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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C22H30N4OS
2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C25H24FN5O2S
N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— N-[(2R)-4-(furan-2-yl)butan-2-yl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C21H20N4O2S
N-[(2R)-4-(furan-2-yl)butan-2-yl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— 2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-2-phenylbutyl]acetamide —— C22H26N4OS
2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-2-phenylbutyl]acetamide
—— 3-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide —— C23H21F3N4O3
3-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide
—— 2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C22H30N4OS
2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— [(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone —— C22H23FN4OS
[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone
—— 2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-2-phenylbutyl]acetamide —— C22H26N4OS
2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-2-phenylbutyl]acetamide
—— ethyl 2-[(4-fluorophenyl)methyl-[(2R)-2-(4-methoxyphenoxy)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C24H25FN2O5S
ethyl 2-[(4-fluorophenyl)methyl-[(2R)-2-(4-methoxyphenoxy)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[(4-fluorophenyl)methyl-[(2S)-2-(4-methoxyphenoxy)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C24H25FN2O5S
ethyl 2-[(4-fluorophenyl)methyl-[(2S)-2-(4-methoxyphenoxy)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— (2S)-1-(4-fluorophenoxy)-3-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]propan-2-ol —— C23H27FN4O3
(2S)-1-(4-fluorophenoxy)-3-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]propan-2-ol
—— 2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C22H30N4OS
2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— [(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone —— C22H23FN4OS
[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone
—— (E,1R,4S)-N-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C21H24ClFN4
(E,1R,4S)-N-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C25H24FN5O2S
N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— (2S)-2-[2-(4-methylanilino)-2-oxoethyl]sulfanyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide —— C23H23F3N4O2S
(2S)-2-[2-(4-methylanilino)-2-oxoethyl]sulfanyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide
—— (Z,1R,4S)-N-[(Z)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C27H29FN4O
(Z,1R,4S)-N-[(Z)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— [1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]methanone —— C22H24FN5O2S
[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]methanone
—— N-[(2R)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C21H21N5O2S
N-[(2R)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— [1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methanone —— C22H24FN5O2S
[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methanone
—— (E,1S,4R)-N-[(E)-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C27H30N4O
(E,1S,4R)-N-[(E)-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— (E,1R,4S)-N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C21H25ClN4
(E,1R,4S)-N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— [(2S)-2-ethylpiperidin-1-yl]-[1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone —— C21H26FN3O
[(2S)-2-ethylpiperidin-1-yl]-[1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone
—— [1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]methanone —— C21H17FN4OS2
[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]methanone
—— (E,1R,4S)-N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C21H25ClN4
(E,1R,4S)-N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— N-[(2S)-4-(furan-2-yl)butan-2-yl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C21H20N4O2S
N-[(2S)-4-(furan-2-yl)butan-2-yl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— 2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C22H30N4OS
2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— 1-(4-fluorophenyl)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C18H17FN4O3S2
1-(4-fluorophenyl)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— [(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-quinolin-8-ylacetate —— C25H24N4O4
[(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-quinolin-8-ylacetate
—— 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-2-methyl-4-oxopentan-3-yl]acetamide —— C21H27FN4O3S
2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-2-methyl-4-oxopentan-3-yl]acetamide
—— [2-[[(2S)-2-cyano-3-methylbutan-2-yl]amino]-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate —— C19H21FN4O3S
[2-[[(2S)-2-cyano-3-methylbutan-2-yl]amino]-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate
—— 4-(4-chlorophenyl)-5-{[(4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]methyl}-2,4-dihydro-3H-1,2,4-triazole-3-thione —— C24H18ClN5S2
4-(4-chlorophenyl)-5-{[(4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]methyl}-2,4-dihydro-3H-1,2,4-triazole-3-thione
—— Cyanomethyl 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate —— C13H10FN3O2S
Cyanomethyl 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate
—— N-[(2S)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C21H21N5O2S
N-[(2S)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— 2-[[5-(2-fluorophenyl)-4-propan-2-yl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-phenylethyl]acetamide —— C21H23FN4OS
2-[[5-(2-fluorophenyl)-4-propan-2-yl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-phenylethyl]acetamide
—— [2-[[(2R)-2-cyano-3-methylbutan-2-yl]amino]-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate —— C19H21FN4O3S
[2-[[(2R)-2-cyano-3-methylbutan-2-yl]amino]-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate
—— (2S)-N-cyclopentyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylpropanamide —— C20H27N3OS
(2S)-N-cyclopentyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylpropanamide
—— N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-methylacetamide —— C22H24N4O3S
N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-methylacetamide
—— (2R)-2-[2-(4-methylanilino)-2-oxoethyl]sulfanyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide —— C23H23F3N4O2S
(2R)-2-[2-(4-methylanilino)-2-oxoethyl]sulfanyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide
—— (3R)-1-(furan-2-ylmethyl)-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide —— C21H19F3N4O3
(3R)-1-(furan-2-ylmethyl)-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide
—— (3S)-1-(furan-2-ylmethyl)-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide —— C21H19F3N4O3
(3S)-1-(furan-2-ylmethyl)-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide
—— (E,1R,4S)-N-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C21H24ClFN4
(E,1R,4S)-N-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— (2S)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-methyl-1,2-oxazol-5-yl)propanamide —— C21H28N6O2S
(2S)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-methyl-1,2-oxazol-5-yl)propanamide
—— [1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methanone —— C21H17FN4OS2
[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methanone
—— 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-2-methyl-4-oxopentan-3-yl]acetamide —— C21H27FN4O3S
2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-2-methyl-4-oxopentan-3-yl]acetamide
—— 2-[1-(3-chloro-2-methylphenyl)imidazol-2-yl]sulfanyl-N-[(3R)-2-methyl-4-oxopentan-3-yl]acetamide —— C18H22ClN3O2S
2-[1-(3-chloro-2-methylphenyl)imidazol-2-yl]sulfanyl-N-[(3R)-2-methyl-4-oxopentan-3-yl]acetamide
—— (3R)-1-cyclopentyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide —— C21H23F3N4O2
(3R)-1-cyclopentyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide
—— (E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C27H29FN4O
(E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— [(2R)-2-ethylpiperidin-1-yl]-[1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone —— C21H26FN3O
[(2R)-2-ethylpiperidin-1-yl]-[1-(4-fluorophenyl)-4,5,6,7-tetrahydroindazol-3-yl]methanone
—— (2R)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-methyl-1,2-oxazol-5-yl)propanamide —— C21H28N6O2S
(2R)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-methyl-1,2-oxazol-5-yl)propanamide