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中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl (2R)-2-[1-[[2-(methoxymethyl)-1,3-thiazol-4-yl]methyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C15H21N3O3S
methyl (2R)-2-[1-[[2-(methoxymethyl)-1,3-thiazol-4-yl]methyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— 3-[(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methylsulfanyl]-5-cyclopropyl-1-phenyl-1,2,4-triazole —— C20H18ClN3O2S
3-[(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methylsulfanyl]-5-cyclopropyl-1-phenyl-1,2,4-triazole
—— 3-(2-propan-2-ylimidazol-1-yl)-N-[(1R)-2,2,2-trifluoro-1-(1-methylpyrrol-3-yl)ethyl]propanamide —— C16H21F3N4O
3-(2-propan-2-ylimidazol-1-yl)-N-[(1R)-2,2,2-trifluoro-1-(1-methylpyrrol-3-yl)ethyl]propanamide
—— methyl (2S)-2-[3,5-dimethyl-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C13H18N4O3
methyl (2S)-2-[3,5-dimethyl-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— methyl (2S)-2-[1-[2-[cyclopropyl(methyl)amino]-2-oxoethyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C15H23N3O3
methyl (2S)-2-[1-[2-[cyclopropyl(methyl)amino]-2-oxoethyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— methyl (2R)-2-[3,5-dimethyl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrazol-4-yl]propanoate —— C15H22N4O3
methyl (2R)-2-[3,5-dimethyl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrazol-4-yl]propanoate
—— methyl 2-[(2R)-2-(4-chloropyrazol-1-yl)propyl]-4-ethyl-1,3-thiazole-5-carboxylate —— C13H16ClN3O2S
methyl 2-[(2R)-2-(4-chloropyrazol-1-yl)propyl]-4-ethyl-1,3-thiazole-5-carboxylate
—— methyl (2S)-2-(3,5-dimethyl-1-pent-4-enylpyrazol-4-yl)propanoate —— C14H22N2O2
methyl (2S)-2-(3,5-dimethyl-1-pent-4-enylpyrazol-4-yl)propanoate
—— N-[(2R)-2-cyano-3-methylbutan-2-yl]-3-methyl-5-propyl-1,2-oxazole-4-carboxamide —— C14H21N3O2
N-[(2R)-2-cyano-3-methylbutan-2-yl]-3-methyl-5-propyl-1,2-oxazole-4-carboxamide
—— (2R,5S)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide —— C21H25N5O3
(2R,5S)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide
—— methyl (2S)-2-[1-[[2-(methoxymethyl)-1,3-thiazol-4-yl]methyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C15H21N3O3S
methyl (2S)-2-[1-[[2-(methoxymethyl)-1,3-thiazol-4-yl]methyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— methyl (2R)-2-[3,5-dimethyl-1-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C16H18N4O3S
methyl (2R)-2-[3,5-dimethyl-1-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— (2S)-1-ethoxy-3-[(3S)-3-(5-phenyl-1H-imidazol-2-yl)piperidin-1-yl]propan-2-ol —— C19H27N3O2
(2S)-1-ethoxy-3-[(3S)-3-(5-phenyl-1H-imidazol-2-yl)piperidin-1-yl]propan-2-ol
—— methyl (2S)-2-[3,5-dimethyl-1-[(1-phenylpyrazol-3-yl)methyl]pyrazol-4-yl]propanoate —— C19H22N4O2
methyl (2S)-2-[3,5-dimethyl-1-[(1-phenylpyrazol-3-yl)methyl]pyrazol-4-yl]propanoate
—— methyl (2S)-2-[3,5-dimethyl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrazol-4-yl]propanoate —— C15H22N4O3
methyl (2S)-2-[3,5-dimethyl-1-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyrazol-4-yl]propanoate
—— (2R)-1-ethoxy-3-[(3S)-3-(5-phenyl-1H-imidazol-2-yl)piperidin-1-yl]propan-2-ol —— C19H27N3O2
(2R)-1-ethoxy-3-[(3S)-3-(5-phenyl-1H-imidazol-2-yl)piperidin-1-yl]propan-2-ol
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-2-(5-phenyltetrazol-2-yl)acetamide —— C14H17N5O3S
