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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(1-ethylpyrazol-4-yl)-2-oxo-N-[(1R)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]acetamide —— C18H19N5O2
2-(1-ethylpyrazol-4-yl)-2-oxo-N-[(1R)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]acetamide
—— 1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3-[(2R)-2-(4-fluorophenyl)-2-hydroxypropyl]urea —— C16H20FN3O2S
1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3-[(2R)-2-(4-fluorophenyl)-2-hydroxypropyl]urea
—— 1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-3-[(2S)-2-(4-fluorophenyl)-2-hydroxypropyl]urea —— C18H24FN3O3
1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-3-[(2S)-2-(4-fluorophenyl)-2-hydroxypropyl]urea
—— (1R,2R)-2-[(2,5-dimethyl-1,3-thiazol-4-yl)methylcarbamoylamino]-N-methylcyclohexane-1-carboxamide —— C15H24N4O2S
(1R,2R)-2-[(2,5-dimethyl-1,3-thiazol-4-yl)methylcarbamoylamino]-N-methylcyclohexane-1-carboxamide
—— 2-(4-methyl-5-oxo-1,2,4-triazol-1-yl)-N-[(1S)-1-thiophen-2-ylethyl]acetamide —— C11H14N4O2S
2-(4-methyl-5-oxo-1,2,4-triazol-1-yl)-N-[(1S)-1-thiophen-2-ylethyl]acetamide
—— 4-Methyl-2-[(4-pyrazol-1-ylphenyl)methyl]-1,2,4-triazol-3-one —— C13H13N5O
4-Methyl-2-[(4-pyrazol-1-ylphenyl)methyl]-1,2,4-triazol-3-one
—— 2-[[1-(2,6-Difluorophenyl)pyrazol-3-yl]methyl]-4-methyl-1,2,4-triazol-3-one —— C13H11F2N5O
2-[[1-(2,6-Difluorophenyl)pyrazol-3-yl]methyl]-4-methyl-1,2,4-triazol-3-one
—— [6-methyl-3-[[2-[(2R)-oxolan-2-yl]-1,3-thiazol-4-yl]methoxy]pyridin-2-yl]methanol —— C15H18N2O3S
[6-methyl-3-[[2-[(2R)-oxolan-2-yl]-1,3-thiazol-4-yl]methoxy]pyridin-2-yl]methanol
—— 2-(4-methyl-5-oxo-1,2,4-triazol-1-yl)-N-[(1R)-1-thiophen-2-ylethyl]acetamide —— C11H14N4O2S
2-(4-methyl-5-oxo-1,2,4-triazol-1-yl)-N-[(1R)-1-thiophen-2-ylethyl]acetamide
—— 4-Methyl-2-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]-1,2,4-triazol-3-one —— C10H14N4OS
4-Methyl-2-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]-1,2,4-triazol-3-one
—— [6-methyl-3-[[2-[(2S)-oxolan-2-yl]-1,3-thiazol-4-yl]methoxy]pyridin-2-yl]methanol —— C15H18N2O3S
[6-methyl-3-[[2-[(2S)-oxolan-2-yl]-1,3-thiazol-4-yl]methoxy]pyridin-2-yl]methanol
—— 1-[[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]methyl]-3-(4-pyridin-3-yl-1,3-thiazol-2-yl)urea —— C21H21N5O2S
1-[[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]methyl]-3-(4-pyridin-3-yl-1,3-thiazol-2-yl)urea
—— N-[(4-fluoro-3-methylphenyl)methyl]-5-methyl-1-[2-[(2R)-oxan-2-yl]oxyethyl]pyrazole-4-carboxamide —— C20H26FN3O3
N-[(4-fluoro-3-methylphenyl)methyl]-5-methyl-1-[2-[(2R)-oxan-2-yl]oxyethyl]pyrazole-4-carboxamide
—— N-[(4-fluoro-3-methylphenyl)methyl]-5-methyl-1-[2-[(2S)-oxan-2-yl]oxyethyl]pyrazole-4-carboxamide —— C20H26FN3O3
N-[(4-fluoro-3-methylphenyl)methyl]-5-methyl-1-[2-[(2S)-oxan-2-yl]oxyethyl]pyrazole-4-carboxamide
—— (5-methylpyrazin-2-yl)-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C18H18N6O
(5-methylpyrazin-2-yl)-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— 5-ethyl-2-[[(3R)-3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl]methyl]-1,3-oxazole —— C17H30N4O
5-ethyl-2-[[(3R)-3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl]methyl]-1,3-oxazole
