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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-5-(3-methoxyphenyl)-1-methylpyrazole-3-carboxamide —— C19H23N3O2
N-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-5-(3-methoxyphenyl)-1-methylpyrazole-3-carboxamide
—— N-[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-1-methylpyrazole-3-carboxamide —— C19H22FN3O2
N-[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-1-methylpyrazole-3-carboxamide
—— N-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-propylpyrazole-3-carboxamide —— C22H29N3O3
N-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-propylpyrazole-3-carboxamide
—— [(2S)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-[4-(5-methylpyrazol-1-yl)phenyl]methanone —— C23H23N3O3
[(2S)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-[4-(5-methylpyrazol-1-yl)phenyl]methanone
—— (2R)-N-(2,6-dichlorophenyl)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C23H27Cl2N5OS
(2R)-N-(2,6-dichlorophenyl)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 5-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-phenylpyrazole-3-carboxamide —— C21H21N3O2
5-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-phenylpyrazole-3-carboxamide
—— N-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-1-ethyl-5-(3-fluorophenyl)pyrazole-3-carboxamide —— C19H22FN3O
N-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]-1-ethyl-5-(3-fluorophenyl)pyrazole-3-carboxamide
—— (E)-N-[(3,4-dimethoxyphenyl)methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C23H25N3O3
(E)-N-[(3,4-dimethoxyphenyl)methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-[(3,4-dimethoxyphenyl)methyl]prop-2-enamide —— C22H22ClN3O3
(E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-[(3,4-dimethoxyphenyl)methyl]prop-2-enamide
—— [(2S)-1-oxo-1-[[(1S)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate —— C23H25N3O3S
[(2S)-1-oxo-1-[[(1S)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate
—— 2-(4-fluorophenyl)-N-[(2-methoxyphenyl)methyl]-1,3-thiazole-4-carboxamide —— C18H15FN2O2S
2-(4-fluorophenyl)-N-[(2-methoxyphenyl)methyl]-1,3-thiazole-4-carboxamide
—— [(2R)-1-oxo-1-[[(1S)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate —— C23H25N3O3S
[(2R)-1-oxo-1-[[(1S)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate
—— [(2S)-1-oxo-1-[[(1R)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate —— C23H25N3O3S
[(2S)-1-oxo-1-[[(1R)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(4-fluorophenyl)ethyl]butanamide —— C19H19ClFN5O
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(4-fluorophenyl)ethyl]butanamide
—— (2S)-2-[1-(3-chlorophenyl)imidazol-2-yl]sulfanyl-N-(2,6-dichlorophenyl)propanamide —— C18H14Cl3N3OS
(2S)-2-[1-(3-chlorophenyl)imidazol-2-yl]sulfanyl-N-(2,6-dichlorophenyl)propanamide
—— (2R)-2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(difluoromethoxy)phenyl]propanamide —— C22H24ClF2N5O2S
(2R)-2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(difluoromethoxy)phenyl]propanamide
—— N-[2-(4-chlorophenyl)ethyl]-1-(4-fluorophenyl)-5-methyl-1,2,4-triazole-3-carboxamide —— C18H16ClFN4O
N-[2-(4-chlorophenyl)ethyl]-1-(4-fluorophenyl)-5-methyl-1,2,4-triazole-3-carboxamide
—— 2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide —— C19H16ClFN2OS
2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
—— 2-(4-chlorophenyl)-N-[(2-methoxyphenyl)methyl]-4-methyl-1,3-thiazole-5-carboxamide —— C19H17ClN2O2S
2-(4-chlorophenyl)-N-[(2-methoxyphenyl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
—— (2R)-N-(3-chloro-4-fluorophenyl)-2-[[4-(4-methylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C22H23ClFN5O2S
(2R)-N-(3-chloro-4-fluorophenyl)-2-[[4-(4-methylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— [(2S)-1-oxo-1-(2-phenylethylamino)propan-2-yl] 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate —— C22H22N2O3S
[(2S)-1-oxo-1-(2-phenylethylamino)propan-2-yl] 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate
—— 2-(3-chlorophenyl)-N-[(2-methoxyphenyl)methyl]-5-methyltriazole-4-carboxamide —— C18H17ClN4O2
2-(3-chlorophenyl)-N-[(2-methoxyphenyl)methyl]-5-methyltriazole-4-carboxamide
—— 1-benzyl-N-[5-[(4-fluorophenyl)methyl]-1,3-thiazol-2-yl]-3,5-dimethylpyrazole-4-carboxamide —— C23H21FN4OS
1-benzyl-N-[5-[(4-fluorophenyl)methyl]-1,3-thiazol-2-yl]-3,5-dimethylpyrazole-4-carboxamide
—— (2R)-N-(2,6-dichlorophenyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C22H23Cl2N5OS
(2R)-N-(2,6-dichlorophenyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— 2-[[(2S)-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]thiophene-3-carboxamide —— C22H26N6O2S2
2-[[(2S)-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]thiophene-3-carboxamide
—— [(2R)-1-oxo-1-(propylamino)propan-2-yl] 3-(5-methylfuran-2-yl)-1-phenylpyrazole-4-carboxylate —— C21H23N3O4
[(2R)-1-oxo-1-(propylamino)propan-2-yl] 3-(5-methylfuran-2-yl)-1-phenylpyrazole-4-carboxylate
—— (2S)-2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N,N-di(propan-2-yl)propanamide —— C20H29N3OS
(2S)-2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N,N-di(propan-2-yl)propanamide
—— (2S)-N-(2,5-dimethylphenyl)-2-[[5-(4-fluorophenyl)-4-(2-morpholin-4-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H30FN5O2S
(2S)-N-(2,5-dimethylphenyl)-2-[[5-(4-fluorophenyl)-4-(2-morpholin-4-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2S)-2-[[5-(4-fluorophenyl)-4-(2-morpholin-4-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-phenylethyl)propanamide —— C25H30FN5O2S
(2S)-2-[[5-(4-fluorophenyl)-4-(2-morpholin-4-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-phenylethyl)propanamide
—— 2-(2,4-dimethylphenyl)-N-[(2-methoxyphenyl)methyl]-5-methyltriazole-4-carboxamide —— C20H22N4O2
2-(2,4-dimethylphenyl)-N-[(2-methoxyphenyl)methyl]-5-methyltriazole-4-carboxamide
—— 5-[(4-Bromo-2-chlorophenoxy)methyl]-1-phenyltetrazole —— C14H10BrClN4O
5-[(4-Bromo-2-chlorophenoxy)methyl]-1-phenyltetrazole
—— 3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-prop-2-enylpropanamide —— C17H21N3O
3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-prop-2-enylpropanamide
—— 2-(4-fluorophenyl)-N-[(2-methoxyphenyl)methyl]-4-methyl-1,3-thiazole-5-carboxamide —— C19H17FN2O2S
2-(4-fluorophenyl)-N-[(2-methoxyphenyl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
—— [(2R)-1-oxo-1-[[(1R)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate —— C23H25N3O3S
[(2R)-1-oxo-1-[[(1R)-1-phenylbutyl]amino]propan-2-yl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate
—— [(2S)-1-(4-methoxy-2-nitroanilino)-1-oxopropan-2-yl] 3-(4-bromophenyl)-1H-pyrazole-5-carboxylate —— C20H17BrN4O6
[(2S)-1-(4-methoxy-2-nitroanilino)-1-oxopropan-2-yl] 3-(4-bromophenyl)-1H-pyrazole-5-carboxylate
—— (2S)-N-(2,6-dimethylphenyl)-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H29N5OS
(2S)-N-(2,6-dimethylphenyl)-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-2-[[4-(4-methylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-phenylethyl)propanamide —— C24H29N5O2S
(2R)-2-[[4-(4-methylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-phenylethyl)propanamide
—— N-[2-(4-chlorophenyl)ethyl]-4-methyl-2-thiophen-2-yl-1,3-thiazole-5-carboxamide —— C17H15ClN2OS2
N-[2-(4-chlorophenyl)ethyl]-4-methyl-2-thiophen-2-yl-1,3-thiazole-5-carboxamide
—— N-[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-ethylpyrazole-3-carboxamide —— C21H27N3O3
N-[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-ethylpyrazole-3-carboxamide
—— (2R)-N-(2,6-dichlorophenyl)-2-[[4-phenyl-5-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C22H18Cl2N4OS2
(2R)-N-(2,6-dichlorophenyl)-2-[[4-phenyl-5-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]-1-ethyl-5-[3-(trifluoromethyl)phenyl]pyrazole-3-carboxamide —— C20H22F3N3O
N-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]-1-ethyl-5-[3-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
—— (E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-[(4-fluorophenyl)methyl]prop-2-enamide —— C20H17ClFN3O
(E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-[(4-fluorophenyl)methyl]prop-2-enamide
—— [(2S)-1-[di(propan-2-yl)amino]-1-oxopropan-2-yl] 2-(2-phenyl-1,3-thiazol-4-yl)acetate —— C20H26N2O3S
[(2S)-1-[di(propan-2-yl)amino]-1-oxopropan-2-yl] 2-(2-phenyl-1,3-thiazol-4-yl)acetate
—— (2S)-2-[[4-(2-chlorophenyl)-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(2,6-dichlorophenyl)propanamide —— C21H20Cl3N5OS
(2S)-2-[[4-(2-chlorophenyl)-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(2,6-dichlorophenyl)propanamide
—— N-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-1-methylpyrazole-3-carboxamide —— C19H22FN3O2
N-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-1-methylpyrazole-3-carboxamide
—— [2-[methyl-[(1S)-1-phenylethyl]amino]-2-oxoethyl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate —— C21H21N3O3S
[2-[methyl-[(1S)-1-phenylethyl]amino]-2-oxoethyl] 2-(2-pyridin-2-yl-1,3-thiazol-4-yl)acetate
—— (2R)-2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(difluoromethoxy)phenyl]propanamide —— C22H24ClF2N5O2S
(2R)-2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(difluoromethoxy)phenyl]propanamide
—— (2R)-2-[[5-(4-fluorophenyl)-4-(2-morpholin-4-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-phenylethyl)propanamide —— C25H30FN5O2S
(2R)-2-[[5-(4-fluorophenyl)-4-(2-morpholin-4-ylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-phenylethyl)propanamide
—— (2R)-N-[2-(4-methoxyphenyl)ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H31N5O2S
(2R)-N-[2-(4-methoxyphenyl)ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— ethyl (2E)-2-[4-oxo-3-[2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C17H16F3N5O3S
ethyl (2E)-2-[4-oxo-3-[2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]ethyl]-1,3-thiazolidin-2-ylidene]acetate