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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(4-fluorophenyl)-N-[(2R)-2-morpholin-4-ylpropyl]-5-propan-2-ylpyrazole-4-carboxamide —— C20H27FN4O2
1-(4-fluorophenyl)-N-[(2R)-2-morpholin-4-ylpropyl]-5-propan-2-ylpyrazole-4-carboxamide
—— methyl 5-[[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]amino]methyl]-2-methylfuran-3-carboxylate —— C21H19ClFN3O4
methyl 5-[[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]amino]methyl]-2-methylfuran-3-carboxylate
—— (3S)-N-[(2R)-2-morpholin-4-ylpropyl]-2,3-diphenyl-3,4-dihydropyrazole-5-carboxamide —— C23H28N4O2
(3S)-N-[(2R)-2-morpholin-4-ylpropyl]-2,3-diphenyl-3,4-dihydropyrazole-5-carboxamide
—— 1-(4-fluorophenyl)-N-[(2S)-2-morpholin-4-ylpropyl]-5-propan-2-ylpyrazole-4-carboxamide —— C20H27FN4O2
1-(4-fluorophenyl)-N-[(2S)-2-morpholin-4-ylpropyl]-5-propan-2-ylpyrazole-4-carboxamide
—— (E)-N-(3-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C25H26FN3O3S
(E)-N-(3-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— 1-(4-bromophenyl)-N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide —— C20H18BrN3O2
1-(4-bromophenyl)-N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide
—— 2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide —— C22H23F3N4O2S
2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide
—— 1-(3-fluorophenyl)-N-[(2S)-2-morpholin-4-ylpropyl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C20H22FN5O2S
1-(3-fluorophenyl)-N-[(2S)-2-morpholin-4-ylpropyl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— 1-(3-fluorophenyl)-N-[(2R)-2-morpholin-4-ylpropyl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C20H22FN5O2S
1-(3-fluorophenyl)-N-[(2R)-2-morpholin-4-ylpropyl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— (3S)-N-[(2S)-2-morpholin-4-ylpropyl]-2,3-diphenyl-3,4-dihydropyrazole-5-carboxamide —— C23H28N4O2
(3S)-N-[(2S)-2-morpholin-4-ylpropyl]-2,3-diphenyl-3,4-dihydropyrazole-5-carboxamide
—— 2-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide —— C21H21F3N4O3S
2-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide —— C20H17F4N3O3
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)butanamide —— C20H19ClN6O2
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)butanamide
—— 4-[(E)-[5-chloro-1-(2,5-dimethylphenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,2,4-triazolidine-3,5-dithione —— C15H15ClN6S2
4-[(E)-[5-chloro-1-(2,5-dimethylphenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,2,4-triazolidine-3,5-dithione
—— methyl 3-[1-[4-[[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]carbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C29H36N4O3
methyl 3-[1-[4-[[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]carbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide —— C20H17F4N3O3
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide
—— 3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide —— C21H20F3N3O4
3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide
—— 1-(2-methylphenyl)-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide —— C21H17F6N3O2
1-(2-methylphenyl)-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide
—— 2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide —— C21H19F3N2O3
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide
—— (2R)-2-(4-nitro-1,3-dioxoisoindol-2-yl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide —— C21H14F3N5O5
(2R)-2-(4-nitro-1,3-dioxoisoindol-2-yl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide
—— 2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide —— C21H19F3N2O3
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide
—— (3S)-1-(1,3-benzodioxol-5-yl)-5-oxo-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]pyrrolidine-3-carboxamide —— C22H17F3N4O4
(3S)-1-(1,3-benzodioxol-5-yl)-5-oxo-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]pyrrolidine-3-carboxamide
—— (3S)-3-acetamido-3-(4-chlorophenyl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide —— C21H18ClF3N4O2
(3S)-3-acetamido-3-(4-chlorophenyl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide
—— 1-(2-methylphenyl)-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide —— C21H17F6N3O2
1-(2-methylphenyl)-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide
—— 3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide —— C21H20F3N3O4
3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide
—— 3-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide —— C21H18F4N2O3
3-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]propanamide
—— (3S)-1-(5-chloro-2-methoxyphenyl)-5-oxo-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]pyrrolidine-3-carboxamide —— C22H18ClF3N4O3
(3S)-1-(5-chloro-2-methoxyphenyl)-5-oxo-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]pyrrolidine-3-carboxamide
—— 2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide —— C22H23F3N4O2S
2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]acetamide
—— N-[[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C28H22N4O3S
N-[[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (3R)-1-(1,3-benzodioxol-5-yl)-5-oxo-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]pyrrolidine-3-carboxamide —— C22H17F3N4O4
(3R)-1-(1,3-benzodioxol-5-yl)-5-oxo-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]pyrrolidine-3-carboxamide
—— (2S)-2-(4-nitro-1,3-dioxoisoindol-2-yl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide —— C21H14F3N5O5
(2S)-2-(4-nitro-1,3-dioxoisoindol-2-yl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide
—— (E)-N-(4-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C25H26FN3O3S
(E)-N-(4-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— (2R)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-oxo-2-[4-pyrazol-1-yl-2-(trifluoromethyl)anilino]ethyl]sulfanylpropanamide —— C19H18F3N5O3S
(2R)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-oxo-2-[4-pyrazol-1-yl-2-(trifluoromethyl)anilino]ethyl]sulfanylpropanamide
—— (2S)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-oxo-2-[4-pyrazol-1-yl-2-(trifluoromethyl)anilino]ethyl]sulfanylpropanamide —— C19H18F3N5O3S
(2S)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-oxo-2-[4-pyrazol-1-yl-2-(trifluoromethyl)anilino]ethyl]sulfanylpropanamide
—— 1-(4-chlorophenyl)-N-[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-5-(trifluoromethyl)pyrazole-4-carboxamide —— C24H24ClF3N4O
1-(4-chlorophenyl)-N-[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-5-(trifluoromethyl)pyrazole-4-carboxamide
—— (Z)-N-(4-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C25H26FN3O3S
(Z)-N-(4-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— (2R)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-[(4-methyl-5-phenyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]sulfanylpropanamide —— C19H20N4O3S2
(2R)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-[(4-methyl-5-phenyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]sulfanylpropanamide
—— (3R)-3-acetamido-3-(4-chlorophenyl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide —— C21H18ClF3N4O2
(3R)-3-acetamido-3-(4-chlorophenyl)-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide
—— (2S)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-[(4-methyl-5-phenyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]sulfanylpropanamide —— C19H20N4O3S2
(2S)-N-(5-methyl-1,2-oxazol-3-yl)-2-[2-[(4-methyl-5-phenyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]sulfanylpropanamide
—— 3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide —— C21H21F3N4O3
3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[4-pyrazol-1-yl-2-(trifluoromethyl)phenyl]propanamide
—— N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C24H24ClF3N4O2
N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— (2R)-2-(4-tert-butylphenoxy)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]propanamide —— C21H23ClN4O2
(2R)-2-(4-tert-butylphenoxy)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]propanamide
—— (3R)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]-1-(2-phenylacetyl)piperidine-3-carboxamide —— C22H22ClN5O2
(3R)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]-1-(2-phenylacetyl)piperidine-3-carboxamide
—— N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C21H22ClN3O2S2
N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— (2S)-2-(4-tert-butylphenoxy)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]propanamide —— C21H23ClN4O2
(2S)-2-(4-tert-butylphenoxy)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]propanamide
—— (3S,5S)-3,5-dimethyl-N-[(1R)-1-(1H-1,2,4-triazol-5-yl)ethyl]adamantane-1-carboxamide —— C17H26N4O
(3S,5S)-3,5-dimethyl-N-[(1R)-1-(1H-1,2,4-triazol-5-yl)ethyl]adamantane-1-carboxamide
—— (3S)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxamide —— C18H16ClN5O3
(3S)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]-1-(furan-2-ylmethyl)-5-oxopyrrolidine-3-carboxamide
—— (5-amino-1-methylpyrazol-4-yl)-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C15H24N4O
(5-amino-1-methylpyrazol-4-yl)-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— (5-amino-1-methylpyrazol-4-yl)-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C15H24N4O
(5-amino-1-methylpyrazol-4-yl)-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— (3S)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]-1-(2-phenylacetyl)piperidine-3-carboxamide —— C22H22ClN5O2
(3S)-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]-1-(2-phenylacetyl)piperidine-3-carboxamide