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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-bromo-N-[(5R)-5-methyl-4,5-dihydro-1,2-oxazol-3-yl]-5-propan-2-yl-1H-pyrazole-3-carboxamide —— C11H15BrN4O2
4-bromo-N-[(5R)-5-methyl-4,5-dihydro-1,2-oxazol-3-yl]-5-propan-2-yl-1H-pyrazole-3-carboxamide
—— N-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-1-ethylpyrazole-4-carboxamide —— C14H15ClFN3O2
N-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-1-ethylpyrazole-4-carboxamide
—— 2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2R)-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C22H24N4O2S
2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2R)-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— (2S)-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-(2-oxopyrrolidin-1-yl)butanamide —— C19H24N4O2
(2S)-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-(2-oxopyrrolidin-1-yl)butanamide
—— 2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R,2R)-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C22H24N4O2S
2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R,2R)-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— (2R)-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-(2-oxopyrrolidin-1-yl)butanamide —— C19H24N4O2
(2R)-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-(2-oxopyrrolidin-1-yl)butanamide
—— (2S)-2-hydroxy-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-phenylacetamide —— C19H19N3O2
(2S)-2-hydroxy-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-phenylacetamide
—— N-[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-pyrazol-1-ylbenzamide —— C19H17N3O2
N-[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-pyrazol-1-ylbenzamide
—— N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(tetrazol-1-yl)benzamide —— C17H15N5O2
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(tetrazol-1-yl)benzamide
—— N-[4-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]butyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C23H34N4O3
N-[4-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]butyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— 1-cyclopentyl-N-(5-methyl-1,3-thiazol-2-yl)methanesulfonamide —— C10H16N2O2S2
1-cyclopentyl-N-(5-methyl-1,3-thiazol-2-yl)methanesulfonamide
—— [(3R)-3-methyl-4-(2,2,2-trifluoroethyl)piperazin-1-yl]-(1-phenyl-5-propan-2-ylpyrazol-4-yl)methanone —— C20H25F3N4O
[(3R)-3-methyl-4-(2,2,2-trifluoroethyl)piperazin-1-yl]-(1-phenyl-5-propan-2-ylpyrazol-4-yl)methanone
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 4-oxo-4-(5-phenyl-3,4-dihydropyrazol-2-yl)butanoate —— C23H21N3O4
(5-Phenyl-1,3-oxazol-2-yl)methyl 4-oxo-4-(5-phenyl-3,4-dihydropyrazol-2-yl)butanoate
—— 5-(2-fluorophenyl)-N-[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-4-carboxamide —— C19H16FN3O2
5-(2-fluorophenyl)-N-[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-4-carboxamide
—— N-[4-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]butyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C23H34N4O3
N-[4-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]butyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— [(3S)-1-[2-(5-chlorothiophen-2-yl)-4-methyl-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]urea —— C14H15ClN4O2S2
[(3S)-1-[2-(5-chlorothiophen-2-yl)-4-methyl-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]urea
—— (2R)-2-hydroxy-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-phenylacetamide —— C19H19N3O2
(2R)-2-hydroxy-N-[[3-(1-methylpyrazol-4-yl)phenyl]methyl]-2-phenylacetamide
—— N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-pyrazol-1-ylbenzamide —— C19H17N3O2
N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-pyrazol-1-ylbenzamide
—— N-[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(tetrazol-1-yl)benzamide —— C17H15N5O2
N-[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(tetrazol-1-yl)benzamide
—— 5-(2-fluorophenyl)-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-4-carboxamide —— C19H16FN3O2
5-(2-fluorophenyl)-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-4-carboxamide
—— [(2S)-1-methoxy-1-oxobutan-2-yl] 2-methyl-5-propan-2-ylpyrazole-3-carboxylate —— C13H20N2O4
[(2S)-1-methoxy-1-oxobutan-2-yl] 2-methyl-5-propan-2-ylpyrazole-3-carboxylate
—— N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(tetrazol-1-yl)benzamide —— C17H15N5O2
N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(tetrazol-1-yl)benzamide
—— N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-pyrazol-1-ylbenzamide —— C19H17N3O2
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-pyrazol-1-ylbenzamide
—— [(3S)-3-methyl-4-(2,2,2-trifluoroethyl)piperazin-1-yl]-(1-phenyl-5-propan-2-ylpyrazol-4-yl)methanone —— C20H25F3N4O
