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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1S)-1-(4-fluorophenyl)ethyl]-N-methyl-3-(1-phenylpyrazol-4-yl)propanamide —— C21H22FN3O
N-[(1S)-1-(4-fluorophenyl)ethyl]-N-methyl-3-(1-phenylpyrazol-4-yl)propanamide
—— 3,5-dimethyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-1-phenylpyrazole-4-carboxamide —— C23H28N4O3
3,5-dimethyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-1-phenylpyrazole-4-carboxamide
—— [(3R,3aS,5R,7E)-5-methyl-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C22H21N3OS3
[(3R,3aS,5R,7E)-5-methyl-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 4-(4-chloro-3,5-dimethylpyrazol-1-yl)-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]benzamide —— C23H27ClN4O3
4-(4-chloro-3,5-dimethylpyrazol-1-yl)-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]benzamide
—— (2R)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-(4-methoxyphenyl)-3-oxopentanamide —— C22H18ClN3O4
(2R)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-(4-methoxyphenyl)-3-oxopentanamide
—— 2-(2-ethoxyphenoxy)-N-[4-(4-ethoxyphenyl)-5-methyl-1,3-thiazol-2-yl]acetamide —— C22H24N2O4S
2-(2-ethoxyphenoxy)-N-[4-(4-ethoxyphenyl)-5-methyl-1,3-thiazol-2-yl]acetamide
—— (2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]propan-1-one —— C20H20FN5OS
(2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S)-2-methyl-2,3-dihydroindol-1-yl]propan-1-one
—— ethyl (1S,9R,13E,16S)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C28H26N4O4S
ethyl (1S,9R,13E,16S)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (1S,9R,13E,16R)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C27H24N4O4S
methyl (1S,9R,13E,16R)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— (E)-3-(1-benzyl-3-phenylpyrazol-4-yl)-N-methyl-N-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]prop-2-enamide —— C26H25N5O3
(E)-3-(1-benzyl-3-phenylpyrazol-4-yl)-N-methyl-N-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]prop-2-enamide
—— (1,3-Dioxoisoindol-2-yl)methyl 3-(tetrazol-1-yl)benzoate —— C17H11N5O4
(1,3-Dioxoisoindol-2-yl)methyl 3-(tetrazol-1-yl)benzoate
—— (3S)-1-[(2-chlorophenyl)methyl]-5-oxo-N-[4-(tetrazol-1-yl)phenyl]pyrrolidine-3-carboxamide —— C19H17ClN6O2
(3S)-1-[(2-chlorophenyl)methyl]-5-oxo-N-[4-(tetrazol-1-yl)phenyl]pyrrolidine-3-carboxamide
—— 5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C18H23N5OS2
5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— 4-(4-chloro-3,5-dimethylpyrazol-1-yl)-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]benzamide —— C19H20ClN3OS
4-(4-chloro-3,5-dimethylpyrazol-1-yl)-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]benzamide
—— (1S)-N'-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-N,N-dimethyl-1-thiophen-2-ylethane-1,2-diamine —— C25H28N4S
(1S)-N'-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-N,N-dimethyl-1-thiophen-2-ylethane-1,2-diamine
—— 4-(4-chloro-3,5-dimethylpyrazol-1-yl)-N-methyl-N-[(1R)-1-thiophen-2-ylethyl]benzamide —— C19H20ClN3OS
4-(4-chloro-3,5-dimethylpyrazol-1-yl)-N-methyl-N-[(1R)-1-thiophen-2-ylethyl]benzamide
—— 3,5-dimethyl-N-(2-methyl-2-morpholin-4-ium-4-ylpropyl)-1-phenylpyrazole-4-carboxamide —— C20H29N4O2+
3,5-dimethyl-N-(2-methyl-2-morpholin-4-ium-4-ylpropyl)-1-phenylpyrazole-4-carboxamide
—— 1-(2-Methylphenyl)-5-[(1-phenyltetrazol-5-yl)methylsulfanyl]tetrazole —— C16H14N8S
1-(2-Methylphenyl)-5-[(1-phenyltetrazol-5-yl)methylsulfanyl]tetrazole
—— (E,2S)-2-cyano-N-cyclohexyl-5-(2-methyl-1,3-thiazol-4-yl)-3-oxopent-4-enamide —— C16H19N3O2S
(E,2S)-2-cyano-N-cyclohexyl-5-(2-methyl-1,3-thiazol-4-yl)-3-oxopent-4-enamide
—— (3,5-dimethyl-1-phenylpyrazol-4-yl)methyl-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ium-1-ylethyl]azanium —— C22H30N4O+2
(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ium-1-ylethyl]azanium
—— (2S)-2-cyano-3-(5-methyl-1-phenylpyrazol-3-yl)-N-naphthalen-1-yl-3-oxopropanamide —— C24H18N4O2
(2S)-2-cyano-3-(5-methyl-1-phenylpyrazol-3-yl)-N-naphthalen-1-yl-3-oxopropanamide
—— 2-[1-[(1-Phenyltetrazol-5-yl)methyl]piperidin-1-ium-4-yl]-1,3-benzothiazole —— C20H21N6S+
2-[1-[(1-Phenyltetrazol-5-yl)methyl]piperidin-1-ium-4-yl]-1,3-benzothiazole
—— (2R)-2-cyano-3-(5-methyl-1-phenylpyrazol-3-yl)-N-naphthalen-1-yl-3-oxopropanamide —— C24H18N4O2
(2R)-2-cyano-3-(5-methyl-1-phenylpyrazol-3-yl)-N-naphthalen-1-yl-3-oxopropanamide
—— (2S)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-naphthalen-1-yl-3-oxopentanamide —— C25H18ClN3O3
(2S)-5-[5-(2-chlorophenyl)-1,3-oxazol-2-yl]-2-cyano-N-naphthalen-1-yl-3-oxopentanamide
—— (2S)-2-cyano-N-cyclohexyl-3-(4-methyl-2-propyl-1,3-thiazol-5-yl)-3-oxopropanamide —— C17H23N3O2S
(2S)-2-cyano-N-cyclohexyl-3-(4-methyl-2-propyl-1,3-thiazol-5-yl)-3-oxopropanamide
—— (2R)-2-cyano-N-(4-ethylphenyl)-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide —— C26H26N4O2
(2R)-2-cyano-N-(4-ethylphenyl)-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide
—— 5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C18H23N5OS2
5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— (2S)-2-cyano-N-(4-ethylphenyl)-3-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]-3-oxopropanamide —— C22H19FN4O2
(2S)-2-cyano-N-(4-ethylphenyl)-3-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]-3-oxopropanamide
—— (2R)-2-cyano-N-(4-ethylphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide —— C23H21N3O3
(2R)-2-cyano-N-(4-ethylphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide
—— (2S)-2-cyano-N-(4-ethylphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide —— C23H21N3O3
(2S)-2-cyano-N-(4-ethylphenyl)-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-oxobutanamide
—— (E,2S)-2-cyano-N-(4-ethylphenyl)-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide —— C23H20N4O2
(E,2S)-2-cyano-N-(4-ethylphenyl)-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide
—— (2S)-2-cyano-N-(4-ethylphenyl)-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide —— C26H26N4O2
(2S)-2-cyano-N-(4-ethylphenyl)-3-oxo-3-(3-phenyl-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-1-yl)propanamide
—— (2R)-2-cyano-N-(4-ethylphenyl)-3-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-3-oxopropanamide —— C23H22N4O2
(2R)-2-cyano-N-(4-ethylphenyl)-3-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-3-oxopropanamide
—— 5-cyclopropyl-N-[(2,3-dimethoxyphenyl)methyl]-N-methyl-2-phenylpyrazole-3-carboxamide —— C23H25N3O3
5-cyclopropyl-N-[(2,3-dimethoxyphenyl)methyl]-N-methyl-2-phenylpyrazole-3-carboxamide
—— N-cyclopropyl-4-methyl-2-thiophen-2-yl-1,3-thiazole-5-carboxamide —— C12H12N2OS2
N-cyclopropyl-4-methyl-2-thiophen-2-yl-1,3-thiazole-5-carboxamide
—— N-[4-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-thiazol-2-yl]acetamide —— C15H15N5O2S2
N-[4-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-thiazol-2-yl]acetamide
—— 5-[(5-Chlorothiadiazol-4-yl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C14H9ClN6OS
5-[(5-Chlorothiadiazol-4-yl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— 1-[(2R)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-2-[5-(4-fluorophenyl)tetrazol-2-yl]ethanone —— C21H20FN5O3
1-[(2R)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-2-[5-(4-fluorophenyl)tetrazol-2-yl]ethanone
—— 5-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-2-phenylpyrazole-3-carboxamide —— C21H20FN3O
5-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-2-phenylpyrazole-3-carboxamide
—— 4-[2-[(3-Thiophen-2-yl-1,2,4-oxadiazol-5-yl)methyl]tetrazol-5-yl]benzamide —— C15H11N7O2S
4-[2-[(3-Thiophen-2-yl-1,2,4-oxadiazol-5-yl)methyl]tetrazol-5-yl]benzamide
—— 5-cyclopropyl-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-phenylpyrazole-3-carboxamide —— C23H23N3O3
5-cyclopropyl-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-phenylpyrazole-3-carboxamide
—— (E,2R)-2-cyano-N-(4-ethylphenyl)-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide —— C23H20N4O2
(E,2R)-2-cyano-N-(4-ethylphenyl)-3-oxo-5-(1-phenylpyrazol-4-yl)pent-4-enamide
—— 5-[(1-Cyclopentyltetrazol-5-yl)sulfanylmethyl]-3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazole —— C17H20N6O3S
5-[(1-Cyclopentyltetrazol-5-yl)sulfanylmethyl]-3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazole
—— (2R)-2-cyano-3-[1-(2-fluorophenyl)pyrazol-3-yl]-N-naphthalen-1-yl-3-oxopropanamide —— C23H15FN4O2
(2R)-2-cyano-3-[1-(2-fluorophenyl)pyrazol-3-yl]-N-naphthalen-1-yl-3-oxopropanamide
—— (2R)-2-cyano-N-cyclohexyl-3-oxo-3-(1-phenyltriazol-4-yl)propanamide —— C18H19N5O2
(2R)-2-cyano-N-cyclohexyl-3-oxo-3-(1-phenyltriazol-4-yl)propanamide
—— 3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]propanamide —— C22H20N4O2S
3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]propanamide
—— ethyl (1S,9R,13E,16R)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C28H26N4O4S
ethyl (1S,9R,13E,16R)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— (2S)-2-cyano-N-(4-ethylphenyl)-5-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-3-oxopentanamide —— C23H20FN3O3
(2S)-2-cyano-N-(4-ethylphenyl)-5-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-3-oxopentanamide
—— methyl (1S,9R,13E,16S)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C27H24N4O4S
methyl (1S,9R,13E,16S)-13-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— 1-(1,3-diphenylpyrazol-4-yl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]methanamine —— C26H23N5O
1-(1,3-diphenylpyrazol-4-yl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]methanamine