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中文名称 英文名称 CAS号 化学式 结构式图片
—— pyridin-2-yl-[4-[(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C21H20F3N5O2
pyridin-2-yl-[4-[(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— [4-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-[4-(trifluoromethyl)phenyl]methanone —— C23H22F4N4O2
[4-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-[4-(trifluoromethyl)phenyl]methanone
—— 2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-(4-chlorophenyl)ethyl]acetamide —— C23H24ClN5O2S
2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-(4-chlorophenyl)ethyl]acetamide
—— 1-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-[(2S)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]urea —— C21H28N6O5
1-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-[(2S)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]urea
—— N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C20H17ClN6O
N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— 1-[(1R)-1-(3-bromophenyl)ethyl]-3-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]urea —— C19H18BrN5O3
1-[(1R)-1-(3-bromophenyl)ethyl]-3-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]urea
—— 1-[(1S)-1-(4-chlorophenyl)propyl]-3-[2-(1-phenylpyrazol-4-yl)ethyl]urea —— C21H23ClN4O
1-[(1S)-1-(4-chlorophenyl)propyl]-3-[2-(1-phenylpyrazol-4-yl)ethyl]urea
—— 2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-(4-chlorophenyl)ethyl]acetamide —— C23H24ClN5O2S
2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-(4-chlorophenyl)ethyl]acetamide
—— (2R)-4-[[5-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]-3-oxo-2-(4-phenyl-1,3-thiazol-2-yl)butanenitrile —— C20H15N5O2S3
(2R)-4-[[5-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]-3-oxo-2-(4-phenyl-1,3-thiazol-2-yl)butanenitrile
—— 3-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-1-methyl-1-[(1-phenylpyrazol-4-yl)methyl]urea —— C24H26N6O2
3-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-1-methyl-1-[(1-phenylpyrazol-4-yl)methyl]urea
—— 1-[(1S)-1-(3-bromophenyl)ethyl]-3-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]urea —— C19H18BrN5O3
1-[(1S)-1-(3-bromophenyl)ethyl]-3-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]urea
—— 5-[(1S)-1-[[5-(4-fluorophenyl)-1,3-oxazol-2-yl]sulfanyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C17H12FN3O2S2
5-[(1S)-1-[[5-(4-fluorophenyl)-1,3-oxazol-2-yl]sulfanyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 3-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methylsulfanyl]-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazol-5-one —— C17H17ClN4O3S
3-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methylsulfanyl]-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazol-5-one
—— 1-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-[(2R)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]urea —— C21H28N6O5
1-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-[(2R)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]urea
—— [5-ethyl-1-(4-fluorophenyl)pyrazol-4-yl]-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]methanone —— C24H26FN3O2
[5-ethyl-1-(4-fluorophenyl)pyrazol-4-yl]-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]methanone
—— 1-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]urea —— C21H28N6O5
1-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]urea
—— 1-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-3-propan-2-ylthiourea —— C15H18ClN5S
1-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-3-propan-2-ylthiourea
—— N-[(2R)-butan-2-yl]-N-methyl-2-[3-(4-nitrophenyl)-1-phenylpyrazol-4-yl]acetamide —— C22H24N4O3
N-[(2R)-butan-2-yl]-N-methyl-2-[3-(4-nitrophenyl)-1-phenylpyrazol-4-yl]acetamide
—— N-[(2S)-butan-2-yl]-N-methyl-2-[3-(4-nitrophenyl)-1-phenylpyrazol-4-yl]acetamide —— C22H24N4O3
N-[(2S)-butan-2-yl]-N-methyl-2-[3-(4-nitrophenyl)-1-phenylpyrazol-4-yl]acetamide
—— 5-[(1R)-1-[[5-(4-fluorophenyl)-1,3-oxazol-2-yl]sulfanyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C17H12FN3O2S2
5-[(1R)-1-[[5-(4-fluorophenyl)-1,3-oxazol-2-yl]sulfanyl]ethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 1-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-3-[(1S)-1-(3-chlorophenyl)ethyl]urea —— C22H23ClN6O
1-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-3-[(1S)-1-(3-chlorophenyl)ethyl]urea
—— (2S)-2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methyl-6-propan-2-ylphenyl)propanamide —— C26H31N5O2S
(2S)-2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methyl-6-propan-2-ylphenyl)propanamide
—— 4-[(E)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C18H14N6S
4-[(E)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— (2R)-2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methyl-6-propan-2-ylphenyl)propanamide —— C26H31N5O2S
(2R)-2-[[4-(3-acetamidophenyl)-5-cyclopropyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methyl-6-propan-2-ylphenyl)propanamide
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzamide —— C22H19F3N4O3
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzamide
—— 4-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C9H12N6S
4-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 1-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-3-[(1R)-1-(3-chlorophenyl)ethyl]urea —— C22H23ClN6O
1-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-3-[(1R)-1-(3-chlorophenyl)ethyl]urea
—— 4-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1H-1,2,4-triazole-5-thione —— C13H10ClFN6S
4-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1H-1,2,4-triazole-5-thione
—— N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-2-phenyl-1,3-thiazole-4-carboxamide —— C18H19N3OS2
N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-2-phenyl-1,3-thiazole-4-carboxamide
—— (3R)-N-[(E)-[1-[(4-chlorophenyl)methyl]-3-(4-methoxyphenyl)pyrazol-4-yl]methylideneamino]-1-ethylsulfonylpiperidine-3-carboxamide —— C26H30ClN5O4S
(3R)-N-[(E)-[1-[(4-chlorophenyl)methyl]-3-(4-methoxyphenyl)pyrazol-4-yl]methylideneamino]-1-ethylsulfonylpiperidine-3-carboxamide
—— 1-(2,3-dimethylphenyl)-3-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiourea —— C18H19N7S
1-(2,3-dimethylphenyl)-3-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiourea
—— N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-2-phenyl-1,3-thiazole-4-carboxamide —— C18H19N3OS2
N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-2-phenyl-1,3-thiazole-4-carboxamide
—— 4-[(5-phenyltetrazol-2-yl)methyl]-N-[(Z)-[(5R)-3,3,5-trimethylcyclohexylidene]amino]benzamide —— C24H28N6O
4-[(5-phenyltetrazol-2-yl)methyl]-N-[(Z)-[(5R)-3,3,5-trimethylcyclohexylidene]amino]benzamide
—— N-[(E)-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)methylideneamino]-3-phenyl-1H-pyrazole-5-carboxamide —— C22H19ClN6O
N-[(E)-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)methylideneamino]-3-phenyl-1H-pyrazole-5-carboxamide
—— (Z)-N-[(4S)-1-(4-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-3-pyridin-2-ylprop-2-enamide —— C23H23FN4O
(Z)-N-[(4S)-1-(4-fluorophenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-3-pyridin-2-ylprop-2-enamide
—— 2-anilino-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]acetamide —— C17H17N7O
2-anilino-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]acetamide
—— N-[(E)-(2-fluorophenyl)methylideneamino]-4-[(5-phenyltetrazol-2-yl)methyl]benzamide —— C22H17FN6O
N-[(E)-(2-fluorophenyl)methylideneamino]-4-[(5-phenyltetrazol-2-yl)methyl]benzamide
—— 2-(2-methoxyanilino)-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]acetamide —— C18H19N7O2
2-(2-methoxyanilino)-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]acetamide
—— 4-[(5-phenyltetrazol-2-yl)methyl]-N-[(E)-1-pyridin-4-ylethylideneamino]benzamide —— C22H19N7O
4-[(5-phenyltetrazol-2-yl)methyl]-N-[(E)-1-pyridin-4-ylethylideneamino]benzamide
—— 4-[(E)-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]methylideneamino]-3-(2-methylphenyl)-1H-1,2,4-triazole-5-thione —— C19H23N5OS
4-[(E)-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]methylideneamino]-3-(2-methylphenyl)-1H-1,2,4-triazole-5-thione
—— 4-[(E)-(3,5-dimethoxyphenyl)methylideneamino]-3-(2-methylphenyl)-1H-1,2,4-triazole-5-thione —— C18H18N4O2S
4-[(E)-(3,5-dimethoxyphenyl)methylideneamino]-3-(2-methylphenyl)-1H-1,2,4-triazole-5-thione
—— 3-(2-methylphenyl)-4-[(E)-(3-phenylmethoxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C23H20N4OS
3-(2-methylphenyl)-4-[(E)-(3-phenylmethoxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(3-methylthiophen-2-yl)methyl]butanamide —— C17H18ClN5OS
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(3-methylthiophen-2-yl)methyl]butanamide
—— 2-methyl-N-[(E)-(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylideneamino]furan-3-carboxamide —— C21H23N5O2
2-methyl-N-[(E)-(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylideneamino]furan-3-carboxamide
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(3-methylthiophen-2-yl)methyl]butanamide —— C17H18ClN5OS
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(3-methylthiophen-2-yl)methyl]butanamide
—— 1-(4-chlorophenyl)-N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-5-propan-2-ylpyrazole-4-carboxamide —— C21H25ClN4OS
1-(4-chlorophenyl)-N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-5-propan-2-ylpyrazole-4-carboxamide
—— (1S,2S,4S)-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]bicyclo[2.2.1]heptane-2-carboxamide —— C18H22N4O
(1S,2S,4S)-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]bicyclo[2.2.1]heptane-2-carboxamide
—— 1-(4-chlorophenyl)-N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-5-propan-2-ylpyrazole-4-carboxamide —— C21H25ClN4OS
1-(4-chlorophenyl)-N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-5-propan-2-ylpyrazole-4-carboxamide
—— [(2S,5R)-2,5-dimethylmorpholin-4-yl]-[5-thiophen-2-yl-1-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]methanone —— C20H19F3N4O2S
[(2S,5R)-2,5-dimethylmorpholin-4-yl]-[5-thiophen-2-yl-1-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]methanone
—— (1S,2R,4S)-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]bicyclo[2.2.1]heptane-2-carboxamide —— C18H22N4O
(1S,2R,4S)-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]bicyclo[2.2.1]heptane-2-carboxamide