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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(pyrazol-1-ylmethyl)phenyl]methyl]butanamide —— C22H22ClN7O
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(pyrazol-1-ylmethyl)phenyl]methyl]butanamide
—— (2R)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(5-methyl-1,2-oxazol-3-yl)-2-phenylacetamide —— C25H24FN5O3S
(2R)-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(5-methyl-1,2-oxazol-3-yl)-2-phenylacetamide
—— (2R)-2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(5-methyl-1,2-oxazol-3-yl)-2-phenylacetamide —— C25H24FN5O3S
(2R)-2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(5-methyl-1,2-oxazol-3-yl)-2-phenylacetamide
—— N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)acetamide —— C25H29N3O3
N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)acetamide
—— 1-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]-2-(2-phenyl-1,3-oxazol-4-yl)ethanone —— C20H25N3O3
1-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]-2-(2-phenyl-1,3-oxazol-4-yl)ethanone
—— N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)acetamide —— C25H29N3O3
N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)acetamide
—— 1-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]-2-(2-phenyl-1,3-oxazol-4-yl)ethanone —— C20H25N3O3
1-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]-2-(2-phenyl-1,3-oxazol-4-yl)ethanone
—— [2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl] 2-[(5S,7R)-3-bromo-1-adamantyl]acetate —— C20H26BrN3O4S
[2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl] 2-[(5S,7R)-3-bromo-1-adamantyl]acetate
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide —— C22H27N3O2
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide
—— 6-bromo-3-(2-methoxyethyl)-2-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one —— C21H19BrN4O3S
6-bromo-3-(2-methoxyethyl)-2-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one
—— N-phenyl-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,3,4-thiadiazol-2-amine —— C18H15N5OS2
N-phenyl-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,3,4-thiadiazol-2-amine
—— N-(3-fluorophenyl)-5-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,3,4-thiadiazol-2-amine —— C18H14FN5OS2
N-(3-fluorophenyl)-5-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,3,4-thiadiazol-2-amine
—— [2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl] 2-[(5R,7R)-3-bromo-1-adamantyl]acetate —— C20H26BrN3O4S
[2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl] 2-[(5R,7R)-3-bromo-1-adamantyl]acetate
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide —— C22H27N3O2
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide
—— 3-(5-methylpyridin-2-yl)-2-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one —— C24H19N5O2S
3-(5-methylpyridin-2-yl)-2-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one
—— 4-[4-(2-methylphenyl)-5-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-3-yl]morpholine —— C23H24N6O2S
4-[4-(2-methylphenyl)-5-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-3-yl]morpholine
—— 6-bromo-3-(2-methoxyethyl)-2-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one —— C21H19BrN4O3S
6-bromo-3-(2-methoxyethyl)-2-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one
—— N-(3-fluorophenyl)-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,3,4-thiadiazol-2-amine —— C18H14FN5OS2
N-(3-fluorophenyl)-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,3,4-thiadiazol-2-amine
—— 3-(5-methylpyridin-2-yl)-2-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one —— C24H19N5O2S
3-(5-methylpyridin-2-yl)-2-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one
—— 4-[4-(2-methylphenyl)-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-3-yl]morpholine —— C23H24N6O2S
4-[4-(2-methylphenyl)-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-3-yl]morpholine
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]propanamide —— C21H21FN6O2S
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]propanamide
—— 4-methoxy-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-1-phenylpyrazole-3-carboxamide —— C21H22N6O2S
4-methoxy-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-1-phenylpyrazole-3-carboxamide
—— [2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl] 2-[(5S,7S)-3-bromo-1-adamantyl]acetate —— C20H26BrN3O4S
[2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl] 2-[(5S,7S)-3-bromo-1-adamantyl]acetate
—— 2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-N-[4-(1,3-oxazol-5-yl)phenyl]acetamide —— C18H20N2O2
2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-N-[4-(1,3-oxazol-5-yl)phenyl]acetamide
—— 4-methoxy-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-1-phenylpyrazole-3-carboxamide —— C21H22N6O2S
4-methoxy-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-1-phenylpyrazole-3-carboxamide
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide —— C22H27N3O2
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide —— C22H27N3O2
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetamide
—— 2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-N-[4-(1,3-oxazol-5-yl)phenyl]acetamide —— C18H20N2O2
2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-N-[4-(1,3-oxazol-5-yl)phenyl]acetamide
—— N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-4-(tetrazol-1-yl)benzamide —— C18H18N8OS
N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]-4-(tetrazol-1-yl)benzamide
—— (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]prop-2-enamide —— C23H22ClFN6OS
(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]prop-2-enamide
—— N-[(S)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide —— C21H18FN5OS
N-[(S)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide
—— N-[(R)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide —— C21H18FN5OS
N-[(R)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]propanamide —— C21H21FN6O2S
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]propanamide
—— N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C23H24N6OS
N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— (E)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enamide —— C27H23N5OS
(E)-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enamide
—— 5-chloro-N-[(R)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide —— C24H23ClFN5O
5-chloro-N-[(R)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide
—— N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C23H24N6OS
N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— (E)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enamide —— C27H23N5OS
(E)-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enamide
—— 3-(2,4-dichlorophenyl)-5-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-4-amine —— C18H14Cl2N6OS
3-(2,4-dichlorophenyl)-5-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-4-amine
—— 3-methyl-5-nitro-N-[[(2S)-pyrrolidin-2-yl]methyl]imidazol-4-amine —— C9H15N5O2
3-methyl-5-nitro-N-[[(2S)-pyrrolidin-2-yl]methyl]imidazol-4-amine
—— 3-[(4-methoxyphenyl)methyl]-2-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one —— C26H22N4O3S
3-[(4-methoxyphenyl)methyl]-2-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one
—— 5-chloro-N-[(S)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide —— C24H23ClFN5O
5-chloro-N-[(S)-(4-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide
—— 3-methyl-5-nitro-N-[[(2R)-pyrrolidin-2-yl]methyl]imidazol-4-amine —— C9H15N5O2
3-methyl-5-nitro-N-[[(2R)-pyrrolidin-2-yl]methyl]imidazol-4-amine
—— 2-[(5S,7S)-3-bromo-1-adamantyl]-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]acetamide —— C23H28BrN3O
2-[(5S,7S)-3-bromo-1-adamantyl]-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]acetamide
—— 3-(2,4-dichlorophenyl)-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-4-amine —— C18H14Cl2N6OS
3-(2,4-dichlorophenyl)-5-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-1,2,4-triazol-4-amine
—— 2-[(5S,7S)-3-bromo-1-adamantyl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]acetamide —— C23H28BrN3O
2-[(5S,7S)-3-bromo-1-adamantyl]-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]acetamide
—— 3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]propanamide —— C21H21ClN6O2S
3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]propanamide
—— 5-[(1R)-1-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C23H22FN5O2S
5-[(1R)-1-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(1S)-1-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C23H22FN5O2S
5-[(1S)-1-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— 3-[3-(dimethylamino)propyl]-2-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H29N5O2S2
3-[3-(dimethylamino)propyl]-2-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one