—— (2R)-1-[[(2S)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]amino]-3-pyrazol-1-ylpropan-2-ol —— C15H25N3O2S
(2R)-1-[[(2S)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]amino]-3-pyrazol-1-ylpropan-2-ol
—— (3S)-N-[[3,5-dimethyl-1-(2-methylphenyl)pyrazol-4-yl]methyl]-3-(3-fluorophenyl)-3-hydroxy-N-methylpropanamide —— C23H26FN3O2
(3S)-N-[[3,5-dimethyl-1-(2-methylphenyl)pyrazol-4-yl]methyl]-3-(3-fluorophenyl)-3-hydroxy-N-methylpropanamide
—— 4-Methyl-2-[(1-propan-2-ylpyrazol-3-yl)methyl]-1,2,4-triazol-3-one —— C10H15N5O
4-Methyl-2-[(1-propan-2-ylpyrazol-3-yl)methyl]-1,2,4-triazol-3-one
—— (3R)-N-[[3,5-dimethyl-1-(2-methylphenyl)pyrazol-4-yl]methyl]-3-(3-fluorophenyl)-3-hydroxy-N-methylpropanamide —— C23H26FN3O2
(3R)-N-[[3,5-dimethyl-1-(2-methylphenyl)pyrazol-4-yl]methyl]-3-(3-fluorophenyl)-3-hydroxy-N-methylpropanamide
—— (1-methylpyrazol-4-yl)-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C17H18N6O
(1-methylpyrazol-4-yl)-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-(2-hydroxyethoxy)piperidin-1-yl]butan-1-one —— C18H24ClN5O3
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-(2-hydroxyethoxy)piperidin-1-yl]butan-1-one
—— (1-methylpyrazol-4-yl)-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C17H18N6O
(1-methylpyrazol-4-yl)-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— [(1R)-2,2,2-trifluoro-1-[(2R)-oxolan-2-yl]ethyl] 1,3-thiazole-4-carboxylate —— C10H10F3NO3S
[(1R)-2,2,2-trifluoro-1-[(2R)-oxolan-2-yl]ethyl] 1,3-thiazole-4-carboxylate
—— (2S)-1-[[(2S)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]amino]-3-pyrazol-1-ylpropan-2-ol —— C15H25N3O2S
(2S)-1-[[(2S)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]amino]-3-pyrazol-1-ylpropan-2-ol
—— 5-ethyl-2-[[(3S)-3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl]methyl]-1,3-oxazole —— C17H30N4O
5-ethyl-2-[[(3S)-3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl]methyl]-1,3-oxazole
—— [(2S)-2-methoxypropyl] 1-(2,4-difluorophenyl)pyrazole-4-carboxylate —— C14H14F2N2O3
[(2S)-2-methoxypropyl] 1-(2,4-difluorophenyl)pyrazole-4-carboxylate
—— 1-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)ethanone —— C22H20N6OS
1-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)ethanone
—— (5-methylpyrazin-2-yl)-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C18H18N6O
(5-methylpyrazin-2-yl)-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— [3-(2-methoxyethoxy)phenyl]-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C22H24N4O3
[3-(2-methoxyethoxy)phenyl]-[(2R)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— 1-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)ethanone —— C22H20N6OS
1-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)ethanone
—— [3-(2-methoxyethoxy)phenyl]-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone —— C22H24N4O3
[3-(2-methoxyethoxy)phenyl]-[(2S)-2-(3-phenyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methanone
—— 4-Methyl-2-[[1-methyl-5-(trifluoromethyl)pyrazol-4-yl]methyl]-1,2,4-triazol-3-one —— C9H10F3N5O
4-Methyl-2-[[1-methyl-5-(trifluoromethyl)pyrazol-4-yl]methyl]-1,2,4-triazol-3-one
—— 1,5-dimethyl-N-[(1R)-3-methyl-1-[3-(1H-1,2,4-triazol-5-yl)-1,2,4-oxadiazol-5-yl]butyl]pyrazole-4-carboxamide —— C15H20N8O2
1,5-dimethyl-N-[(1R)-3-methyl-1-[3-(1H-1,2,4-triazol-5-yl)-1,2,4-oxadiazol-5-yl]butyl]pyrazole-4-carboxamide
—— 1-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[(1-thiophen-2-ylcyclopentyl)methyl]urea —— C17H24N4O2S
1-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[(1-thiophen-2-ylcyclopentyl)methyl]urea
—— 1-[[1-(2,6-difluorophenyl)pyrazol-3-yl]methyl]-3-[(3R)-2-oxopiperidin-3-yl]urea —— C16H17F2N5O2
1-[[1-(2,6-difluorophenyl)pyrazol-3-yl]methyl]-3-[(3R)-2-oxopiperidin-3-yl]urea
—— [2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2-methylfuran-3-carboxylate —— C18H17N3O4
[2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2-methylfuran-3-carboxylate
—— 1-[(1S)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[(1-thiophen-2-ylcyclopentyl)methyl]urea —— C17H24N4O2S
1-[(1S)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[(1-thiophen-2-ylcyclopentyl)methyl]urea
—— 1-[2-(dimethylamino)-2-methylpropyl]-3-[(1R)-1-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]urea —— C15H28N4O2
1-[2-(dimethylamino)-2-methylpropyl]-3-[(1R)-1-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]urea
—— 1-[2-(dimethylamino)-2-methylpropyl]-3-[(1S)-1-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]urea —— C15H28N4O2
1-[2-(dimethylamino)-2-methylpropyl]-3-[(1S)-1-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]urea
—— 2-ethyl-N-(3-fluoropyridin-4-yl)-1,3-thiazole-5-carboxamide —— C11H10FN3OS
2-ethyl-N-(3-fluoropyridin-4-yl)-1,3-thiazole-5-carboxamide
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-(2-hydroxyethoxy)piperidin-1-yl]butan-1-one —— C18H24ClN5O3
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-(2-hydroxyethoxy)piperidin-1-yl]butan-1-one
—— 1-(1-adamantylmethyl)-3-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]urea —— C18H28N4O2
1-(1-adamantylmethyl)-3-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]urea
—— 1,5-dimethyl-N-[(1S)-3-methyl-1-[3-(1H-1,2,4-triazol-5-yl)-1,2,4-oxadiazol-5-yl]butyl]pyrazole-4-carboxamide —— C15H20N8O2
1,5-dimethyl-N-[(1S)-3-methyl-1-[3-(1H-1,2,4-triazol-5-yl)-1,2,4-oxadiazol-5-yl]butyl]pyrazole-4-carboxamide
—— [(2R)-2-methoxypropyl] 1-(2,4-difluorophenyl)pyrazole-4-carboxylate —— C14H14F2N2O3
[(2R)-2-methoxypropyl] 1-(2,4-difluorophenyl)pyrazole-4-carboxylate
—— 1-(1-adamantylmethyl)-3-[(1S)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]urea —— C18H28N4O2
1-(1-adamantylmethyl)-3-[(1S)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]urea
—— (2S)-N-[[1-(2,6-difluorophenyl)pyrazol-3-yl]methyl]-4-methylmorpholine-2-carboxamide —— C16H18F2N4O2
(2S)-N-[[1-(2,6-difluorophenyl)pyrazol-3-yl]methyl]-4-methylmorpholine-2-carboxamide
—— [(1S)-2,2,2-trifluoro-1-[(2S)-oxolan-2-yl]ethyl] 1,3-thiazole-4-carboxylate —— C10H10F3NO3S
[(1S)-2,2,2-trifluoro-1-[(2S)-oxolan-2-yl]ethyl] 1,3-thiazole-4-carboxylate
—— [(1R)-2,2,2-trifluoro-1-[(2S)-oxolan-2-yl]ethyl] 1,3-thiazole-4-carboxylate —— C10H10F3NO3S
[(1R)-2,2,2-trifluoro-1-[(2S)-oxolan-2-yl]ethyl] 1,3-thiazole-4-carboxylate
—— 1-[[1-(2,6-difluorophenyl)pyrazol-3-yl]methyl]-3-[(3S)-2-oxopiperidin-3-yl]urea —— C16H17F2N5O2
1-[[1-(2,6-difluorophenyl)pyrazol-3-yl]methyl]-3-[(3S)-2-oxopiperidin-3-yl]urea