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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C19H26N4O2S
2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S)-2-methylcyclohexyl]acetamide —— C21H28N4O2S
2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S)-2-methylcyclohexyl]acetamide
—— N-(1-adamantylmethyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C23H30N4OS
N-(1-adamantylmethyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-pentan-2-yl]acetamide —— C19H26N4O2S
2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-pentan-2-yl]acetamide
—— (2S)-N-(4-fluoro-3-nitrophenyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C17H14FN5O3S
(2S)-N-(4-fluoro-3-nitrophenyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— N-[(2S)-butan-2-yl]-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C17H24N4O2S
N-[(2S)-butan-2-yl]-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— N-(1-cyanocyclohexyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H23N5OS
N-(1-cyanocyclohexyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 1-(3,4-dihydro-2H-quinolin-1-yl)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C22H24N4O2S
1-(3,4-dihydro-2H-quinolin-1-yl)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— N-[(4-Methylphenyl)methyl]-2-[(5-phenyl-4H-1,2,4-triazol-3-YL)sulfanyl]acetamide —— C18H18N4OS
N-[(4-Methylphenyl)methyl]-2-[(5-phenyl-4H-1,2,4-triazol-3-YL)sulfanyl]acetamide
—— (2S)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C14H18N4O2S
(2S)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-(1,3-benzodioxol-5-yl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C18H16N4O3S
(2R)-N-(1,3-benzodioxol-5-yl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— (2S)-1-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propan-1-one —— C20H20N4OS
(2S)-1-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propan-1-one
—— (5R)-7-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5R)-7-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (5S)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5S)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (2R)-N-cyclopentyl-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H26N4O2S
(2R)-N-cyclopentyl-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-cyclohexyl-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2R)-N-cyclohexyl-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C18H24N4O3S
1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— 2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-methyl-N-[(2-methylphenyl)methyl]acetamide —— C23H26N4O2S
2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-methyl-N-[(2-methylphenyl)methyl]acetamide
—— (2S)-N-(4-fluorophenyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C19H19FN4OS
(2S)-N-(4-fluorophenyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(2S)-3-methylbutan-2-yl]-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C17H24N4OS
N-[(2S)-3-methylbutan-2-yl]-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-[[5-(4-methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C17H22N4O3S2
N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-[[5-(4-methylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— N-benzyl-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-propan-2-ylacetamide —— C23H28N4O2S
N-benzyl-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-propan-2-ylacetamide
—— 2-[[[(1S)-1-phenylethyl]-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]methyl]phenol —— C24H23N3O2
2-[[[(1S)-1-phenylethyl]-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]methyl]phenol
—— 3,3-dimethyl-4-[2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1H-quinoxalin-2-one —— C22H23N5O2S
3,3-dimethyl-4-[2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1H-quinoxalin-2-one
—— (5R)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane —— C18H19N5O
(5R)-7-(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (2S)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-(2,3,4-trifluorophenyl)propanamide —— C17H13F3N4OS
(2S)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-(2,3,4-trifluorophenyl)propanamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C17H22N4O3S2
N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— [2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate —— C21H27N3O3
[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate
—— (2R)-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propan-1-one —— C18H24N4OS
(2R)-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propan-1-one
—— N-[(4-fluorophenyl)methyl]-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H19FN4OS
N-[(4-fluorophenyl)methyl]-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— Tert-butyl 2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C17H23N3O3S
Tert-butyl 2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— 1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C21H28N4O2S
1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— N-[(3R)-1,1-dioxothiolan-3-yl]-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C16H20N4O3S2
N-[(3R)-1,1-dioxothiolan-3-yl]-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 1-[(R)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-3-[(1S,2S)-2-(hydroxymethyl)cycloheptyl]urea —— C17H27N3O2S
1-[(R)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-3-[(1S,2S)-2-(hydroxymethyl)cycloheptyl]urea
—— 1-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R,2S)-2-(hydroxymethyl)cycloheptyl]urea —— C17H27N3O2S
1-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R,2S)-2-(hydroxymethyl)cycloheptyl]urea
—— 2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C18H24N4OS
2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— N-(2-methoxyethyl)-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C17H22N4O3S
N-(2-methoxyethyl)-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (1S,2S,4R)-N-[1-(2-fluorophenyl)pyrazol-4-yl]-7-oxabicyclo[2.2.1]heptane-2-carboxamide —— C16H16FN3O2
(1S,2S,4R)-N-[1-(2-fluorophenyl)pyrazol-4-yl]-7-oxabicyclo[2.2.1]heptane-2-carboxamide
—— 5-(2-fluorophenyl)-N-[(2S)-2-pyridin-4-ylpropyl]-1H-pyrazole-4-carboxamide —— C18H17FN4O
5-(2-fluorophenyl)-N-[(2S)-2-pyridin-4-ylpropyl]-1H-pyrazole-4-carboxamide
—— 1-[(2R)-2-cyclohexyl-1-hydroxypropan-2-yl]-3-[[2-(dimethylamino)-3-methylimidazol-4-yl]methyl]urea —— C17H31N5O2
1-[(2R)-2-cyclohexyl-1-hydroxypropan-2-yl]-3-[[2-(dimethylamino)-3-methylimidazol-4-yl]methyl]urea
—— (4R)-6-amino-3-(3-ethoxyphenyl)-4-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C19H16N4O2S
(4R)-6-amino-3-(3-ethoxyphenyl)-4-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— ethyl 2-[(1S)-1-[(5-chloropyrimidin-2-yl)amino]ethyl]-4-methyl-1,3-thiazole-5-carboxylate —— C13H15ClN4O2S
ethyl 2-[(1S)-1-[(5-chloropyrimidin-2-yl)amino]ethyl]-4-methyl-1,3-thiazole-5-carboxylate
—— 2-(1-Phenylpyrazol-3-yl)-1-pyrrolidin-1-ylethanone —— C15H17N3O
2-(1-Phenylpyrazol-3-yl)-1-pyrrolidin-1-ylethanone
—— (2S)-N-(2-cyanoethyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-phenylpropanamide —— C22H23N5OS
(2S)-N-(2-cyanoethyl)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-phenylpropanamide
—— 5-[2-[(1S,3S)-3-methylcyclohexyl]ethylsulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole —— C14H24N2O3S2
5-[2-[(1S,3S)-3-methylcyclohexyl]ethylsulfanylmethyl]-3-(methylsulfonylmethyl)-1,2,4-oxadiazole
—— [(4aR,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[4,3-b]pyridin-1-yl]-[1-(3-bromophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone —— C22H26BrN3O2
[(4aR,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[4,3-b]pyridin-1-yl]-[1-(3-bromophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone
—— [(4aS,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[4,3-b]pyridin-1-yl]-[1-(3-bromophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone —— C22H26BrN3O2
[(4aS,8aR)-2,3,4,4a,5,7,8,8a-octahydropyrano[4,3-b]pyridin-1-yl]-[1-(3-bromophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone
—— 1-[(1R,3S)-3-ethylsulfanylcyclopentyl]-3-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-1-methylurea —— C15H22N4OS2
1-[(1R,3S)-3-ethylsulfanylcyclopentyl]-3-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-1-methylurea
—— 1-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R,2S)-2-(hydroxymethyl)cycloheptyl]urea —— C17H27N3O2S
1-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(1R,2S)-2-(hydroxymethyl)cycloheptyl]urea
—— 1-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C21H28N4O2S
1-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone