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中文名称 英文名称 CAS号 化学式 结构式图片
—— [2-oxo-2-(2-oxopyrrolidin-1-yl)ethyl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C19H17ClFN3O4
[2-oxo-2-(2-oxopyrrolidin-1-yl)ethyl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— [(2R)-1-(cyclopentylamino)-1-oxopropan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C21H23ClFN3O3
[(2R)-1-(cyclopentylamino)-1-oxopropan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— methyl 2-[[(3S)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C16H17N3O5S
methyl 2-[[(3S)-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carbonyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— (8S)-1-(4-chlorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14ClN3O2S
(8S)-1-(4-chlorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-(5-methyltetrazol-1-yl)benzamide —— C16H22N6O
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-(5-methyltetrazol-1-yl)benzamide
—— 3-Phenyl-5-(quinolin-2-ylsulfanylmethyl)-1,2,4-oxadiazole —— C18H13N3OS
3-Phenyl-5-(quinolin-2-ylsulfanylmethyl)-1,2,4-oxadiazole
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-5-(4-methoxyphenyl)-2-methylpyrazole-3-carboxamide —— C19H26N4O2
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-5-(4-methoxyphenyl)-2-methylpyrazole-3-carboxamide
—— 2-(1H-benzimidazol-2-ylsulfanyl)-N-[5-(4-chlorophenyl)-2-methylpyrazol-3-yl]acetamide —— C19H16ClN5OS
2-(1H-benzimidazol-2-ylsulfanyl)-N-[5-(4-chlorophenyl)-2-methylpyrazol-3-yl]acetamide
—— (3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate —— C21H18N2O4
(3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate
—— 3,4-dimethyl-2-(tetrazol-1-yl)-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]benzamide —— C18H18N8O
3,4-dimethyl-2-(tetrazol-1-yl)-N-[(1S)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]benzamide
—— (8S)-8-(4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8S)-8-(4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-8-(4-hydroxy-3-methoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H19N3O4S
(8S)-8-(4-hydroxy-3-methoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(3-methoxyphenyl)-8-(3-methoxy-4-propan-2-yloxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C23H25N3O4S
(8R)-1-(3-methoxyphenyl)-8-(3-methoxy-4-propan-2-yloxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [(1S)-2-oxocyclopentyl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C18H16ClFN2O3
[(1S)-2-oxocyclopentyl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— (8S)-1-(3-methoxyphenyl)-8-(3-methoxy-4-propan-2-yloxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C23H25N3O4S
(8S)-1-(3-methoxyphenyl)-8-(3-methoxy-4-propan-2-yloxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [3-(2-Methylphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate —— C22H20N2O4
[3-(2-Methylphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-5-(4-methoxyphenyl)-2-methylpyrazole-3-carboxamide —— C19H26N4O2
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-5-(4-methoxyphenyl)-2-methylpyrazole-3-carboxamide
—— (8R)-1-(4-chlorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14ClN3O2S
(8R)-1-(4-chlorophenyl)-8-(3-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [(2R)-1-oxo-1-piperidin-1-ylpropan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C21H23ClFN3O3
[(2R)-1-oxo-1-piperidin-1-ylpropan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— [(2S)-1-(cyclopentylamino)-1-oxopropan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C21H23ClFN3O3
[(2S)-1-(cyclopentylamino)-1-oxopropan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— [(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl] (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate —— C22H21N5O3
[(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl] (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate
—— (8S)-1-(3-bromophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13BrN4OS
(8S)-1-(3-bromophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide —— C17H18N6O3
N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
—— N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide —— C17H18N6O3
N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-4-(2-propan-2-yltetrazol-5-yl)benzamide —— C15H19N5O3S
N-[(3S)-1,1-dioxothiolan-3-yl]-4-(2-propan-2-yltetrazol-5-yl)benzamide
—— (8S)-1-(4-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H18ClN5OS
(8S)-1-(4-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [(2S)-3-oxobutan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C17H16ClFN2O3
[(2S)-3-oxobutan-2-yl] (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— (8R)-1-(4-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H18ClN5OS
(8R)-1-(4-chlorophenyl)-8-(1,3,5-trimethylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(3R)-1,1-dioxothiolan-3-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C17H21N3O4S
N-[(3R)-1,1-dioxothiolan-3-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— (4-chlorophenyl)methyl (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate —— C23H17ClN4O2
(4-chlorophenyl)methyl (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate
—— (8R)-8-(3-chloro-4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8R)-8-(3-chloro-4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-8-(4-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H15N3O2S
(8S)-8-(4-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 3-(3,5-dimethylpyrazol-1-yl)-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]benzamide —— C18H20N6O2
3-(3,5-dimethylpyrazol-1-yl)-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]benzamide
—— 3-(3,5-dimethylpyrazol-1-yl)-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]benzamide —— C18H20N6O2
3-(3,5-dimethylpyrazol-1-yl)-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]benzamide
—— (2-morpholin-4-yl-2-oxoethyl) (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate —— C22H21N5O4
(2-morpholin-4-yl-2-oxoethyl) (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]prop-2-enoate
—— (8R)-8-(4-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H15N3O2S
(8R)-8-(4-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— methyl 2-[[2-[4-[(1R)-2,2-dichlorocyclopropyl]phenoxy]-2-methylpropanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C19H20Cl2N2O4S
methyl 2-[[2-[4-[(1R)-2,2-dichlorocyclopropyl]phenoxy]-2-methylpropanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— (8R)-1-(3-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8R)-1-(3-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-8-(3-chloro-4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8S)-8-(3-chloro-4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— methyl 2-[[2-[4-[(1S)-2,2-dichlorocyclopropyl]phenoxy]-2-methylpropanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C19H20Cl2N2O4S
methyl 2-[[2-[4-[(1S)-2,2-dichlorocyclopropyl]phenoxy]-2-methylpropanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— N-[(3S)-1,1-dioxothiolan-3-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C17H21N3O4S
N-[(3S)-1,1-dioxothiolan-3-yl]-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3,4-dimethyl-2-(tetrazol-1-yl)benzamide —— C17H24N6O
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3,4-dimethyl-2-(tetrazol-1-yl)benzamide
—— (4R)-4-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-4,8-dihydro-1H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C15H12FN5OS
(4R)-4-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-4,8-dihydro-1H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-(4-chlorophenyl)-4-methyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,3-thiazole-5-carboxamide —— C17H16ClN5O2S
2-(4-chlorophenyl)-4-methyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,3-thiazole-5-carboxamide
—— (8S)-1-(3-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8S)-1-(3-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-chloro-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide —— C13H15ClN4O2S2
2-chloro-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-5-propan-2-yl-1,3-thiazole-4-carboxamide
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3,4-dimethyl-2-(tetrazol-1-yl)benzamide —— C17H24N6O
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3,4-dimethyl-2-(tetrazol-1-yl)benzamide
—— (4S)-4-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-4,8-dihydro-1H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C15H12FN5OS
(4S)-4-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-4,8-dihydro-1H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-(4-chlorophenyl)-4-methyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,3-thiazole-5-carboxamide —— C17H16ClN5O2S
2-(4-chlorophenyl)-4-methyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,3-thiazole-5-carboxamide
—— N-[2-[(3R)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C19H21N5O4S
N-[2-[(3R)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide