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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazole-3-carboxamide —— C22H28FN3O3S
N-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]-1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazole-3-carboxamide
—— (E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C24H29N5O2S
(E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— [(3S)-1-[3-(5-methylfuran-2-yl)-1-phenylpyrazole-4-carbonyl]piperidin-3-yl]-morpholin-4-ylmethanone —— C25H28N4O4
[(3S)-1-[3-(5-methylfuran-2-yl)-1-phenylpyrazole-4-carbonyl]piperidin-3-yl]-morpholin-4-ylmethanone
—— N-butyl-2-(4-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-4-methyl-1,3-thiazole-5-carboxamide —— C19H23ClN2O3S2
N-butyl-2-(4-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
—— [(3R)-1-[3-(5-methylfuran-2-yl)-1-phenylpyrazole-4-carbonyl]piperidin-3-yl]-morpholin-4-ylmethanone —— C25H28N4O4
[(3R)-1-[3-(5-methylfuran-2-yl)-1-phenylpyrazole-4-carbonyl]piperidin-3-yl]-morpholin-4-ylmethanone
—— 3-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-methyl-1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C23H30N6O2
3-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-methyl-1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 1-[(2R)-2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-[1-(2-methylphenyl)imidazol-2-yl]sulfanylethanone —— C23H25N3O2S
1-[(2R)-2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-[1-(2-methylphenyl)imidazol-2-yl]sulfanylethanone
—— N-methyl-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methoxy]-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide —— C27H26N6O2
N-methyl-2-[(8-methylimidazo[1,2-a]pyridin-2-yl)methoxy]-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide
—— 1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-[1-(2-methylphenyl)imidazol-2-yl]sulfanylethanone —— C23H25N3O2S
1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-[1-(2-methylphenyl)imidazol-2-yl]sulfanylethanone
—— N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C23H20N4O2S
N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— N-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C23H20N4O2S
N-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— (5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl 2-[[(2S)-oxolan-2-yl]methylsulfanyl]benzoate —— C23H23NO4S
(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl 2-[[(2S)-oxolan-2-yl]methylsulfanyl]benzoate
—— 2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]acetamide —— C21H24N4O3
2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]acetamide
—— [3-[4-(difluoromethoxy)-3-methoxyphenyl]-1,2,4-oxadiazol-5-yl]methyl (2R)-2,3-dihydro-1-benzothiophene-2-carboxylate —— C20H16F2N2O5S
[3-[4-(difluoromethoxy)-3-methoxyphenyl]-1,2,4-oxadiazol-5-yl]methyl (2R)-2,3-dihydro-1-benzothiophene-2-carboxylate
—— 1-methyl-3-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C22H28N6OS
1-methyl-3-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 3-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-methyl-1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C23H30N6O2
3-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-methyl-1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide —— C21H22N4OS2
N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide
—— 1-O-tert-butyl 3-O-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl] (3R)-piperidine-1,3-dicarboxylate —— C22H28N2O5
1-O-tert-butyl 3-O-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl] (3R)-piperidine-1,3-dicarboxylate
—— (1R,2R)-2-(2,3-dihydroindole-1-carbonyl)-N-[2-(1-phenylpyrazol-4-yl)ethyl]cyclohexane-1-carboxamide —— C27H30N4O2
(1R,2R)-2-(2,3-dihydroindole-1-carbonyl)-N-[2-(1-phenylpyrazol-4-yl)ethyl]cyclohexane-1-carboxamide
—— (2S)-2-(4-chloro-2-methylphenoxy)-N-[2-(1-phenylpyrazol-4-yl)ethyl]propanamide —— C21H22ClN3O2
(2S)-2-(4-chloro-2-methylphenoxy)-N-[2-(1-phenylpyrazol-4-yl)ethyl]propanamide
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]butanamide —— C22H22ClN7O
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]butanamide
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]butanamide —— C22H22ClN7O
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]butanamide
—— (4-cyano-5-methyl-2-phenylpyrazol-3-yl)methyl (3S)-3-acetamido-3-thiophen-2-ylpropanoate —— C21H20N4O3S
(4-cyano-5-methyl-2-phenylpyrazol-3-yl)methyl (3S)-3-acetamido-3-thiophen-2-ylpropanoate
—— [3-(2-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (2R)-2,3-dihydro-1-benzothiophene-2-carboxylate —— C20H18N2O4S
[3-(2-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (2R)-2,3-dihydro-1-benzothiophene-2-carboxylate
—— [3-[4-(difluoromethoxy)-3-methoxyphenyl]-1,2,4-oxadiazol-5-yl]methyl (2S)-2,3-dihydro-1-benzothiophene-2-carboxylate —— C20H16F2N2O5S
[3-[4-(difluoromethoxy)-3-methoxyphenyl]-1,2,4-oxadiazol-5-yl]methyl (2S)-2,3-dihydro-1-benzothiophene-2-carboxylate
—— (5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl (2R)-2-(4-nitrophenyl)sulfanylpropanoate —— C20H18N2O5S
(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl (2R)-2-(4-nitrophenyl)sulfanylpropanoate
—— N-[(R)-cyclopropyl-(4-methylphenyl)methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C23H26N4OS
N-[(R)-cyclopropyl-(4-methylphenyl)methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 2-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]acetamide —— C21H24N4O3
2-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]acetamide
—— (1R,2S)-2-(2,3-dihydroindole-1-carbonyl)-N-[2-(1-phenylpyrazol-4-yl)ethyl]cyclohexane-1-carboxamide —— C27H30N4O2
(1R,2S)-2-(2,3-dihydroindole-1-carbonyl)-N-[2-(1-phenylpyrazol-4-yl)ethyl]cyclohexane-1-carboxamide
—— (5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl (2S)-2-(4-nitrophenyl)sulfanylpropanoate —— C20H18N2O5S
(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl (2S)-2-(4-nitrophenyl)sulfanylpropanoate
—— 1-O-tert-butyl 3-O-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl] (3S)-piperidine-1,3-dicarboxylate —— C22H28N2O5
1-O-tert-butyl 3-O-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl] (3S)-piperidine-1,3-dicarboxylate
—— (2S)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[2-(1-phenylpyrazol-4-yl)ethyl]propanamide —— C22H23FN4O2S
(2S)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[2-(1-phenylpyrazol-4-yl)ethyl]propanamide
—— (4-cyano-5-methyl-2-phenylpyrazol-3-yl)methyl (3R)-3-acetamido-3-thiophen-2-ylpropanoate —— C21H20N4O3S
(4-cyano-5-methyl-2-phenylpyrazol-3-yl)methyl (3R)-3-acetamido-3-thiophen-2-ylpropanoate
—— (1S,2S)-2-(2,3-dihydroindole-1-carbonyl)-N-[2-(1-phenylpyrazol-4-yl)ethyl]cyclohexane-1-carboxamide —— C27H30N4O2
(1S,2S)-2-(2,3-dihydroindole-1-carbonyl)-N-[2-(1-phenylpyrazol-4-yl)ethyl]cyclohexane-1-carboxamide
—— N-[(S)-cyclopropyl-(4-methylphenyl)methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C23H26N4OS
N-[(S)-cyclopropyl-(4-methylphenyl)methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (Z)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]prop-2-enamide —— C26H26ClN5O
(Z)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]prop-2-enamide
—— [3-(2-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (2S)-2,3-dihydro-1-benzothiophene-2-carboxylate —— C20H18N2O4S
[3-(2-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (2S)-2,3-dihydro-1-benzothiophene-2-carboxylate
—— dimethyl-[(1S)-2-[(3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carbonyl)amino]-1-thiophen-2-ylethyl]azanium —— C21H23N4OS2+
dimethyl-[(1S)-2-[(3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carbonyl)amino]-1-thiophen-2-ylethyl]azanium
—— 1-Cyclopentyl-3-[(3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carbonyl)amino]thiourea —— C19H21N5OS2
1-Cyclopentyl-3-[(3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carbonyl)amino]thiourea
—— N-[(1R)-1-(3-acetamidophenyl)ethyl]-N-benzyl-3-(1-phenylpyrazol-4-yl)propanamide —— C29H30N4O2
N-[(1R)-1-(3-acetamidophenyl)ethyl]-N-benzyl-3-(1-phenylpyrazol-4-yl)propanamide
—— (3S)-1-(5-chloro-2-methoxyphenyl)-5-oxo-N-[2-(1-phenylpyrazol-4-yl)ethyl]pyrrolidine-3-carboxamide —— C23H23ClN4O3
(3S)-1-(5-chloro-2-methoxyphenyl)-5-oxo-N-[2-(1-phenylpyrazol-4-yl)ethyl]pyrrolidine-3-carboxamide
—— N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C22H17FN6OS
N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— 4-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-2-phenyl-1,3-oxazole —— C25H26N4O3S
4-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-2-phenyl-1,3-oxazole
—— (2S)-N-[2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]-2-(4-methoxyphenoxy)propanamide —— C22H25N3O3
(2S)-N-[2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]-2-(4-methoxyphenoxy)propanamide
—— (2R)-N-[2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]-2-(4-methoxyphenoxy)propanamide —— C22H25N3O3
(2R)-N-[2-(3,5-dimethylphenyl)-5-methylpyrazol-3-yl]-2-(4-methoxyphenoxy)propanamide
—— 3-(4-fluorophenyl)-N-[(E)-(2-oxo-3,3a,4,5,5a,6,7,8,8a,8b-decahydroacenaphthylen-1-ylidene)amino]imidazole-4-carboxamide —— C22H23FN4O2
3-(4-fluorophenyl)-N-[(E)-(2-oxo-3,3a,4,5,5a,6,7,8,8a,8b-decahydroacenaphthylen-1-ylidene)amino]imidazole-4-carboxamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-1-phenyl-N-propyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C20H22N4O3S2
N-[(3R)-1,1-dioxothiolan-3-yl]-1-phenyl-N-propyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— (3R)-1-(5-chloro-2-methoxyphenyl)-5-oxo-N-[2-(1-phenylpyrazol-4-yl)ethyl]pyrrolidine-3-carboxamide —— C23H23ClN4O3
(3R)-1-(5-chloro-2-methoxyphenyl)-5-oxo-N-[2-(1-phenylpyrazol-4-yl)ethyl]pyrrolidine-3-carboxamide
—— 4-[[5-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-2-phenyl-1,3-oxazole —— C25H26N4O3S
4-[[5-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-2-phenyl-1,3-oxazole
—— N-[(3S)-1,1-dioxothiolan-3-yl]-1-phenyl-N-propyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C20H22N4O3S2
N-[(3S)-1,1-dioxothiolan-3-yl]-1-phenyl-N-propyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide