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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8R)-8-(3-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8R)-8-(3-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(2,3-dimethoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H21N3O4S
(8R)-8-(2,3-dimethoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 3-[(3S)-3-methyl-2,5-dioxo-3-phenylpyrrolidin-1-yl]-N-[4-(tetrazol-1-yl)phenyl]propanamide —— C21H20N6O3
3-[(3S)-3-methyl-2,5-dioxo-3-phenylpyrrolidin-1-yl]-N-[4-(tetrazol-1-yl)phenyl]propanamide
—— (8S)-8-(4-hydroxy-3-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8S)-8-(4-hydroxy-3-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— methyl (3S)-3-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-3-(5-phenyl-1H-pyrazol-4-yl)propanoate —— C17H18N4O3
methyl (3S)-3-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-3-(5-phenyl-1H-pyrazol-4-yl)propanoate
—— (8S)-1-(3-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H18ClN5OS
(8S)-1-(3-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— methyl 4-[(8S)-1-(4-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoate —— C21H19N3O4S
methyl 4-[(8S)-1-(4-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoate
—— (8R)-1-(3-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H18ClN5OS
(8R)-1-(3-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(4-hydroxy-3-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8R)-8-(4-hydroxy-3-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-8-(3-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8S)-8-(3-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[[(1R,2S,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide —— C15H20N2O2
N-[[(1R,2S,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide
—— (8R)-1-(3-chlorophenyl)-8-(4-hydroxy-3,5-dimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H18ClN3O4S
(8R)-1-(3-chlorophenyl)-8-(4-hydroxy-3,5-dimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(3-chloro-4-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14ClN3O2S
(8R)-8-(3-chloro-4-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 3-[(4S)-1-(2-chlorophenyl)-6-methyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol —— C18H14ClN3OS
3-[(4S)-1-(2-chlorophenyl)-6-methyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol
—— N-[[(1R,2R,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide —— C15H20N2O2
N-[[(1R,2R,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)acetamide
—— [2-[(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-thiophen-3-ylacetate —— C19H19N3O4S
[2-[(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-thiophen-3-ylacetate
—— (8R)-1-(3-bromophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14BrN3O2S
(8R)-1-(3-bromophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(1-methylpyrazol-4-yl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H15N5OS
(8R)-8-(1-methylpyrazol-4-yl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(3-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14ClN3O2S
(8S)-1-(3-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(3-bromophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14BrN3O2S
(8S)-1-(3-bromophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-thiophen-3-ylacetate —— C20H21N3O4S
[(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-thiophen-3-ylacetate
—— (8S)-1-phenyl-8-(2,4,5-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H21N3O4S
(8S)-1-phenyl-8-(2,4,5-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(4R)-2,2-dimethyloxan-4-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C18H23N3O3
N-[(4R)-2,2-dimethyloxan-4-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— 3-[(4R)-1-(2-chlorophenyl)-6-methyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol —— C18H14ClN3OS
3-[(4R)-1-(2-chlorophenyl)-6-methyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol
—— (8R)-1-phenyl-8-(2,4,5-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H21N3O4S
(8R)-1-phenyl-8-(2,4,5-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(4S)-2,2-dimethyloxan-4-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C18H23N3O3
N-[(4S)-2,2-dimethyloxan-4-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— (8R)-1-(3-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14ClN3O2S
(8R)-1-(3-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2,4-difluorobenzoate —— C19H15F2N3O3
[2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2,4-difluorobenzoate
—— (8S)-1-(4-chlorophenyl)-8-(4-hydroxy-3,5-dimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H18ClN3O4S
(8S)-1-(4-chlorophenyl)-8-(4-hydroxy-3,5-dimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-8-(2-methylpropyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H19N3OS
(8S)-8-(2-methylpropyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 4-[(8R)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14ClN3O3S
4-[(8R)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— (8S)-1-(4-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14ClN3O2S
(8S)-1-(4-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 4-[(8S)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14ClN3O3S
4-[(8S)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— (8R)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H19N5O2S
(8R)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(2-methylpropyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H19N3OS
(8R)-8-(2-methylpropyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(4-chlorophenyl)-8-(4-hydroxy-3,5-dimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H18ClN3O4S
(8R)-1-(4-chlorophenyl)-8-(4-hydroxy-3,5-dimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— methyl 2-[[(3S)-2,2-dimethyl-5-oxooxolane-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C13H16N2O5S
methyl 2-[[(3S)-2,2-dimethyl-5-oxooxolane-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— methyl 2-[[(3R)-2,2-dimethyl-5-oxooxolane-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C13H16N2O5S
methyl 2-[[(3R)-2,2-dimethyl-5-oxooxolane-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— (8S)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H19N5O2S
(8S)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(4-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14ClN3O2S
(8R)-1-(4-chlorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(3S)-1,1-dioxothiolan-3-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C16H18FN3O3S
N-[(3S)-1,1-dioxothiolan-3-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— (3S)-3-(tetrazol-1-yl)-3-thiophen-3-ylpropanoic acid —— C8H8N4O2S
(3S)-3-(tetrazol-1-yl)-3-thiophen-3-ylpropanoic acid
—— (3R)-3-(tetrazol-1-yl)-3-thiophen-3-ylpropanoic acid —— C8H8N4O2S
(3R)-3-(tetrazol-1-yl)-3-thiophen-3-ylpropanoic acid
—— (8S)-8-(4-hydroxy-3-methoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H19N3O4S
(8S)-8-(4-hydroxy-3-methoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(3R)-1,1-dioxothiolan-3-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C16H18FN3O3S
N-[(3R)-1,1-dioxothiolan-3-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— (8S)-8-(1,5-dimethylpyrazol-4-yl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H17N5OS
(8S)-8-(1,5-dimethylpyrazol-4-yl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(4-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13ClN4OS
(8R)-1-(4-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(3-fluorophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16FN3O3S
(8S)-1-(3-fluorophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(4-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13ClN4OS
(8S)-1-(4-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2,4-difluorobenzoate —— C21H19F2N3O4
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2,4-difluorobenzoate