[(3S)-3-methyl-4-(2,2,2-trifluoroethyl)piperazin-1-yl]-(1-phenyl-5-propan-2-ylpyrazol-4-yl)methanone
—— 5-[2-(1-Adamantyl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C23H24N4O2
5-[2-(1-Adamantyl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— [(3R)-1-[2-(5-chlorothiophen-2-yl)-4-methyl-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]urea —— C14H15ClN4O2S2
[(3R)-1-[2-(5-chlorothiophen-2-yl)-4-methyl-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]urea
—— [(2R)-1-methoxy-1-oxobutan-2-yl] 2-methyl-5-propan-2-ylpyrazole-3-carboxylate —— C13H20N2O4
[(2R)-1-methoxy-1-oxobutan-2-yl] 2-methyl-5-propan-2-ylpyrazole-3-carboxylate
—— (2S,3R)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide —— C17H21N3O3
(2S,3R)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide
—— 1-[(2R)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(5-methyl-1,3-thiazol-2-yl)methyl]urea —— C14H15ClFN3O2S
1-[(2R)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(5-methyl-1,3-thiazol-2-yl)methyl]urea
—— (2R)-2-[[5-[4-(diethylamino)phenyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H25N5OS
(2R)-2-[[5-[4-(diethylamino)phenyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2S,3S)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide —— C17H21N3O3
(2S,3S)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide
—— (2R,3R)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide —— C17H21N3O3
(2R,3R)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide
—— (E)-3-(furan-2-yl)-N-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]prop-2-en-1-amine —— C13H16N2OS
(E)-3-(furan-2-yl)-N-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]prop-2-en-1-amine
—— 1-[(2R)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]urea —— C15H17ClFN3O3
1-[(2R)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]urea
—— 1-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]urea —— C15H17ClFN3O3
1-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]urea
—— 2-[[4-(Furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-morpholin-4-ylethanone —— C20H22N4O3S
2-[[4-(Furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-morpholin-4-ylethanone
—— (E)-3-(furan-2-yl)-N-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]prop-2-en-1-amine —— C13H16N2OS
(E)-3-(furan-2-yl)-N-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]prop-2-en-1-amine
—— (2R,3S)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide —— C17H21N3O3
(2R,3S)-N-[5-(3-methoxyphenyl)-2-methylpyrazol-3-yl]-3-methyloxolane-2-carboxamide
—— 1-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-(5-methyl-1,3-thiazol-2-yl)urea —— C13H13ClFN3O2S
1-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-(5-methyl-1,3-thiazol-2-yl)urea
—— 1-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(5-methyl-1,3-thiazol-2-yl)methyl]urea —— C14H15ClFN3O2S
1-[(2S)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-[(5-methyl-1,3-thiazol-2-yl)methyl]urea
—— 2,4,6-trimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}benzenesulfonamide —— C19H21N3O3S
2,4,6-trimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}benzenesulfonamide
—— (2S)-N-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxy-N-propan-2-ylpropanamide —— C22H25N3O3
(2S)-N-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxy-N-propan-2-ylpropanamide
—— 1-[(2R)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-(5-methyl-1,3-thiazol-2-yl)urea —— C13H13ClFN3O2S
1-[(2R)-2-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-3-(5-methyl-1,3-thiazol-2-yl)urea
—— N-(2,6-difluorophenyl)-2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetamide —— C19H13F2N5O2
N-(2,6-difluorophenyl)-2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetamide
—— N-[(4-methylphenyl)methyl]-2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetamide —— C21H19N5O2
N-[(4-methylphenyl)methyl]-2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetamide
—— 5-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C22H19N5O2
5-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— ethyl 2,4-dimethyl-5-[2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetyl]-1H-pyrrole-3-carboxylate —— C22H21N5O4
ethyl 2,4-dimethyl-5-[2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetyl]-1H-pyrrole-3-carboxylate
—— 5-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C19H21N5O2
5-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C20H23N5O2
5-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— N-[(3-chlorophenyl)methyl]-2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetamide —— C20H16ClN5O2
N-[(3-chlorophenyl)methyl]-2-(4-oxo-1-phenylpyrazolo[3,4-d]pyrimidin-5-yl)acetamide