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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[[(1R,9aS)-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizin-1-yl]methylamino]-1,5-dimethyl-2-phenylpyrazol-3-one —— C21H30N4O
4-[[(1R,9aS)-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizin-1-yl]methylamino]-1,5-dimethyl-2-phenylpyrazol-3-one
—— [2-Oxo-2-(2-oxopyrrolidin-1-yl)ethyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C21H19N3O4S
[2-Oxo-2-(2-oxopyrrolidin-1-yl)ethyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— 2-[2-[(3S)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl]imidazol-1-yl]acetamide —— C19H22N6O2
2-[2-[(3S)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl]imidazol-1-yl]acetamide
—— Cyanomethyl 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C17H13N3O2S
Cyanomethyl 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— [2-(2-Methoxyethylamino)-2-oxoethyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C20H21N3O4S
[2-(2-Methoxyethylamino)-2-oxoethyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— [(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C21H21N3O3S
[(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— [(1R)-2-oxocyclohexyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C21H20N2O3S
[(1R)-2-oxocyclohexyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— (4S)-4-benzyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-one —— C16H18N2O2
(4S)-4-benzyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-one
—— [(1S)-2-oxocyclohexyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C21H20N2O3S
[(1S)-2-oxocyclohexyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— [2-oxo-2-[[(2R)-pentan-2-yl]amino]ethyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C22H25N3O3S
[2-oxo-2-[[(2R)-pentan-2-yl]amino]ethyl] 1-benzyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-naphthalen-2-ylacetate —— C25H23N3O3
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-naphthalen-2-ylacetate
—— (4R)-4-benzyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-one —— C16H18N2O2
(4R)-4-benzyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-one
—— 3-(4-methoxyanilino)-2-phenyl-5-[(6-sulfanylidenecyclohexa-2,4-dien-1-ylidene)methyl]imidazol-4-olate —— C23H18N3O2S-
3-(4-methoxyanilino)-2-phenyl-5-[(6-sulfanylidenecyclohexa-2,4-dien-1-ylidene)methyl]imidazol-4-olate
—— (2R)-2-(2-pyridin-2-ylethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide —— C20H23N7O
(2R)-2-(2-pyridin-2-ylethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide
—— 2-(3-methoxyphenyl)-N-[(1R)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide —— C19H17N5O4
2-(3-methoxyphenyl)-N-[(1R)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
—— 2-(3-methoxyphenyl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide —— C20H19N5O3
2-(3-methoxyphenyl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
—— (4S)-4-benzyl-1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-one —— C17H20N2OS
(4S)-4-benzyl-1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-one
—— (2R)-2-(2-propan-2-ylimidazol-1-yl)-N-[2-(2-pyrimidin-2-yl-1,3-thiazol-4-yl)ethyl]propanamide —— C18H22N6OS
(2R)-2-(2-propan-2-ylimidazol-1-yl)-N-[2-(2-pyrimidin-2-yl-1,3-thiazol-4-yl)ethyl]propanamide
—— 3-phenyl-5-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole —— C22H22N6O
3-phenyl-5-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole
—— (2S)-2-(2-propan-2-ylimidazol-1-yl)-N-[2-(2-pyrimidin-2-yl-1,3-thiazol-4-yl)ethyl]propanamide —— C18H22N6OS
(2S)-2-(2-propan-2-ylimidazol-1-yl)-N-[2-(2-pyrimidin-2-yl-1,3-thiazol-4-yl)ethyl]propanamide
—— (4R)-1-[2-(dimethylamino)ethyl]-4-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-5-carbonyl)pyrrolidin-2-one —— C21H27N5O2
(4R)-1-[2-(dimethylamino)ethyl]-4-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-5-carbonyl)pyrrolidin-2-one
—— (2R)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C17H26N4OS
(2R)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— 2-({[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl}methyl)quinazolin-4-ol —— C18H15N5O2S
2-({[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl}methyl)quinazolin-4-ol
—— 2-[(1S)-1-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one —— C19H19N5O2S2
2-[(1S)-1-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one
—— (2S)-2-(2-pyridin-2-ylethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide —— C20H23N7O
(2S)-2-(2-pyridin-2-ylethyl)-N-[3-(tetrazol-1-yl)phenyl]piperidine-1-carboxamide
