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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-N-benzyl-N-methyl-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide —— C18H19N5OS
(2R)-N-benzyl-N-methyl-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide
—— N-(1-adamantylmethyl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C20H25N5OS
N-(1-adamantylmethyl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— [4-Amino-6-(2-ethylanilino)-1,3,5-triazin-2-yl]methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate —— C18H20N6O2S
[4-Amino-6-(2-ethylanilino)-1,3,5-triazin-2-yl]methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate
—— N-[(1R)-1-(3-chlorophenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C17H16ClN5OS
N-[(1R)-1-(3-chlorophenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— (7R)-7-methyl-2-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H18N6OS2
(7R)-7-methyl-2-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (E)-3-(furan-2-yl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]prop-2-enamide —— C20H20N4O2
(E)-3-(furan-2-yl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]prop-2-enamide
—— 4-[(8R)-1-(3-fluorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14FN3O3S
4-[(8R)-1-(3-fluorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]cyclobutanecarboxamide —— C18H22N4O
N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]cyclobutanecarboxamide
—— 3-(3,5-dimethylpyrazol-1-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]benzamide —— C16H19N3O3S
3-(3,5-dimethylpyrazol-1-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]benzamide
—— N-[(4R)-2,2-dimethyloxan-4-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C18H23N3O3
N-[(4R)-2,2-dimethyloxan-4-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— (8S)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H19N3O4S
(8S)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [2-Oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] 2-(4-fluorophenyl)acetate —— C22H19FN2O3S
[2-Oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] 2-(4-fluorophenyl)acetate
—— 5-(2-chlorophenyl)-N-[(4S)-2,2-dimethyloxan-4-yl]-2-methyl-1,3-thiazole-4-carboxamide —— C18H21ClN2O2S
5-(2-chlorophenyl)-N-[(4S)-2,2-dimethyloxan-4-yl]-2-methyl-1,3-thiazole-4-carboxamide
—— N-[2-[(3R)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C19H21N5O4S
N-[2-[(3R)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— 4-[(8S)-1-(3-fluorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14FN3O3S
4-[(8S)-1-(3-fluorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— 4-[(8R)-1-(4-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14ClN3O3S
4-[(8R)-1-(4-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— N-[2-[(3S)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C19H21N5O4S
N-[2-[(3S)-1,1-dioxothiolan-3-yl]-5-methylpyrazol-3-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— 2-chloro-4-[(4R)-6-methyl-1-phenyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol —— C18H14ClN3OS
2-chloro-4-[(4R)-6-methyl-1-phenyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol
—— 4-[(8S)-1-(4-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14ClN3O3S
4-[(8S)-1-(4-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— (8R)-1-(4-methoxyphenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H17N5O2S
(8R)-1-(4-methoxyphenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[(4S)-2,2-dimethyloxan-4-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C18H23N3O3
N-[(4S)-2,2-dimethyloxan-4-yl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— 5-(3-chlorophenyl)-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-methylpyrazole-3-carboxamide —— C18H23ClN4O
5-(3-chlorophenyl)-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-methylpyrazole-3-carboxamide
—— (8R)-1-(3-chlorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H14ClN5OS
(8R)-1-(3-chlorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 1-[(3R)-1,1-dioxothiolan-3-yl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3,5-dimethylpyrazole-4-carboxamide —— C17H28N4O3S
1-[(3R)-1,1-dioxothiolan-3-yl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-3,5-dimethylpyrazole-4-carboxamide
—— 5-(3-chlorophenyl)-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-methylpyrazole-3-carboxamide —— C18H23ClN4O
5-(3-chlorophenyl)-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-methylpyrazole-3-carboxamide
—— (8S)-8-(3-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8S)-8-(3-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 4-methyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-1,3-thiazole-5-carboxamide —— C17H17N5O2S
4-methyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-1,3-thiazole-5-carboxamide
—— 4-methyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-1,3-thiazole-5-carboxamide —— C17H17N5O2S
4-methyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-1,3-thiazole-5-carboxamide
—— (8S)-8-(3-chloro-4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8S)-8-(3-chloro-4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(4-fluorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13FN4OS
(8S)-1-(4-fluorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-1-(3-chlorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H14ClN5OS
(8S)-1-(3-chlorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(4-fluorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H13FN4OS
(8R)-1-(4-fluorophenyl)-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[5-[(8R)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]-2-methoxyphenoxy]acetamide —— C21H19ClN4O4S
2-[5-[(8R)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]-2-methoxyphenoxy]acetamide
—— 1-[(3R)-1,1-dioxothiolan-3-yl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3,5-dimethylpyrazole-4-carboxamide —— C17H28N4O3S
1-[(3R)-1,1-dioxothiolan-3-yl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-3,5-dimethylpyrazole-4-carboxamide
—— (8R)-8-(3-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8R)-8-(3-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (2-Thiophen-2-yl-1,3-oxazol-4-yl)methyl 2-(4-fluorophenyl)acetate —— C16H12FNO3S
(2-Thiophen-2-yl-1,3-oxazol-4-yl)methyl 2-(4-fluorophenyl)acetate
—— (8S)-1-(4-fluorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H14FN5OS
(8S)-1-(4-fluorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [4-(Tetrazol-1-yl)phenyl] 2-(2-fluorophenoxy)acetate —— C15H11FN4O3
[4-(Tetrazol-1-yl)phenyl] 2-(2-fluorophenoxy)acetate
—— (8R)-8-(3-chloro-4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8R)-8-(3-chloro-4-hydroxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[5-[(8S)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]-2-methoxyphenoxy]acetamide —— C21H19ClN4O4S
2-[5-[(8S)-1-(3-chlorophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]-2-methoxyphenoxy]acetamide
—— (8R)-1-(4-fluorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C16H14FN5OS
(8R)-1-(4-fluorophenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2-ethoxybenzoate —— C21H21N3O4
[2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2-ethoxybenzoate
—— N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide —— C19H22N6O2
N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide
—— N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide —— C19H22N6O2
N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-2-phenyl-5-propan-2-ylpyrazole-3-carboxamide
—— [4-(Tetrazol-1-yl)phenyl] 2-(3,4,5-trimethoxyphenyl)acetate —— C18H18N4O5
[4-(Tetrazol-1-yl)phenyl] 2-(3,4,5-trimethoxyphenyl)acetate
—— (8R)-1-(4-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16ClN3O3S
(8R)-1-(4-chlorophenyl)-8-(3-hydroxy-4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— [2-[[3,5-Dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 3-fluorobenzoate —— C21H20FN3O3
[2-[[3,5-Dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 3-fluorobenzoate
—— (2R)-2-phenyl-2-(tetrazol-1-yl)-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]acetamide —— C17H14N8O
(2R)-2-phenyl-2-(tetrazol-1-yl)-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]acetamide
—— methyl 2-[[(3R)-3-(4-chlorophenyl)-4-pyrrol-1-ylbutanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate —— C20H20ClN3O3S
methyl 2-[[(3R)-3-(4-chlorophenyl)-4-pyrrol-1-ylbutanoyl]amino]-5-methyl-1,3-thiazole-4-carboxylate
—— (8S)-1-(3-bromophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14BrN3O2S
(8S)-1-(3-bromophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one