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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[(3R)-3-(1-methylimidazol-2-yl)piperidin-1-yl]ethanone —— C22H27N5O
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[(3R)-3-(1-methylimidazol-2-yl)piperidin-1-yl]ethanone
—— (6R)-5-[5-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C18H17N5O4
(6R)-5-[5-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— N-[(1R)-1-phenylethyl]-3-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propanamide —— C23H26N4O
N-[(1R)-1-phenylethyl]-3-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propanamide
—— (6R)-1-benzyl-4-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-1,4-diazepan-6-ol —— C22H25ClN4O
(6R)-1-benzyl-4-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-1,4-diazepan-6-ol
—— (3S)-3-(methylsulfonylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide —— C17H22N4O3S
(3S)-3-(methylsulfonylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide
—— [2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 5-chloro-2-hydroxybenzoate —— C19H16ClN3O4
[2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 5-chloro-2-hydroxybenzoate
—— (2S)-N-[2-methyl-3-(4-methyl-1,2,4-triazol-3-yl)phenyl]-2-pyridin-2-ylpyrrolidine-1-carboxamide —— C20H22N6O
(2S)-N-[2-methyl-3-(4-methyl-1,2,4-triazol-3-yl)phenyl]-2-pyridin-2-ylpyrrolidine-1-carboxamide
—— 5-phenyl-3-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole —— C22H22N6O
5-phenyl-3-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole
—— (6S)-5-[5-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C18H17N5O4
(6S)-5-[5-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (2R)-N-[2-methyl-3-(4-methyl-1,2,4-triazol-3-yl)phenyl]-2-pyridin-2-ylpyrrolidine-1-carboxamide —— C20H22N6O
(2R)-N-[2-methyl-3-(4-methyl-1,2,4-triazol-3-yl)phenyl]-2-pyridin-2-ylpyrrolidine-1-carboxamide
—— N-[(1S)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide —— C13H23N5OS
N-[(1S)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
—— N-[(1S)-1-phenylethyl]-3-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propanamide —— C23H26N4O
N-[(1S)-1-phenylethyl]-3-(2-phenyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl)propanamide
—— (3R)-3-(methylsulfonylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide —— C17H22N4O3S
(3R)-3-(methylsulfonylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide
—— (2R)-N-(4-pyrazol-1-ylphenyl)-2-(2-pyridin-2-ylethyl)piperidine-1-carboxamide —— C22H25N5O
(2R)-N-(4-pyrazol-1-ylphenyl)-2-(2-pyridin-2-ylethyl)piperidine-1-carboxamide
—— 5-phenyl-3-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole —— C22H22N6O
5-phenyl-3-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]-1,2,4-oxadiazole
—— 1-[[(3R)-1,1-dioxothiolan-3-yl]methyl]-3-[4-(1H-pyrazol-4-yl)phenyl]urea —— C15H18N4O3S
1-[[(3R)-1,1-dioxothiolan-3-yl]methyl]-3-[4-(1H-pyrazol-4-yl)phenyl]urea
—— (2S)-N-(4-pyrazol-1-ylphenyl)-2-(2-pyridin-2-ylethyl)piperidine-1-carboxamide —— C22H25N5O
(2S)-N-(4-pyrazol-1-ylphenyl)-2-(2-pyridin-2-ylethyl)piperidine-1-carboxamide
—— 1-methyl-1-[(3R)-1-methylpyrrolidin-3-yl]-3-(2-phenyl-1,3-benzoxazol-5-yl)urea —— C20H22N4O2
1-methyl-1-[(3R)-1-methylpyrrolidin-3-yl]-3-(2-phenyl-1,3-benzoxazol-5-yl)urea
—— 1-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-3-(1,3,5-trimethylpyrazol-4-yl)urea —— C13H18N4O3
1-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-3-(1,3,5-trimethylpyrazol-4-yl)urea
—— N-[(1R)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide —— C13H23N5OS
N-[(1R)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
—— [2-[[3,5-Dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 5-chloro-2-hydroxybenzoate —— C21H20ClN3O4
[2-[[3,5-Dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 5-chloro-2-hydroxybenzoate
—— [2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2-oxochromene-3-carboxylate —— C22H17N3O5
[2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 2-oxochromene-3-carboxylate
—— 1-[2-[5-[(2R)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]-3-[2-(tetrazol-1-yl)phenyl]urea —— C16H18N8O3
1-[2-[5-[(2R)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]-3-[2-(tetrazol-1-yl)phenyl]urea
—— 3-[3-(Benzylsulfonylamino)phenyl]-5-methyl-1-phenylpyrazole-4-carboxylic acid —— C24H21N3O4S
3-[3-(Benzylsulfonylamino)phenyl]-5-methyl-1-phenylpyrazole-4-carboxylic acid
—— 1-[2-[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]-3-[2-(tetrazol-1-yl)phenyl]urea —— C16H18N8O3
1-[2-[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]-3-[2-(tetrazol-1-yl)phenyl]urea
—— 1-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-3-(1,3,5-trimethylpyrazol-4-yl)urea —— C13H18N4O3
1-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-3-(1,3,5-trimethylpyrazol-4-yl)urea
—— 1-methyl-1-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]-3-[4-(tetrazol-1-yl)phenyl]urea —— C20H23N7O
1-methyl-1-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]-3-[4-(tetrazol-1-yl)phenyl]urea
—— 3-(4-Amino(1,2,5-oxadiazol-3-yl))-5-{[3-(4-fluorophenyl)pyrazol-4-yl]methylene}-2-imino-1,3-thiazolidin-4-one —— C15H10FN7O2S
3-(4-Amino(1,2,5-oxadiazol-3-yl))-5-{[3-(4-fluorophenyl)pyrazol-4-yl]methylene}-2-imino-1,3-thiazolidin-4-one
—— 1-methyl-1-[(3S)-1-methylpyrrolidin-3-yl]-3-(2-phenyl-1,3-benzoxazol-5-yl)urea —— C20H22N4O2
1-methyl-1-[(3S)-1-methylpyrrolidin-3-yl]-3-(2-phenyl-1,3-benzoxazol-5-yl)urea
—— 1-[[(3S)-1,1-dioxothiolan-3-yl]methyl]-3-[4-(1H-pyrazol-4-yl)phenyl]urea —— C15H18N4O3S
1-[[(3S)-1,1-dioxothiolan-3-yl]methyl]-3-[4-(1H-pyrazol-4-yl)phenyl]urea
—— 1-methyl-1-[[(3S)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]-3-[4-(tetrazol-1-yl)phenyl]urea —— C20H23N7O
1-methyl-1-[[(3S)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]-3-[4-(tetrazol-1-yl)phenyl]urea
—— 1-[2-(dimethylamino)ethyl]-1-[[(2S)-oxolan-2-yl]methyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea —— C19H27N5O2
1-[2-(dimethylamino)ethyl]-1-[[(2S)-oxolan-2-yl]methyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea
—— (2R)-2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(4-pyrazol-1-ylphenyl)acetic acid —— C21H28N4O2
(2R)-2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(4-pyrazol-1-ylphenyl)acetic acid
—— (3R)-1-ethylsulfonyl-N-[4-(2-methylimidazol-1-yl)phenyl]piperidine-3-carboxamide —— C18H24N4O3S
(3R)-1-ethylsulfonyl-N-[4-(2-methylimidazol-1-yl)phenyl]piperidine-3-carboxamide
—— (3S)-1-ethylsulfonyl-N-[4-(2-methylimidazol-1-yl)phenyl]piperidine-3-carboxamide —— C18H24N4O3S
(3S)-1-ethylsulfonyl-N-[4-(2-methylimidazol-1-yl)phenyl]piperidine-3-carboxamide
—— 1-[2-(dimethylamino)ethyl]-1-[[(2R)-oxolan-2-yl]methyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea —— C19H27N5O2
1-[2-(dimethylamino)ethyl]-1-[[(2R)-oxolan-2-yl]methyl]-3-[4-(1H-pyrazol-5-yl)phenyl]urea
—— (2S)-2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(4-pyrazol-1-ylphenyl)acetic acid —— C21H28N4O2
(2S)-2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(4-pyrazol-1-ylphenyl)acetic acid
—— N-[(1R)-1-(1H-indol-2-yl)ethyl]-N-methyl-2-(2-phenylimidazol-1-yl)acetamide —— C22H22N4O
N-[(1R)-1-(1H-indol-2-yl)ethyl]-N-methyl-2-(2-phenylimidazol-1-yl)acetamide
—— (3R)-1-(2-imidazol-1-ylacetyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide —— C20H22N6O2
(3R)-1-(2-imidazol-1-ylacetyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
—— N-[(1S)-1-(1H-indol-2-yl)ethyl]-N-methyl-2-(2-phenylimidazol-1-yl)acetamide —— C22H22N4O
N-[(1S)-1-(1H-indol-2-yl)ethyl]-N-methyl-2-(2-phenylimidazol-1-yl)acetamide
—— (3R)-N-[5-ethyl-4-(4-fluorophenyl)-2-methylpyrazol-3-yl]-3-methoxypiperidine-1-carboxamide —— C19H25FN4O2
(3R)-N-[5-ethyl-4-(4-fluorophenyl)-2-methylpyrazol-3-yl]-3-methoxypiperidine-1-carboxamide
—— N-(5-methyl-2-phenylpyrazol-3-yl)-2-(1H-1,2,4-triazol-5-ylsulfanyl)acetamide —— C14H14N6OS
N-(5-methyl-2-phenylpyrazol-3-yl)-2-(1H-1,2,4-triazol-5-ylsulfanyl)acetamide
—— (3S)-N-[5-ethyl-4-(4-fluorophenyl)-2-methylpyrazol-3-yl]-3-methoxypiperidine-1-carboxamide —— C19H25FN4O2
(3S)-N-[5-ethyl-4-(4-fluorophenyl)-2-methylpyrazol-3-yl]-3-methoxypiperidine-1-carboxamide
—— (3S)-1-(2-imidazol-1-ylacetyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide —— C20H22N6O2
(3S)-1-(2-imidazol-1-ylacetyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
—— (4S)-3-[[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one —— C15H15FN2O4
(4S)-3-[[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one
—— (4R)-3-[[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one —— C15H15FN2O4
(4R)-3-[[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one
—— [(3S)-3-(1-butylimidazol-2-yl)piperidin-1-yl]-(1-phenyltriazol-4-yl)methanone —— C21H26N6O
[(3S)-3-(1-butylimidazol-2-yl)piperidin-1-yl]-(1-phenyltriazol-4-yl)methanone
—— 2-[1-(2-chlorophenyl)-5-[(3S)-oxolan-3-yl]-1,2,4-triazol-3-yl]acetamide —— C14H15ClN4O2
2-[1-(2-chlorophenyl)-5-[(3S)-oxolan-3-yl]-1,2,4-triazol-3-yl]acetamide
—— 2-[1-(2-chlorophenyl)-5-[(3R)-oxolan-3-yl]-1,2,4-triazol-3-yl]acetamide —— C14H15ClN4O2
2-[1-(2-chlorophenyl)-5-[(3R)-oxolan-3-yl]-1,2,4-triazol-3-yl]acetamide
—— N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-2-[4-(5-methyltetrazol-1-yl)phenyl]acetamide —— C20H21N5O2
N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-2-[4-(5-methyltetrazol-1-yl)phenyl]acetamide