—— (4R)-4-benzyl-1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-one —— C17H20N2OS
(4R)-4-benzyl-1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-one
—— (4S)-1-[2-(dimethylamino)ethyl]-4-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-5-carbonyl)pyrrolidin-2-one —— C21H27N5O2
(4S)-1-[2-(dimethylamino)ethyl]-4-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-5-carbonyl)pyrrolidin-2-one
—— 3-phenyl-5-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole —— C22H22N6O
3-phenyl-5-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole
—— 2-(3-methoxyphenyl)-N-[(1S)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide —— C19H17N5O4
2-(3-methoxyphenyl)-N-[(1S)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
—— 3-[3-methoxy-5-(tetrazol-1-yl)phenyl]-1-methyl-1-[2-[(2S)-oxan-2-yl]ethyl]urea —— C17H24N6O3
3-[3-methoxy-5-(tetrazol-1-yl)phenyl]-1-methyl-1-[2-[(2S)-oxan-2-yl]ethyl]urea
—— (3R)-3-(3,5-dimethylpyrazol-1-yl)-N-[3-(1,3-oxazol-5-yl)phenyl]pyrrolidine-1-carboxamide —— C19H21N5O2
(3R)-3-(3,5-dimethylpyrazol-1-yl)-N-[3-(1,3-oxazol-5-yl)phenyl]pyrrolidine-1-carboxamide
—— 2-(3-methoxyphenyl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide —— C20H19N5O3
2-(3-methoxyphenyl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
—— 1-(2-propylpyrazol-3-yl)-3-[(2R)-1-thiophen-3-ylpropan-2-yl]urea —— C14H20N4OS
1-(2-propylpyrazol-3-yl)-3-[(2R)-1-thiophen-3-ylpropan-2-yl]urea
—— (3S)-3-(3,5-dimethylpyrazol-1-yl)-N-[3-(1,3-oxazol-5-yl)phenyl]pyrrolidine-1-carboxamide —— C19H21N5O2
(3S)-3-(3,5-dimethylpyrazol-1-yl)-N-[3-(1,3-oxazol-5-yl)phenyl]pyrrolidine-1-carboxamide
—— (6R)-1-benzyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,4-diazepan-6-ol —— C20H22N4O2
(6R)-1-benzyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,4-diazepan-6-ol
—— (2S)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C17H26N4OS
(2S)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— 1-(2-propylpyrazol-3-yl)-3-[(2S)-1-thiophen-3-ylpropan-2-yl]urea —— C14H20N4OS
1-(2-propylpyrazol-3-yl)-3-[(2S)-1-thiophen-3-ylpropan-2-yl]urea
—— 2-[(1R)-1-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3H-quinazolin-4-one —— C19H17N5O2S
2-[(1R)-1-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3H-quinazolin-4-one
—— 2-ethanimidoyl-4-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-oxobutanenitrile —— C15H15N5O2S
2-ethanimidoyl-4-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-oxobutanenitrile
—— 3-[3-methoxy-5-(tetrazol-1-yl)phenyl]-1-methyl-1-[2-[(2R)-oxan-2-yl]ethyl]urea —— C17H24N6O3
3-[3-methoxy-5-(tetrazol-1-yl)phenyl]-1-methyl-1-[2-[(2R)-oxan-2-yl]ethyl]urea
—— 1-[2-(dimethylamino)ethyl]-1-[[(2S)-oxolan-2-yl]methyl]-3-(4-pyrazol-1-ylphenyl)urea —— C19H27N5O2
1-[2-(dimethylamino)ethyl]-1-[[(2S)-oxolan-2-yl]methyl]-3-(4-pyrazol-1-ylphenyl)urea
—— 1-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]-3-[4-(tetrazol-1-yl)phenyl]urea —— C20H23N7O
1-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]-3-[4-(tetrazol-1-yl)phenyl]urea
—— (3S)-3-(morpholine-4-carbonyl)-N-[3-(1,3-oxazol-5-yl)phenyl]piperidine-1-carboxamide —— C20H24N4O4
(3S)-3-(morpholine-4-carbonyl)-N-[3-(1,3-oxazol-5-yl)phenyl]piperidine-1-carboxamide
—— 2-(5-Oxo-4-phenyltetrazol-1-yl)acetate —— C9H7N4O3-
2-(5-Oxo-4-phenyltetrazol-1-yl)acetate
—— N-[[(3R)-1-[[1-(2-fluorophenyl)pyrazol-4-yl]methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide —— C22H24FN5O
N-[[(3R)-1-[[1-(2-fluorophenyl)pyrazol-4-yl]methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide
—— 2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one —— C18H17N5O2S2
2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one
—— N-[[(3S)-1-[[1-(2-fluorophenyl)pyrazol-4-yl]methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide —— C22H24FN5O
N-[[(3S)-1-[[1-(2-fluorophenyl)pyrazol-4-yl]methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide
—— (2S)-N-[(2S)-2-cyano-3-methylbutan-2-yl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C18H23N5O2S
(2S)-N-[(2S)-2-cyano-3-methylbutan-2-yl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(2-fluorophenyl)methyl]-3-[(3S)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl]propanamide —— C20H26FN3OS
N-[(2-fluorophenyl)methyl]-3-[(3S)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl]propanamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-methylacetamide —— C16H20N4O4S2
N-[(3R)-1,1-dioxothiolan-3-yl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-methylacetamide