N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-2-(5-phenyltetrazol-2-yl)acetamide
—— N-(3-tert-butyl-1,2-oxazol-5-yl)-2-[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylacetamide —— C16H18N6O3S
N-(3-tert-butyl-1,2-oxazol-5-yl)-2-[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylacetamide
—— methyl 2-[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]-4-ethyl-1,3-thiazole-5-carboxylate —— C14H20N2O3S
methyl 2-[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]-4-ethyl-1,3-thiazole-5-carboxylate
—— 3-(2-propan-2-ylimidazol-1-yl)-N-[(1S)-2,2,2-trifluoro-1-(1-methylpyrrol-3-yl)ethyl]propanamide —— C16H21F3N4O
3-(2-propan-2-ylimidazol-1-yl)-N-[(1S)-2,2,2-trifluoro-1-(1-methylpyrrol-3-yl)ethyl]propanamide
—— methyl (2S)-2-[3,5-dimethyl-1-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C16H18N4O3S
methyl (2S)-2-[3,5-dimethyl-1-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— methyl 2-[(2S)-2-(4-chloropyrazol-1-yl)propyl]-4-ethyl-1,3-thiazole-5-carboxylate —— C13H16ClN3O2S
methyl 2-[(2S)-2-(4-chloropyrazol-1-yl)propyl]-4-ethyl-1,3-thiazole-5-carboxylate
—— (2S,5S)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide —— C21H25N5O3
(2S,5S)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide
—— methyl (2R)-2-[3,5-dimethyl-1-[(1-propyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C14H22N6O2
methyl (2R)-2-[3,5-dimethyl-1-[(1-propyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— methyl (2R)-2-(3,5-dimethyl-1-pent-4-enylpyrazol-4-yl)propanoate —— C14H22N2O2
methyl (2R)-2-(3,5-dimethyl-1-pent-4-enylpyrazol-4-yl)propanoate
—— methyl (2R)-2-[1-[2-[cyclopropyl(methyl)amino]-2-oxoethyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C15H23N3O3
methyl (2R)-2-[1-[2-[cyclopropyl(methyl)amino]-2-oxoethyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— methyl 2-[(2S)-4-benzylmorpholin-2-yl]-4-ethyl-1,3-thiazole-5-carboxylate —— C18H22N2O3S
methyl 2-[(2S)-4-benzylmorpholin-2-yl]-4-ethyl-1,3-thiazole-5-carboxylate
—— (2R,5R)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide —— C21H25N5O3
(2R,5R)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide
—— (2S,5R)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide —— C21H25N5O3
(2S,5R)-5-(hydroxymethyl)-2-methyl-N-[3-[(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)methyl]phenyl]piperidine-1-carboxamide
—— [(2S)-1-(6-methylpyridazin-3-yl)pyrrolidin-2-yl]methyl 4,5,6,7-tetrahydro-1H-indazole-3-carboxylate —— C18H23N5O2
[(2S)-1-(6-methylpyridazin-3-yl)pyrrolidin-2-yl]methyl 4,5,6,7-tetrahydro-1H-indazole-3-carboxylate
—— methyl (2R)-2-[3,5-dimethyl-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C13H18N4O3
methyl (2R)-2-[3,5-dimethyl-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— methyl (2S)-2-[3,5-dimethyl-1-[(1-propyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate —— C14H22N6O2
methyl (2S)-2-[3,5-dimethyl-1-[(1-propyltetrazol-5-yl)methyl]pyrazol-4-yl]propanoate
—— 4-chloro-3-methyl-1-(4-methylphenyl)-N-(thiophen-2-ylmethyl)pyrazolo[3,4-b]pyridine-5-carboxamide —— C20H17ClN4OS
4-chloro-3-methyl-1-(4-methylphenyl)-N-(thiophen-2-ylmethyl)pyrazolo[3,4-b]pyridine-5-carboxamide
—— 4-chloro-N-[(3-methoxyphenyl)methyl]-3-methyl-1-(4-methylphenyl)pyrazolo[3,4-b]pyridine-5-carboxamide —— C23H21ClN4O2
4-chloro-N-[(3-methoxyphenyl)methyl]-3-methyl-1-(4-methylphenyl)pyrazolo[3,4-b]pyridine-5-carboxamide
—— 4-chloro-1-(4-methoxyphenyl)-3-methyl-N-propylpyrazolo[3,4-b]pyridine-5-carboxamide —— C18H19ClN4O2
4-chloro-1-(4-methoxyphenyl)-3-methyl-N-propylpyrazolo[3,4-b]pyridine-5-carboxamide
—— 4-chloro-N,N-diethyl-3-methyl-1-phenylpyrazolo[3,4-b]pyridine-5-carboxamide —— C18H19ClN4O
4-chloro-N,N-diethyl-3-methyl-1-phenylpyrazolo[3,4-b]pyridine-5-carboxamide
—— 4-chloro-3-methyl-N-(4-methyl-1,3-thiazol-2-yl)-1-phenylpyrazolo[3,4-b]pyridine-5-carboxamide —— C18H14ClN5OS
4-chloro-3-methyl-N-(4-methyl-1,3-thiazol-2-yl)-1-phenylpyrazolo[3,4-b]pyridine-5-carboxamide
—— N-benzyl-4-chloro-N-ethyl-3-methyl-1-(4-methylphenyl)pyrazolo[3,4-b]pyridine-5-carboxamide —— C24H23ClN4O
N-benzyl-4-chloro-N-ethyl-3-methyl-1-(4-methylphenyl)pyrazolo[3,4-b]pyridine-5-carboxamide
—— 3-[[5-(4-Tert-butylphenyl)-4-cyclopentyl-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-1,2-oxazole —— C22H28N4OS
3-[[5-(4-Tert-butylphenyl)-4-cyclopentyl-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-1,2-oxazole
—— 4-chloro-3-methyl-1-phenyl-N,N-dipropylpyrazolo[3,4-b]pyridine-5-carboxamide —— C20H23ClN4O
4-chloro-3-methyl-1-phenyl-N,N-dipropylpyrazolo[3,4-b]pyridine-5-carboxamide
—— 4-chloro-3-methyl-1-phenyl-N-[(1S)-1-phenylethyl]pyrazolo[3,4-b]pyridine-5-carboxamide —— C22H19ClN4O
4-chloro-3-methyl-1-phenyl-N-[(1S)-1-phenylethyl]pyrazolo[3,4-b]pyridine-5-carboxamide
—— [4-chloro-1-(3-methoxyphenyl)-3-methylpyrazolo[3,4-b]pyridin-5-yl]-[(2S)-2-ethylpiperidin-1-yl]methanone —— C22H25ClN4O2
[4-chloro-1-(3-methoxyphenyl)-3-methylpyrazolo[3,4-b]pyridin-5-yl]-[(2S)-2-ethylpiperidin-1-yl]methanone
—— N-[(3S)-1-[(5-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl]methanesulfonamide —— C15H19N3O2S2
N-[(3S)-1-[(5-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl]methanesulfonamide
—— 4-chloro-1-(3-methoxyphenyl)-3-methyl-N-(4-methyl-1,3-thiazol-2-yl)pyrazolo[3,4-b]pyridine-5-carboxamide —— C19H16ClN5O2S
4-chloro-1-(3-methoxyphenyl)-3-methyl-N-(4-methyl-1,3-thiazol-2-yl)pyrazolo[3,4-b]pyridine-5-carboxamide
—— 4-chloro-3-methyl-1-(4-methylphenyl)-N-(2-methylpropyl)pyrazolo[3,4-b]pyridine-5-carboxamide —— C19H21ClN4O
4-chloro-3-methyl-1-(4-methylphenyl)-N-(2-methylpropyl)pyrazolo[3,4-b]pyridine-5-carboxamide
—— [4-Chloro-1-(4-fluorophenyl)-3-methylpyrazolo[3,4-b]pyridin-5-yl]-(4-ethylpiperazin-1-yl)methanone —— C20H21ClFN5O
[4-Chloro-1-(4-fluorophenyl)-3-methylpyrazolo[3,4-b]pyridin-5-yl]-(4-ethylpiperazin-1-yl)methanone
—— 3-[(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methylsulfanyl]-5-(2-fluorophenyl)-4-methyl-1,2,4-triazole —— C18H15ClFN3O2S
3-[(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methylsulfanyl]-5-(2-fluorophenyl)-4-methyl-1,2,4-triazole
—— (4-chloro-3-methyl-1-phenylpyrazolo[3,4-b]pyridin-5-yl)-[(2S,6S)-2,6-dimethylmorpholin-4-yl]methanone —— C20H21ClN4O2
(4-chloro-3-methyl-1-phenylpyrazolo[3,4-b]pyridin-5-yl)-[(2S,6S)-2,6-dimethylmorpholin-4-yl]methanone
—— N-[(2S)-2-hydroxy-2-pyridin-2-ylethyl]-1-(4-methylphenyl)-3-phenylpyrazole-4-carboxamide —— C24H22N4O2
N-[(2S)-2-hydroxy-2-pyridin-2-ylethyl]-1-(4-methylphenyl)-3-phenylpyrazole-4-carboxamide
—— 4-chloro-N-[3-(diethylamino)propyl]-3-methyl-1-phenylpyrazolo[3,4-b]pyridine-5-carboxamide —— C21H26ClN5O
4-chloro-N-[3-(diethylamino)propyl]-3-methyl-1-phenylpyrazolo[3,4-b]pyridine-5-carboxamide