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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-chloro-N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide —— C13H15ClN4O2S2
2-chloro-N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide
—— (8R)-1-(4-chlorophenyl)-8-thiophen-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H12ClN3OS2
(8R)-1-(4-chlorophenyl)-8-thiophen-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[2-[(3S)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C19H21N5O4S
N-[2-[(3S)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— (8S)-1-(4-chlorophenyl)-8-thiophen-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H12ClN3OS2
(8S)-1-(4-chlorophenyl)-8-thiophen-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(3-fluorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14FN3O2S
(8S)-1-(3-fluorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C20H28N4O2
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— (2R)-N-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-2-phenyl-2-(tetrazol-1-yl)acetamide —— C20H19N7O
(2R)-N-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-2-phenyl-2-(tetrazol-1-yl)acetamide
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide —— C16H22N6O
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide —— C20H28N4O
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide —— C16H22N6O
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide —— C20H28N4O
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide
—— (8R)-1-(3-fluorophenyl)-8-(2,3,4-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H20FN3O4S
(8R)-1-(3-fluorophenyl)-8-(2,3,4-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(3-fluorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14FN3O2S
(8R)-1-(3-fluorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (2R)-N-[4-(3,5-dimethylpyrazol-1-yl)-3-methoxyphenyl]-2-phenyl-2-(tetrazol-1-yl)acetamide —— C21H21N7O2
(2R)-N-[4-(3,5-dimethylpyrazol-1-yl)-3-methoxyphenyl]-2-phenyl-2-(tetrazol-1-yl)acetamide
—— (8S)-1-(3-fluorophenyl)-8-(2,3,4-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H20FN3O4S
(8S)-1-(3-fluorophenyl)-8-(2,3,4-trimethoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(4-methylsulfonylphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S2
(8R)-8-(4-methylsulfonylphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(3-methoxyphenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H16N4O2S
(8S)-1-(3-methoxyphenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[[(1R,2R,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C21H25N3O2
N-[[(1R,2R,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— (8R)-1-phenyl-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C13H10F3N3OS
(8R)-1-phenyl-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(3-methoxyphenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H16N4O2S
(8R)-1-(3-methoxyphenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[2-methoxy-5-[(8S)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]phenoxy]acetamide —— C22H22N4O5S
2-[2-methoxy-5-[(8S)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]phenoxy]acetamide
—— (3R)-3-(4-hydroxy-6-methyl-2-oxo-1H-pyridin-3-yl)-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]propanoic acid —— C19H19N3O5
(3R)-3-(4-hydroxy-6-methyl-2-oxo-1H-pyridin-3-yl)-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]propanoic acid
—— (8S)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-fluorophenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H16FN5OS
(8S)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-fluorophenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C20H28N4O2
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— (8S)-8-(3-hydroxy-4-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8S)-8-(3-hydroxy-4-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-methyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-5-phenylpyrazole-3-carboxamide —— C17H18N6O2
2-methyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-5-phenylpyrazole-3-carboxamide
—— (8R)-8-(3-hydroxy-4-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8R)-8-(3-hydroxy-4-methoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[2-methoxy-5-[(8R)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]phenoxy]acetamide —— C22H22N4O5S
2-[2-methoxy-5-[(8R)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]phenoxy]acetamide
—— (8R)-1-(3-bromophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16BrN3O3S
(8R)-1-(3-bromophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[(1R)-1-[(4-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-quinazolin-4-one —— C18H15N5OS
2-[(1R)-1-[(4-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-quinazolin-4-one
—— 2-methyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-5-phenylpyrazole-3-carboxamide —— C17H18N6O2
2-methyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-5-phenylpyrazole-3-carboxamide
—— (8S)-1-(3-bromophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16BrN3O3S
(8S)-1-(3-bromophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (Z)-3-(furan-3-yl)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]prop-2-enenitrile —— C17H12N2OS
(Z)-3-(furan-3-yl)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]prop-2-enenitrile
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 4-methylsulfonylbenzoate —— C18H15NO5S
(5-Phenyl-1,3-oxazol-2-yl)methyl 4-methylsulfonylbenzoate
—— (2S)-2-ethanimidoyl-4-[[5-methyl-4-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-3-oxobutanenitrile —— C16H17N5OS
(2S)-2-ethanimidoyl-4-[[5-methyl-4-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-3-oxobutanenitrile
—— (3S)-3-(4-hydroxy-6-methyl-2-oxo-1H-pyridin-3-yl)-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]propanoic acid —— C19H19N3O5
(3S)-3-(4-hydroxy-6-methyl-2-oxo-1H-pyridin-3-yl)-3-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]propanoic acid
—— (8S)-8-(4-methylsulfonylphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S2
(8S)-8-(4-methylsulfonylphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (5E)-5-(2-furylmethylene)-2-(4-methylphenyl)[1,3]thiazolo[3,2-b][1,2,4]triazol-6(5H)-one —— C16H11N3O2S
(5E)-5-(2-furylmethylene)-2-(4-methylphenyl)[1,3]thiazolo[3,2-b][1,2,4]triazol-6(5H)-one
—— (8R)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-fluorophenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H16FN5OS
(8R)-8-(1,5-dimethylpyrazol-4-yl)-1-(3-fluorophenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (2S)-2-(3-chloro-4-fluorophenoxy)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide —— C20H19ClFN3O3
(2S)-2-(3-chloro-4-fluorophenoxy)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide
—— N-[[(1R,2S,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C21H25N3O2
N-[[(1R,2S,4R)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 4-ethoxybenzoate —— C23H25N3O5
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 4-ethoxybenzoate
—— (8S)-1-phenyl-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C13H10F3N3OS
(8S)-1-phenyl-8-(trifluoromethyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 4-ethoxybenzoate —— C22H23N3O4
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 4-ethoxybenzoate
—— 2-bromo-N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide —— C13H15BrN4O2S2
2-bromo-N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide
—— (3S)-1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-oxopyrrolidine-3-carboxylic acid —— C16H17N3O4
(3S)-1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-5-oxopyrrolidine-3-carboxylic acid
—— N-[(3R)-1,1-dioxothiolan-3-yl]-2-[(4-methoxyphenyl)methylamino]-1,3-thiazole-4-carboxamide —— C16H19N3O4S2
N-[(3R)-1,1-dioxothiolan-3-yl]-2-[(4-methoxyphenyl)methylamino]-1,3-thiazole-4-carboxamide
—— 3,5-dimethyl-N-(tricyclo[3.3.1.1~3,7~]dec-1-ylmethyl)-1,2-oxazole-4-carboxamide —— C17H24N2O2
3,5-dimethyl-N-(tricyclo[3.3.1.1~3,7~]dec-1-ylmethyl)-1,2-oxazole-4-carboxamide
—— 4-[(8R)-1-(4-fluorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14FN3O3S
4-[(8R)-1-(4-fluorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— 2-bromo-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide —— C13H15BrN4O2S2
2-bromo-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide