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中文名称 英文名称 CAS号 化学式 结构式图片
—— (7S)-2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H21F2N7OS2
(7S)-2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— [(2S)-1-(4-methoxycarbonyl-3,5-dimethyl-1H-pyrrol-2-yl)-1-oxopropan-2-yl] 1-[(2-chlorophenyl)methyl]pyrazole-4-carboxylate —— C22H22ClN3O5
[(2S)-1-(4-methoxycarbonyl-3,5-dimethyl-1H-pyrrol-2-yl)-1-oxopropan-2-yl] 1-[(2-chlorophenyl)methyl]pyrazole-4-carboxylate
—— 2-[1-[(5-Phenyltetrazol-2-yl)methyl]piperidin-4-yl]-1,3-benzothiazole —— C20H20N6S
2-[1-[(5-Phenyltetrazol-2-yl)methyl]piperidin-4-yl]-1,3-benzothiazole
—— 6-[(1S)-1-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-N-phenyl-1,3,5-triazine-2,4-diamine —— C20H20N8OS
6-[(1S)-1-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-N-phenyl-1,3,5-triazine-2,4-diamine
—— (2R)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-4-phenylbutan-2-yl]propanamide —— C23H28N4OS
(2R)-2-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-4-phenylbutan-2-yl]propanamide
—— (2S)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)-3-methylbutanamide —— C25H29FN4O3S
(2S)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)-3-methylbutanamide
—— morpholin-4-yl-[(2R)-4-(2-phenyltriazole-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]methanone —— C22H21N5O4
morpholin-4-yl-[(2R)-4-(2-phenyltriazole-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]methanone
—— 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]pyridine —— C19H19FN4OS
2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]pyridine
—— (7S)-7-methyl-2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C23H24N6S2
(7S)-7-methyl-2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (2R)-N-cyclopropyl-2-phenyl-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylacetamide —— C22H19N5OS
(2R)-N-cyclopropyl-2-phenyl-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylacetamide
—— N-[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide —— C18H16N4O4
N-[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
—— 5-Phenyl-2-(piperidin-1-ylmethyl)-1,3-oxazole —— C15H18N2O
5-Phenyl-2-(piperidin-1-ylmethyl)-1,3-oxazole
—— (7R)-2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H21F2N7OS2
(7R)-2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]pyridine —— C19H19FN4OS
2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]pyridine
—— (2R)-2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)-3-methylbutanamide —— C25H29FN4O3S
(2R)-2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)-3-methylbutanamide
—— (2R)-N-(4-methoxyphenyl)-3-methyl-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]butanamide —— C25H31N5O2S
(2R)-N-(4-methoxyphenyl)-3-methyl-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]butanamide
—— morpholin-4-yl-[(2S)-4-(2-phenyltriazole-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]methanone —— C22H21N5O4
morpholin-4-yl-[(2S)-4-(2-phenyltriazole-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]methanone
—— 2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[(1R)-1-naphthalen-1-ylethyl]acetamide —— C23H23N5OS
2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[(1R)-1-naphthalen-1-ylethyl]acetamide
—— (3R,5R)-3-[[5-(2-methoxyphenyl)-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-5-methyloxolan-2-one —— C22H23N3O3S
(3R,5R)-3-[[5-(2-methoxyphenyl)-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-5-methyloxolan-2-one
—— (2S)-2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)-3-methylbutanamide —— C25H29FN4O3S
(2S)-2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)-3-methylbutanamide
—— 5-[(2,2-dimethyl-3H-1-benzofuran-7-yl)oxymethyl]-3-(3-methoxyphenyl)-1,2,4-oxadiazole —— C20H20N2O4
5-[(2,2-dimethyl-3H-1-benzofuran-7-yl)oxymethyl]-3-(3-methoxyphenyl)-1,2,4-oxadiazole
—— [3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 1-(2-fluorophenyl)cyclopentane-1-carboxylate —— C22H21FN2O4
[3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 1-(2-fluorophenyl)cyclopentane-1-carboxylate
—— (3S)-1-[2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]piperidine-3-carboxamide —— C17H22N6O2S
(3S)-1-[2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]piperidine-3-carboxamide
—— 3-[4-[(Z)-(2-cyclohexylimino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-3-phenylpyrazol-1-yl]propanenitrile —— C22H23N5OS
3-[4-[(Z)-(2-cyclohexylimino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-3-phenylpyrazol-1-yl]propanenitrile
—— (2R)-1-(azepan-1-yl)-2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylpropan-1-one —— C16H20FN5OS
(2R)-1-(azepan-1-yl)-2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylpropan-1-one
—— (7S)-2-[[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H23N7S2
(7S)-2-[[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— N-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylpropyl]-2-[3-(tetrazol-1-yl)phenoxy]acetamide —— C22H25N5O4
N-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylpropyl]-2-[3-(tetrazol-1-yl)phenoxy]acetamide
—— 6-[(1R)-1-[[5-(4-chlorophenyl)-4-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-N,2-N-dimethyl-1,3,5-triazine-2,4-diamine —— C22H23ClN8S
6-[(1R)-1-[[5-(4-chlorophenyl)-4-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-N,2-N-dimethyl-1,3,5-triazine-2,4-diamine
—— (7R)-7-methyl-2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C23H24N6S2
(7R)-7-methyl-2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (7S)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H23N7OS2
(7S)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (7R)-2-[[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H23N7S2
(7R)-2-[[1-(2,3-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 4-[[4-Cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-2-thiophen-2-yl-1,3-thiazole —— C19H15FN4S3
4-[[4-Cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-2-thiophen-2-yl-1,3-thiazole
—— N-[(2R)-2-morpholin-4-ium-4-yl-2-thiophen-2-ylethyl]-1-phenyltetrazol-5-amine —— C17H21N6OS+
N-[(2R)-2-morpholin-4-ium-4-yl-2-thiophen-2-ylethyl]-1-phenyltetrazol-5-amine
—— (7R)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H23N7OS2
(7R)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 2-[3-[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]phenoxy]acetate —— C21H15ClFN2O4-
2-[3-[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]phenoxy]acetate
—— (1R,2R,4R)-N-[5-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]bicyclo[2.2.1]heptane-2-carboxamide —— C17H20N4O2
(1R,2R,4R)-N-[5-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]bicyclo[2.2.1]heptane-2-carboxamide
—— N'-[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]-1,5-diphenyl-1,2,4-triazole-3-carbohydrazide —— C23H23N5O2
N'-[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]-1,5-diphenyl-1,2,4-triazole-3-carbohydrazide
—— ethyl (2Z)-2-[(5Z)-5-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-ylidene]acetate —— C18H16ClN3O2S2
ethyl (2Z)-2-[(5Z)-5-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-ylidene]acetate
—— 6-[(1R)-1-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-N-phenyl-1,3,5-triazine-2,4-diamine —— C20H20N8OS
6-[(1R)-1-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-2-N-phenyl-1,3,5-triazine-2,4-diamine
—— N-[(R)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide —— C24H24FN5O3S
N-[(R)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide
—— ethyl (2Z)-2-[(5Z)-2-sulfanylidene-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-4-ylidene]acetate —— C12H11NO2S3
ethyl (2Z)-2-[(5Z)-2-sulfanylidene-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-4-ylidene]acetate
—— (E)-N-[(1S)-2,3-dihydro-1H-inden-1-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C23H23N3O
(E)-N-[(1S)-2,3-dihydro-1H-inden-1-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide —— C24H24FN5O3S
N-[(S)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide
—— (1R,2S,4R)-N-[5-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]bicyclo[2.2.1]heptane-2-carboxamide —— C17H20N4O2
(1R,2S,4R)-N-[5-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]bicyclo[2.2.1]heptane-2-carboxamide
—— (3S)-N'-[2-[3-(3-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]acetyl]-2,3-dihydro-1,4-benzodioxine-3-carbohydrazide —— C20H19N5O4S
(3S)-N'-[2-[3-(3-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]acetyl]-2,3-dihydro-1,4-benzodioxine-3-carbohydrazide
—— (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-1-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-one —— C20H16ClFN2O3
(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-1-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-one
—— N-[(2S)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]-1-(4-fluorophenyl)-5-methyl-1,2,4-triazole-3-carboxamide —— C23H28FN5O2
N-[(2S)-2-(diethylamino)-2-(3-methoxyphenyl)ethyl]-1-(4-fluorophenyl)-5-methyl-1,2,4-triazole-3-carboxamide
—— N'-[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]-1,5-diphenyl-1,2,4-triazole-3-carbohydrazide —— C23H23N5O2
N'-[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]-1,5-diphenyl-1,2,4-triazole-3-carbohydrazide
—— prop-2-enyl (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-2-cyanoprop-2-enoate —— C17H13ClFN3O2
prop-2-enyl (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-2-cyanoprop-2-enoate
—— butyl (E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-2-cyanoprop-2-enoate —— C18H18ClN3O2
butyl (E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-2-cyanoprop-2-enoate