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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3,5-dimethoxy-4-phenylmethoxybenzamide —— C28H28FN3O4
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3,5-dimethoxy-4-phenylmethoxybenzamide
—— 2-cyclopentyl-1-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethanone —— C22H30N4O2
2-cyclopentyl-1-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethanone
—— (3R)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(4-methylphenyl)-5-oxopyrrolidine-3-carboxamide —— C24H25FN4O2
(3R)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(4-methylphenyl)-5-oxopyrrolidine-3-carboxamide
—— (2R)-N-(3-methoxypropyl)-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]propanamide —— C15H18F3N5O2
(2R)-N-(3-methoxypropyl)-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]propanamide
—— (2S)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2,3-dihydro-1-benzothiophene-2-carboxamide —— C22H21N5OS
(2S)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2,3-dihydro-1-benzothiophene-2-carboxamide
—— 4-tert-butyl-N-[3-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-3-oxopropyl]benzamide —— C26H31FN4O2
4-tert-butyl-N-[3-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-3-oxopropyl]benzamide
—— (2R)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2,3-dihydro-1-benzothiophene-2-carboxamide —— C22H21N5OS
(2R)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2,3-dihydro-1-benzothiophene-2-carboxamide
—— (2S)-N-(3-methoxypropyl)-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]propanamide —— C15H18F3N5O2
(2S)-N-(3-methoxypropyl)-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]propanamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3,4-dimethyl-5-(methylsulfamoyl)benzamide —— C22H25FN4O3S
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3,4-dimethyl-5-(methylsulfamoyl)benzamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3,4-dimethyl-5-(methylsulfamoyl)benzamide —— C22H25FN4O3S
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3,4-dimethyl-5-(methylsulfamoyl)benzamide
—— 2-cyclopentyl-1-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethanone —— C22H30N4O2
2-cyclopentyl-1-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethanone
—— (2R)-3-methyl-N-[(2R)-4-phenylbutan-2-yl]-2-(5-phenyltetrazol-2-yl)butanamide —— C22H27N5O
(2R)-3-methyl-N-[(2R)-4-phenylbutan-2-yl]-2-(5-phenyltetrazol-2-yl)butanamide
—— 2-(3-ethyl-2,4-dioxoquinazolin-1-yl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C24H24FN5O3
2-(3-ethyl-2,4-dioxoquinazolin-1-yl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide
—— 1-(3-chlorophenyl)-N-[(1R)-1-phenylethyl]-5-propan-2-ylpyrazole-4-carboxamide —— C21H22ClN3O
1-(3-chlorophenyl)-N-[(1R)-1-phenylethyl]-5-propan-2-ylpyrazole-4-carboxamide
—— (2R)-N-(2-cyanoethyl)-N-(4-methylphenyl)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide —— C24H22N6O2S
(2R)-N-(2-cyanoethyl)-N-(4-methylphenyl)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide
—— 2-chloro-5-(diethylsulfamoyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide —— C23H26ClFN4O3S
2-chloro-5-(diethylsulfamoyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide —— C22H21FN4O2S
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide
—— (5-bromofuran-2-yl)-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C20H21BrN4O3
(5-bromofuran-2-yl)-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-piperidin-1-ylsulfonylbenzamide —— C24H27FN4O3S
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-piperidin-1-ylsulfonylbenzamide
—— ethyl (3R)-1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl]piperidine-3-carboxylate —— C21H27N3O5
ethyl (3R)-1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl]piperidine-3-carboxylate
—— 1-(3-chlorophenyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide —— C23H18ClF4N5O
1-(3-chlorophenyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide
—— (2R)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]-N-quinolin-5-ylpropanamide —— C23H18N6O2S
(2R)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]-N-quinolin-5-ylpropanamide
—— 4-ethoxy-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide —— C21H22FN3O2
4-ethoxy-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide —— C22H21FN4O2S
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide
—— N'-{(E)-[1-phenyl-3-(tricyclo[3.3.1.1~3,7~]dec-1-yl)-1H-pyrazol-4-yl]methylidene}pyridine-3-carbohydrazide —— C26H27N5O
N'-{(E)-[1-phenyl-3-(tricyclo[3.3.1.1~3,7~]dec-1-yl)-1H-pyrazol-4-yl]methylidene}pyridine-3-carbohydrazide
—— (2S)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2-(4-bromophenoxy)propanamide —— C22H22BrN5O2
(2S)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2-(4-bromophenoxy)propanamide
—— (2S)-N-(2-cyanoethyl)-N-(4-methylphenyl)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide —— C24H22N6O2S
(2S)-N-(2-cyanoethyl)-N-(4-methylphenyl)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide
—— N-[(1R)-1-(3-bromophenyl)ethyl]-3-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]propanamide —— C20H18BrClN2O2
N-[(1R)-1-(3-bromophenyl)ethyl]-3-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]propanamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide —— C22H21FN4O2S
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetamide
—— N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-2-(4-fluorophenyl)acetamide —— C19H16ClFN4O
N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-2-(4-fluorophenyl)acetamide
—— N-[(1S)-1-(3-bromophenyl)ethyl]-3-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]propanamide —— C20H18BrClN2O2
N-[(1S)-1-(3-bromophenyl)ethyl]-3-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]propanamide
—— 1-(3-chlorophenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide —— C23H18ClF4N5O
1-(3-chlorophenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-(trifluoromethyl)pyrazole-4-carboxamide
—— (5-bromofuran-2-yl)-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C20H21BrN4O3
(5-bromofuran-2-yl)-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 4-[5-[(1R)-1-(3-butyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-yl]-N,N-diethylaniline —— C21H30N6OS
4-[5-[(1R)-1-(3-butyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-yl]-N,N-diethylaniline
—— (2R)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2-(4-bromophenoxy)propanamide —— C22H22BrN5O2
(2R)-N-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propyl]-2-(4-bromophenoxy)propanamide
—— (E)-N-[(1S)-1-(3-bromophenyl)ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C15H15BrN2OS
(E)-N-[(1S)-1-(3-bromophenyl)ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— 2-chloro-5-(diethylsulfamoyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide —— C23H26ClFN4O3S
2-chloro-5-(diethylsulfamoyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-piperidin-1-ylsulfonylbenzamide —— C24H27FN4O3S
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-piperidin-1-ylsulfonylbenzamide
—— ethyl (2Z)-[1-(3-chlorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl](hydroxyimino)acetate —— C15H16ClN3O3
ethyl (2Z)-[1-(3-chlorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl](hydroxyimino)acetate
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-oxo-3-phenylphthalazine-1-carboxamide —— C27H22FN5O2
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-oxo-3-phenylphthalazine-1-carboxamide
—— 4-ethoxy-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide —— C21H22FN3O2
4-ethoxy-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide
—— [(3R,5R)-3,5-dimethylpiperidin-1-yl]-[1-(2-fluorophenyl)-5-pyrrol-1-ylpyrazol-4-yl]methanone —— C21H23FN4O
[(3R,5R)-3,5-dimethylpiperidin-1-yl]-[1-(2-fluorophenyl)-5-pyrrol-1-ylpyrazol-4-yl]methanone
—— ethyl (3S)-1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl]piperidine-3-carboxylate —— C21H27N3O5
ethyl (3S)-1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl]piperidine-3-carboxylate
—— 4-[5-[(1S)-1-(3-butyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-yl]-N,N-diethylaniline —— C21H30N6OS
4-[5-[(1S)-1-(3-butyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-yl]-N,N-diethylaniline
—— N-[(1S)-1-(3-bromophenyl)ethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C21H23BrN4OS
N-[(1S)-1-(3-bromophenyl)ethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— [(3S,5S)-3,5-dimethylpiperidin-1-yl]-[1-(2-fluorophenyl)-5-pyrrol-1-ylpyrazol-4-yl]methanone —— C21H23FN4O
[(3S,5S)-3,5-dimethylpiperidin-1-yl]-[1-(2-fluorophenyl)-5-pyrrol-1-ylpyrazol-4-yl]methanone
—— (E)-N-[(1S)-1-(3-bromophenyl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C20H18BrN3O
(E)-N-[(1S)-1-(3-bromophenyl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-N-[(1R)-1-(3-bromophenyl)ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C15H15BrN2OS
(E)-N-[(1R)-1-(3-bromophenyl)ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— 1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoylamino]-3-[(1S,2S)-2-methylcyclohexyl]thiourea —— C21H29N5O3S
1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoylamino]-3-[(1S,2S)-2-methylcyclohexyl]thiourea
—— 1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoylamino]-3-[(1S,2R)-2-methylcyclohexyl]thiourea —— C21H29N5O3S
1-[3-[3-(4-ethoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoylamino]-3-[(1S,2R)-2-methylcyclohexyl]thiourea