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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-cyano-N-cyclohexyl-3-(4-methyl-2-propyl-1,3-thiazol-5-yl)-3-oxopropanamide —— C17H23N3O2S
(2R)-2-cyano-N-cyclohexyl-3-(4-methyl-2-propyl-1,3-thiazol-5-yl)-3-oxopropanamide
—— (2R)-2-cyano-N-(4-ethylphenyl)-3-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]-3-oxopropanamide —— C22H19FN4O2
(2R)-2-cyano-N-(4-ethylphenyl)-3-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]-3-oxopropanamide
—— ethyl (4R)-6-[[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H31N5O3
ethyl (4R)-6-[[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (2S)-2-cyano-N-cyclohexyl-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide —— C24H28N4O2
(2S)-2-cyano-N-cyclohexyl-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide
—— 1-benzyl-N-[2-(furan-2-yl)ethyl]-3-(4-methoxyphenyl)pyrazole-4-carboxamide —— C24H23N3O3
1-benzyl-N-[2-(furan-2-yl)ethyl]-3-(4-methoxyphenyl)pyrazole-4-carboxamide
—— [(Z)-[(1S,2R,5S)-2-[4-(3-chlorophenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea —— C14H14ClN7O2S2
[(Z)-[(1S,2R,5S)-2-[4-(3-chlorophenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea
—— (E,2S)-2-cyano-N-cyclohexyl-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide —— C21H22N4O2
(E,2S)-2-cyano-N-cyclohexyl-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide
—— [(E)-[(1S,2S,5S)-2-[4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea —— C16H19N7O2S2
[(E)-[(1S,2S,5S)-2-[4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea
—— (2S)-2-cyano-N-cyclohexyl-3-oxo-3-(1-phenyltriazol-4-yl)propanamide —— C18H19N5O2
(2S)-2-cyano-N-cyclohexyl-3-oxo-3-(1-phenyltriazol-4-yl)propanamide
—— 3-[[3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(furan-2-yl)-1,2,4-triazol-4-amine —— C17H16N6O2S
3-[[3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(furan-2-yl)-1,2,4-triazol-4-amine
—— (2R)-2-cyano-N-cyclohexyl-3-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-3-oxopropanamide —— C21H24N4O2
(2R)-2-cyano-N-cyclohexyl-3-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-3-oxopropanamide
—— (2S)-2-cyano-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)-N-(3-propan-2-yloxypropyl)propanamide —— C24H30N4O3
(2S)-2-cyano-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)-N-(3-propan-2-yloxypropyl)propanamide
—— (2S)-2-cyano-5-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-(3-methoxyphenyl)-3-oxopentanamide —— C22H18FN3O4
(2S)-2-cyano-5-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-(3-methoxyphenyl)-3-oxopentanamide
—— 2-[(4-chlorophenoxy)methyl]-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C23H26ClN3O3S
2-[(4-chlorophenoxy)methyl]-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— (E,2R)-2-cyano-N-cyclohexyl-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide —— C21H22N4O2
(E,2R)-2-cyano-N-cyclohexyl-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide
—— ethyl N-[2-[(1,3-diphenylpyrazol-4-yl)methyl-methylamino]acetyl]carbamate —— C22H24N4O3
ethyl N-[2-[(1,3-diphenylpyrazol-4-yl)methyl-methylamino]acetyl]carbamate
—— (2R)-4-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-2-cyano-3-oxo-N-(3-propan-2-yloxypropyl)butanamide —— C20H22ClN3O3S
(2R)-4-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-2-cyano-3-oxo-N-(3-propan-2-yloxypropyl)butanamide
—— (2R)-2-cyano-5-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-(3-methoxyphenyl)-3-oxopentanamide —— C22H18FN3O4
(2R)-2-cyano-5-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-(3-methoxyphenyl)-3-oxopentanamide
—— (2S)-2-cyano-N-(3-methoxyphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide —— C22H19N3O4
(2S)-2-cyano-N-(3-methoxyphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide
—— (6-Chloro-7-methyl-2-oxochromen-4-yl)methyl-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-methylazanium —— C24H25ClN3O2+
(6-Chloro-7-methyl-2-oxochromen-4-yl)methyl-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-methylazanium
—— (E,2S)-2-cyano-3-oxo-5-(1-phenylpyrazol-4-yl)-N-(3-propan-2-yloxypropyl)pent-4-enamide —— C21H24N4O3
(E,2S)-2-cyano-3-oxo-5-(1-phenylpyrazol-4-yl)-N-(3-propan-2-yloxypropyl)pent-4-enamide
—— 1-[(2-chlorophenyl)methyl]-N-[2-(furan-2-yl)ethyl]-3-phenylpyrazole-4-carboxamide —— C23H20ClN3O2
1-[(2-chlorophenyl)methyl]-N-[2-(furan-2-yl)ethyl]-3-phenylpyrazole-4-carboxamide
—— 2-[2-(3-bromophenyl)-1,3-thiazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]acetamide —— C22H24BrN3O2S
2-[2-(3-bromophenyl)-1,3-thiazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]acetamide
—— (2R)-2-cyano-N-(3-methoxyphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide —— C22H19N3O4
(2R)-2-cyano-N-(3-methoxyphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide
—— (E,2R)-2-cyano-5-(2-methyl-1,3-thiazol-4-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide —— C16H21N3O3S
(E,2R)-2-cyano-5-(2-methyl-1,3-thiazol-4-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide
—— [(E)-[(1S,2R,5S)-2-[4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea —— C16H19N7O2S2
[(E)-[(1S,2R,5S)-2-[4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea
—— (2S)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-(3-methoxyphenyl)-3-oxopentanamide —— C22H18ClN3O4
(2S)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-(3-methoxyphenyl)-3-oxopentanamide
—— (2R)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-(3-methoxyphenyl)-3-oxopentanamide —— C22H18ClN3O4
(2R)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-(3-methoxyphenyl)-3-oxopentanamide
—— (2S)-2-cyano-3-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]-3-oxo-N-(3-propan-2-yloxypropyl)propanamide —— C20H23FN4O3
(2S)-2-cyano-3-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]-3-oxo-N-(3-propan-2-yloxypropyl)propanamide
—— (2R)-2-cyano-N-cyclohexyl-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide —— C24H28N4O2
(2R)-2-cyano-N-cyclohexyl-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide
—— N-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide —— C21H24N4O2S
N-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide
—— (E,2R)-2-cyano-N-(3-methoxyphenyl)-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide —— C22H18N4O3
(E,2R)-2-cyano-N-(3-methoxyphenyl)-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide
—— (2R)-2-cyano-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)-N-(3-propan-2-yloxypropyl)propanamide —— C24H30N4O3
(2R)-2-cyano-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)-N-(3-propan-2-yloxypropyl)propanamide
—— (2S)-4-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-2-cyano-3-oxo-N-(3-propan-2-yloxypropyl)butanamide —— C20H22ClN3O3S
(2S)-4-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-2-cyano-3-oxo-N-(3-propan-2-yloxypropyl)butanamide
—— (E,2S)-2-cyano-5-(2-methyl-1,3-thiazol-4-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide —— C16H21N3O3S
(E,2S)-2-cyano-5-(2-methyl-1,3-thiazol-4-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide
—— N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide —— C21H24N4O2S
N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetamide
—— [(Z)-[(1S,2S,5S)-2-[4-(3-chlorophenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea —— C14H14ClN7O2S2
[(Z)-[(1S,2S,5S)-2-[4-(3-chlorophenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-ylidene]amino]thiourea
—— 2-(4-chlorophenyl)-N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C22H24ClN3O2S
2-(4-chlorophenyl)-N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— [(2R)-1-[benzyl(methyl)amino]-1-oxopropan-2-yl] 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetate —— C24H25N3O4
[(2R)-1-[benzyl(methyl)amino]-1-oxopropan-2-yl] 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-oxoacetate
—— 2-(4-chlorophenyl)-N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C22H24ClN3O2S
2-(4-chlorophenyl)-N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— 2-methyl-5-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1,3-thiazole-4-carboxylic acid —— C16H24N2O2S
2-methyl-5-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1,3-thiazole-4-carboxylic acid
—— (2S)-2-cyano-N-cyclohexyl-3-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-3-oxopropanamide —— C21H24N4O2
(2S)-2-cyano-N-cyclohexyl-3-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-3-oxopropanamide
—— N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-(4-methylphenyl)-1,3-thiazole-4-carboxamide —— C22H25N3O2S
N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-(4-methylphenyl)-1,3-thiazole-4-carboxamide
—— N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-(4-methylphenyl)-1,3-thiazole-4-carboxamide —— C22H25N3O2S
N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-(4-methylphenyl)-1,3-thiazole-4-carboxamide
—— 2-[(4-chlorophenoxy)methyl]-N-[(2S)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C23H26ClN3O3S
2-[(4-chlorophenoxy)methyl]-N-[(2S)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— (Z)-1,1,1-trifluoro-4-[[5-methyl-2-(4-methylphenyl)pyrazol-3-yl]amino]but-3-en-2-one —— C15H14F3N3O
(Z)-1,1,1-trifluoro-4-[[5-methyl-2-(4-methylphenyl)pyrazol-3-yl]amino]but-3-en-2-one
—— [(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl] 2-[(4-chlorophenoxy)methyl]-4-methyl-1,3-thiazole-5-carboxylate —— C21H25ClN2O4S
[(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl] 2-[(4-chlorophenoxy)methyl]-4-methyl-1,3-thiazole-5-carboxylate
—— 2-[(4-chlorophenoxy)methyl]-N-[(2R)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C23H26ClN3O3S
2-[(4-chlorophenoxy)methyl]-N-[(2R)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— 3-[(5-Cyclopropyl-1-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-5-(4-fluorophenyl)-4-methyl-1,2-oxazole —— C22H19FN4OS
3-[(5-Cyclopropyl-1-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-5-(4-fluorophenyl)-4-methyl-1,2-oxazole
—— (3,5-Dimethyl-1-phenylpyrazol-4-yl)methyl-methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]azanium —— C22H24N5O+
(3,5-Dimethyl-1-phenylpyrazol-4-yl)methyl-methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]azanium