl)-1-phenylpyrazole-4-carboxylate
—— N-[(1S)-1-[2-(3-fluorophenyl)-5-(2-methoxyethyl)-1,2,4-triazol-3-yl]-2-methylpropyl]acetamide —— C17H23FN4O2
N-[(1S)-1-[2-(3-fluorophenyl)-5-(2-methoxyethyl)-1,2,4-triazol-3-yl]-2-methylpropyl]acetamide
—— [(3R)-2-oxooxolan-3-yl] 3-(2-methylphenyl)-1-phenylpyrazole-4-carboxylate —— C21H18N2O4
[(3R)-2-oxooxolan-3-yl] 3-(2-methylphenyl)-1-phenylpyrazole-4-carboxylate
—— 1-[(1-ethylimidazol-2-yl)methyl]-1-methyl-3-[2-[(1S)-1-phenylethyl]pyrazol-3-yl]urea —— C19H24N6O
1-[(1-ethylimidazol-2-yl)methyl]-1-methyl-3-[2-[(1S)-1-phenylethyl]pyrazol-3-yl]urea
—— 1-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea —— C16H21N5O4S
1-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea
—— 1-[(1-ethylimidazol-2-yl)methyl]-1-methyl-3-[2-[(1R)-1-phenylethyl]pyrazol-3-yl]urea —— C19H24N6O
1-[(1-ethylimidazol-2-yl)methyl]-1-methyl-3-[2-[(1R)-1-phenylethyl]pyrazol-3-yl]urea
—— 1-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea —— C16H21N5O4S
1-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea
—— N-[(1R)-1-[2-(3-fluorophenyl)-5-(2-methoxyethyl)-1,2,4-triazol-3-yl]-2-methylpropyl]acetamide —— C17H23FN4O2
N-[(1R)-1-[2-(3-fluorophenyl)-5-(2-methoxyethyl)-1,2,4-triazol-3-yl]-2-methylpropyl]acetamide
—— N-[(1R)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)tetrazol-1-yl]acetamide —— C12H19N9O2S
N-[(1R)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)tetrazol-1-yl]acetamide
—— (3S)-1-[2-[methyl-[(3-pyrazol-1-ylphenyl)methyl]amino]pyrimidin-4-yl]piperidin-3-ol —— C20H24N6O
(3S)-1-[2-[methyl-[(3-pyrazol-1-ylphenyl)methyl]amino]pyrimidin-4-yl]piperidin-3-ol
—— 4-fluoro-3-[3-(furan-2-yl)-5-[(3R)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzenesulfonamide —— C16H15FN4O4S
4-fluoro-3-[3-(furan-2-yl)-5-[(3R)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzenesulfonamide
—— (3S)-3-[3-cyclopentyl-5-(tetrazol-1-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide —— C13H19N7O2S
(3S)-3-[3-cyclopentyl-5-(tetrazol-1-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide
—— N-[(1S)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)tetrazol-1-yl]acetamide —— C12H19N9O2S
N-[(1S)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)tetrazol-1-yl]acetamide
—— [3-(2-Methylphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(phenylcarbamoylamino)propanoate —— C20H20N4O4
[3-(2-Methylphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(phenylcarbamoylamino)propanoate
—— 4-fluoro-3-[3-(furan-2-yl)-5-[(3S)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzenesulfonamide —— C16H15FN4O4S
4-fluoro-3-[3-(furan-2-yl)-5-[(3S)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzenesulfonamide
—— 1-[[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea —— C21H25N5O2
1-[[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea
—— 3-[(3R)-1-methylpiperidin-3-yl]-1-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propan-1-one —— C21H28N4O
3-[(3R)-1-methylpiperidin-3-yl]-1-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propan-1-one
—— 3-[(3S)-1-methylpiperidin-3-yl]-1-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propan-1-one —— C21H28N4O
3-[(3S)-1-methylpiperidin-3-yl]-1-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propan-1-one
—— 1,3-dimethyl-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine —— C12H16N6S
1,3-dimethyl-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine
—— 1-[[(3R)-1-(furan-2-ylmethyl)piperidin-3-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea —— C21H25N5O2
1-[[(3R)-1-(furan-2-ylmethyl)piperidin-3-yl]methyl]-3-(2-pyrazol-1-ylphenyl)urea
—— 1,3-dimethyl-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine —— C12H16N6S
1,3-dimethyl-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrazolo[3,4-d][1,3]thiazol-5-amine
—— (3R)-3-[3-cyclopentyl-5-(tetrazol-1-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide —— C13H19N7O2S
(3R)-3-[3-cyclopentyl-5-(tetrazol-1-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide
—— (3S)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide —— C20H24N6O2
(3S)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
—— (3S)-1-(5-methyl-1,3-oxazole-4-carbonyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-3-carboxamide —— C18H19N7O3
(3S)-1-(5-methyl-1,3-oxazole-4-carbonyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-3-carboxamide