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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8S)-1-(4-chlorophenyl)-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C13H9ClF3N3OS
(8S)-1-(4-chlorophenyl)-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 4-[(8S)-5-oxo-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H15N3O3S
4-[(8S)-5-oxo-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— 4-(1H-tetrazol-1-yl)phenyl [5-methyl-2-(propan-2-yl)phenoxy]acetate —— C19H20N4O3
4-(1H-tetrazol-1-yl)phenyl [5-methyl-2-(propan-2-yl)phenoxy]acetate
—— (8R)-1-(3-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13ClN4OS
(8R)-1-(3-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(4-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8S)-1-(4-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(4S)-2,2-dimethyloxan-4-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C20H27N3O3
N-[(4S)-2,2-dimethyloxan-4-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— 3-(3,4-dimethoxyphenyl)-N-[(4R)-2,2-dimethyloxan-4-yl]-1H-pyrazole-5-carboxamide —— C19H25N3O4
3-(3,4-dimethoxyphenyl)-N-[(4R)-2,2-dimethyloxan-4-yl]-1H-pyrazole-5-carboxamide
—— 3-(3,4-dimethoxyphenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazole-5-carboxamide —— C16H19N3O5S
3-(3,4-dimethoxyphenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-1H-pyrazole-5-carboxamide
—— methyl 2-[[(3S)-3-(4-chlorophenyl)-4-pyrrol-1-ylbutanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C20H20ClN3O3S
methyl 2-[[(3S)-3-(4-chlorophenyl)-4-pyrrol-1-ylbutanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— N-[(4R)-2,2-dimethyloxan-4-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C20H27N3O3
N-[(4R)-2,2-dimethyloxan-4-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— 4-[(8R)-5-oxo-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H15N3O3S
4-[(8R)-5-oxo-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— (8R)-8-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H21N3O4S
(8R)-8-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [(1R)-1-cyanoethyl] 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H19FN4O3S
[(1R)-1-cyanoethyl] 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— 3-(4-fluorophenyl)-5-[2-(4-methylphenoxy)ethylsulfanyl]-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazole —— C22H24FN3O2S
3-(4-fluorophenyl)-5-[2-(4-methylphenoxy)ethylsulfanyl]-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazole
—— (8R)-1-(3-bromophenyl)-8-(1,5-dimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H16BrN5OS
(8R)-1-(3-bromophenyl)-8-(1,5-dimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-8-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H21N3O4S
(8S)-8-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]acetamide —— C19H21N5O2S
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]acetamide
—— (8R)-8-(4-hydroxy-3-methoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H19N3O4S
(8R)-8-(4-hydroxy-3-methoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 1-[2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]pyrrolidin-2-one —— C19H21FN4O3S
1-[2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]pyrrolidin-2-one
—— [(1S)-1-cyanoethyl] 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H19FN4O3S
[(1S)-1-cyanoethyl] 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— 3-(4-fluorophenyl)-5-[2-(4-methylphenoxy)ethylsulfanyl]-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazole —— C22H24FN3O2S
3-(4-fluorophenyl)-5-[2-(4-methylphenoxy)ethylsulfanyl]-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazole
—— (8R)-1-(4-chlorophenyl)-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C13H9ClF3N3OS
(8R)-1-(4-chlorophenyl)-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(3R)-1,1-dioxothiolan-3-yl]-4-(2-propan-2-yltetrazol-5-yl)benzamide —— C15H19N5O3S
N-[(3R)-1,1-dioxothiolan-3-yl]-4-(2-propan-2-yltetrazol-5-yl)benzamide
—— 3-(3,4-dimethoxyphenyl)-N-[(4S)-2,2-dimethyloxan-4-yl]-1H-pyrazole-5-carboxamide —— C19H25N3O4
3-(3,4-dimethoxyphenyl)-N-[(4S)-2,2-dimethyloxan-4-yl]-1H-pyrazole-5-carboxamide
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-(5-methyltetrazol-1-yl)benzamide —— C16H22N6O
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-(5-methyltetrazol-1-yl)benzamide
—— 3-(3,4-dimethoxyphenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-1H-pyrazole-5-carboxamide —— C16H19N3O5S
3-(3,4-dimethoxyphenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-1H-pyrazole-5-carboxamide
—— [2-(dimethylamino)-2-oxoethyl] 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C19H23FN4O4S
[2-(dimethylamino)-2-oxoethyl] 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— (8R)-8-(4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8R)-8-(4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [(2R)-1-amino-1-oxopropan-2-yl] 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C18H21FN4O4S
[(2R)-1-amino-1-oxopropan-2-yl] 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— (8S)-1-(3-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13ClN4OS
(8S)-1-(3-chlorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(3-bromophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13BrN4OS
(8R)-1-(3-bromophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylacetamide —— C17H21FN4O2S
2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylacetamide
—— (5-phenyl-1,3-oxazol-2-yl)methyl (3S)-3-(carbamoylamino)-3-(2-chlorophenyl)propanoate —— C20H18ClN3O4
(5-phenyl-1,3-oxazol-2-yl)methyl (3S)-3-(carbamoylamino)-3-(2-chlorophenyl)propanoate
—— methyl 2-[[(3R)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C16H17N3O5S
methyl 2-[[(3R)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C14H17N5O3S2
N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— N-[(1R)-1-(4-ethylphenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C19H21N5OS
N-[(1R)-1-(4-ethylphenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— (8R)-1-(3-bromophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14BrN3O2S
(8R)-1-(3-bromophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (2R)-N-[2-[(2S)-butan-2-yl]pyrazol-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide —— C17H21N7OS
(2R)-N-[2-[(2S)-butan-2-yl]pyrazol-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide
—— (2S)-N-[2-[(2R)-butan-2-yl]pyrazol-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide —— C17H21N7OS
(2S)-N-[2-[(2R)-butan-2-yl]pyrazol-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide
—— N-[(3-chlorophenyl)methyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C16H14ClN5OS
N-[(3-chlorophenyl)methyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— N-(5-chloro-2-nitrophenyl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C15H11ClN6O3S
N-(5-chloro-2-nitrophenyl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— N-[(1R)-1-(3,4-dimethylphenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C19H21N5OS
N-[(1R)-1-(3,4-dimethylphenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C18H17N5O3S
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— 6-Methyl-2-[(1-phenyltetrazol-5-yl)sulfanylmethyl]imidazo[1,2-a]pyridine —— C16H14N6S
6-Methyl-2-[(1-phenyltetrazol-5-yl)sulfanylmethyl]imidazo[1,2-a]pyridine
—— (2R)-1-(2,3-dihydro-1H-inden-5-yl)-2-(1-phenyltetrazol-5-yl)sulfanylpropan-1-one —— C19H18N4OS
(2R)-1-(2,3-dihydro-1H-inden-5-yl)-2-(1-phenyltetrazol-5-yl)sulfanylpropan-1-one
—— (2-oxo-2-thiophen-2-ylethyl) (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C19H14ClFN2O3S
(2-oxo-2-thiophen-2-ylethyl) (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— 2-[[3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-1,3-benzoxazole —— C17H13N3O3S
2-[[3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-1,3-benzoxazole
—— [2-[[(2S)-3-methylbutan-2-yl]amino]-2-oxoethyl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C20H23ClFN3O3
[2-[[(2S)-3-methylbutan-2-yl]amino]-2-oxoethyl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— (8S)-1-(3-bromophenyl)-8-(1,5-dimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H16BrN5OS
(8S)-1-(3-bromophenyl)-8-(1,5-dimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [2-(methylamino)-2-oxoethyl] (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate —— C19H17N5O3
[2-(methylamino)-2-oxoethyl] (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate