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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8R)-8-(1,5-dimethylpyrazol-4-yl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H17N5OS
(8R)-8-(1,5-dimethylpyrazol-4-yl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-(3-fluorophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H16FN3O3S
(8R)-1-(3-fluorophenyl)-8-(4-hydroxy-3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(4R)-2,2-dimethyloxan-4-yl]acetamide —— C19H24ClN3O2
2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(4R)-2,2-dimethyloxan-4-yl]acetamide
—— 3,5-dimethyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,2-oxazole-4-carboxamide —— C12H15N5O3
3,5-dimethyl-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,2-oxazole-4-carboxamide
—— (8S)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H21N3O5S
(8S)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]acetamide —— C19H22N6O2
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]acetamide
—— (8R)-1-(3-fluorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14FN3O2S
(8R)-1-(3-fluorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C16H18ClN3O3S
2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— 4-[(8S)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C20H17N3O4S
4-[(8S)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— (8S)-8-(4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8S)-8-(4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (2-bromo-5-propan-2-yl-1,3-thiazol-4-yl)-[4-[(3S)-1,1-dioxothiolan-3-yl]piperazin-1-yl]methanone —— C15H22BrN3O3S2
(2-bromo-5-propan-2-yl-1,3-thiazol-4-yl)-[4-[(3S)-1,1-dioxothiolan-3-yl]piperazin-1-yl]methanone
—— 2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(4S)-2,2-dimethyloxan-4-yl]acetamide —— C19H24ClN3O2
2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(4S)-2,2-dimethyloxan-4-yl]acetamide
—— (8R)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C21H21N3O5S
(8R)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 3,5-dimethyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,2-oxazole-4-carboxamide —— C12H15N5O3
3,5-dimethyl-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]-1,2-oxazole-4-carboxamide
—— N-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-2-(2-formylphenoxy)acetamide —— C20H19N3O4
N-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-2-(2-formylphenoxy)acetamide
—— 2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C18H23N3O3
2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]acetamide —— C19H22N6O2
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-[(2R)-oxolan-2-yl]-1H-1,2,4-triazol-3-yl]acetamide
—— 4-[(8R)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C20H17N3O4S
4-[(8R)-1-(3-methoxyphenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— (8S)-1-(3-fluorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H14FN3O2S
(8S)-1-(3-fluorophenyl)-8-(4-hydroxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(4-hydroxy-3-methoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H19N3O4S
(8R)-8-(4-hydroxy-3-methoxyphenyl)-1-(4-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— 2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C18H23N3O3
2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide —— C16H18ClN3O3S
2-[3-(4-chlorophenyl)-5-methyl-1H-pyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide
—— (2-bromo-5-propan-2-yl-1,3-thiazol-4-yl)-[4-[(3R)-1,1-dioxothiolan-3-yl]piperazin-1-yl]methanone —— C15H22BrN3O3S2
(2-bromo-5-propan-2-yl-1,3-thiazol-4-yl)-[4-[(3R)-1,1-dioxothiolan-3-yl]piperazin-1-yl]methanone
—— (8R)-8-(4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C19H17N3O3S
(8R)-8-(4-hydroxyphenyl)-1-(3-methoxyphenyl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-1-phenyl-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H14N4OS
(8R)-1-phenyl-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8S)-8-(3-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H15N3O2S
(8S)-8-(3-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-(2-pyrrol-1-yl-1,3-thiazol-4-yl)acetamide —— C16H22N4OS
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-(2-pyrrol-1-yl-1,3-thiazol-4-yl)acetamide
—— (8S)-1-(4-methoxyphenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H17N5O2S
(8S)-1-(4-methoxyphenyl)-8-(1-methylpyrazol-4-yl)-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— (8R)-8-(3-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C18H15N3O2S
(8R)-8-(3-hydroxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide —— C15H15N7O2S
N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide
—— 2-chloro-4-[(4S)-6-methyl-1-phenyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol —— C18H14ClN3OS
2-chloro-4-[(4S)-6-methyl-1-phenyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]phenol
—— 5-(2-chlorophenyl)-N-[(4R)-2,2-dimethyloxan-4-yl]-2-methyl-1,3-thiazole-4-carboxamide —— C18H21ClN2O2S
5-(2-chlorophenyl)-N-[(4R)-2,2-dimethyloxan-4-yl]-2-methyl-1,3-thiazole-4-carboxamide
—— 1-[2,5-Dimethyl-1-(1,3-thiazol-2-yl)pyrrol-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylethanone —— C18H16N6OS2
1-[2,5-Dimethyl-1-(1,3-thiazol-2-yl)pyrrol-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylethanone
—— (8S)-1-phenyl-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C17H14N4OS
(8S)-1-phenyl-8-pyridin-3-yl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-(2-pyrrol-1-yl-1,3-thiazol-4-yl)acetamide —— C16H22N4OS
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-(2-pyrrol-1-yl-1,3-thiazol-4-yl)acetamide
—— 5-[(1R)-1-(2-chlorophenyl)ethyl]sulfanyl-1-phenyltetrazole —— C15H13ClN4S
5-[(1R)-1-(2-chlorophenyl)ethyl]sulfanyl-1-phenyltetrazole
—— (2R)-N-[(1S,2S)-2-methylcyclohexyl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide —— C17H23N5OS
(2R)-N-[(1S,2S)-2-methylcyclohexyl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide
—— N-[(4R)-2,2-dimethyloxan-4-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C19H24FN3O2
N-[(4R)-2,2-dimethyloxan-4-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide —— C15H15N7O2S
N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide
—— 4-[(8S)-1-(3-bromophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14BrN3O3S
4-[(8S)-1-(3-bromophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— 3-(3,5-dimethylpyrazol-1-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]benzamide —— C16H19N3O3S
3-(3,5-dimethylpyrazol-1-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]benzamide
—— N-(6-fluoro-1,3-benzothiazol-2-yl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C16H11FN6OS2
N-(6-fluoro-1,3-benzothiazol-2-yl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— 4-[(8R)-1-(3-bromophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid —— C19H14BrN3O3S
4-[(8R)-1-(3-bromophenyl)-5-oxo-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-8-yl]benzoic acid
—— (8R)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one —— C20H19N3O4S
(8R)-8-(4-hydroxy-3,5-dimethoxyphenyl)-1-phenyl-4,8-dihydroimidazo[4,5-e][1,4]thiazepin-5-one
—— Ethyl 4-[2-(1-phenyltetrazol-5-yl)sulfanylacetyl]piperazine-1-carboxylate —— C16H20N6O3S
Ethyl 4-[2-(1-phenyltetrazol-5-yl)sulfanylacetyl]piperazine-1-carboxylate
—— N-[(2R)-butan-2-yl]-N-[(3S)-1,1-dioxothiolan-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C17H23N5O3S2
N-[(2R)-butan-2-yl]-N-[(3S)-1,1-dioxothiolan-3-yl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— N-[(4S)-2,2-dimethyloxan-4-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide —— C19H24FN3O2
N-[(4S)-2,2-dimethyloxan-4-yl]-2-[3-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]acetamide
—— 3-[3-[2-(1-Phenyltetrazol-5-yl)sulfanylacetyl]indol-1-yl]propanenitrile —— C20H16N6OS
3-[3-[2-(1-Phenyltetrazol-5-yl)sulfanylacetyl]indol-1-yl]propanenitrile
—— 2-(4-Chlorophenyl)-4-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-thiazole —— C17H12ClN5S2
2-(4-Chlorophenyl)-4-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-thiazole
—— (2S)-N-(1-cyanocyclohexyl)-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide —— C17H20N6OS
(2S)-N-(1-cyanocyclohexyl)-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide