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中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl 3-[3,5-dimethyl-1-[4-[[(2R)-oxolan-2-yl]methyl-[(3S)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate —— C25H33N3O4S
methyl 3-[3,5-dimethyl-1-[4-[[(2R)-oxolan-2-yl]methyl-[(3S)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate
—— 1-(3-chlorophenyl)-N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide —— C20H18ClN3O2
1-(3-chlorophenyl)-N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide
—— 1-(3-fluorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C22H23FN4O2S2
1-(3-fluorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— N-[[(2S)-oxolan-2-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-thiolan-3-yl]propanamide —— C23H31N3O3S
N-[[(2S)-oxolan-2-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-thiolan-3-yl]propanamide
—— (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]prop-2-enamide —— C23H28FN3O2S
(E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]prop-2-enamide
—— N-[[(2R)-oxolan-2-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-thiolan-3-yl]propanamide —— C23H31N3O3S
N-[[(2R)-oxolan-2-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-thiolan-3-yl]propanamide
—— methyl 3-[3,5-dimethyl-1-[4-[[(2R)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate —— C25H33N3O4S
methyl 3-[3,5-dimethyl-1-[4-[[(2R)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate
—— 4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-2-phenyl-N-[(3S)-thiolan-3-yl]-1,3-thiazole-5-carboxamide —— C20H24N2O2S2
4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-2-phenyl-N-[(3S)-thiolan-3-yl]-1,3-thiazole-5-carboxamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)-N-[(3R)-thiolan-3-yl]acetamide —— C20H24N2O3S
N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)-N-[(3R)-thiolan-3-yl]acetamide
—— N-[[(2S)-oxolan-2-yl]methyl]-2-(6-phenylimidazo[2,1-b][1,3]thiazol-3-yl)-N-[(3S)-thiolan-3-yl]acetamide —— C22H25N3O2S2
N-[[(2S)-oxolan-2-yl]methyl]-2-(6-phenylimidazo[2,1-b][1,3]thiazol-3-yl)-N-[(3S)-thiolan-3-yl]acetamide
—— N-[[(2R)-oxolan-2-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3R)-thiolan-3-yl]propanamide —— C23H31N3O3S
N-[[(2R)-oxolan-2-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3R)-thiolan-3-yl]propanamide
—— 4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-phenyl-N-[(3R)-thiolan-3-yl]-1,3-thiazole-5-carboxamide —— C20H24N2O2S2
4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-phenyl-N-[(3R)-thiolan-3-yl]-1,3-thiazole-5-carboxamide
—— N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]-3-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C18H23N3O3S2
N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]-3-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]-3-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C18H23N3O3S2
N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]-3-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-(6-phenylimidazo[2,1-b][1,3]thiazol-3-yl)-N-[(3S)-thiolan-3-yl]acetamide —— C22H25N3O2S2
N-[[(2R)-oxolan-2-yl]methyl]-2-(6-phenylimidazo[2,1-b][1,3]thiazol-3-yl)-N-[(3S)-thiolan-3-yl]acetamide
—— (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]prop-2-enamide —— C23H28FN3O2S
(E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]prop-2-enamide
—— (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide —— C23H28FN3O2S
(E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide
—— 2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]acetamide —— C19H24N2O3S2
2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]acetamide
—— 2-[[4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]acetamide —— C20H26N4O3S2
2-[[4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]acetamide
—— 4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-2-phenyl-N-[(3R)-thiolan-3-yl]-1,3-thiazole-5-carboxamide —— C20H24N2O2S2
4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-2-phenyl-N-[(3R)-thiolan-3-yl]-1,3-thiazole-5-carboxamide
—— 2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]acetamide —— C19H24N2O3S2
2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]acetamide
—— 4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-phenyl-N-[(3S)-thiolan-3-yl]-1,3-thiazole-5-carboxamide —— C20H24N2O2S2
4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-phenyl-N-[(3S)-thiolan-3-yl]-1,3-thiazole-5-carboxamide
—— 1-(3-fluorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C22H23FN4O2S2
1-(3-fluorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— methyl 3-[3,5-dimethyl-1-[4-[[(2S)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate —— C25H33N3O4S
methyl 3-[3,5-dimethyl-1-[4-[[(2S)-oxolan-2-yl]methyl-[(3R)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate
—— 2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]acetamide —— C19H24N2O3S2
2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]acetamide
—— methyl 3-[3,5-dimethyl-1-[4-[[(2S)-oxolan-2-yl]methyl-[(3S)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate —— C25H33N3O4S
methyl 3-[3,5-dimethyl-1-[4-[[(2S)-oxolan-2-yl]methyl-[(3S)-thiolan-3-yl]carbamoyl]phenyl]pyrazol-4-yl]propanoate
—— 1-(3-fluorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C22H23FN4O2S2
1-(3-fluorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-2-(4-methoxyphenoxy)acetamide —— C21H22N4O3
N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-2-(4-methoxyphenoxy)acetamide
—— 2-[[4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]acetamide —— C20H26N4O3S2
2-[[4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]acetamide
—— N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]-3-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C18H23N3O3S2
N-[[(2S)-oxolan-2-yl]methyl]-N-[(3S)-thiolan-3-yl]-3-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— 2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]acetamide —— C19H24N2O3S2
2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]acetamide
—— (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide —— C23H28FN3O2S
(E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)-N-[(3S)-thiolan-3-yl]acetamide —— C20H24N2O3S
N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenyl-1,3-oxazol-4-yl)-N-[(3S)-thiolan-3-yl]acetamide
—— N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-(furan-2-yl)-2-phenylpyrazole-3-carboxamide —— C23H19N3O3
N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-(furan-2-yl)-2-phenylpyrazole-3-carboxamide
—— methyl 3-[1-[4-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methylcarbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C25H27N3O4
methyl 3-[1-[4-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methylcarbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-1-phenyl-3-thiophen-2-ylpyrazole-4-carboxamide —— C23H19N3O2S
N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-1-phenyl-3-thiophen-2-ylpyrazole-4-carboxamide
—— N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-(furan-2-yl)-2-phenylpyrazole-3-carboxamide —— C23H19N3O3
N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-(furan-2-yl)-2-phenylpyrazole-3-carboxamide
—— (E)-N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C23H22FN3O2
(E)-N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— 1-(4-bromophenyl)-N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide —— C20H18BrN3O2
1-(4-bromophenyl)-N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide
—— (E)-N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C23H22FN3O2
(E)-N-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl]-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— 2-(2,5-dimethylphenoxy)-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]acetamide —— C19H20N6O2
2-(2,5-dimethylphenoxy)-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]acetamide
—— 1-(3-chlorophenyl)-N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide —— C20H18ClN3O2
1-(3-chlorophenyl)-N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-5-methylpyrazole-4-carboxamide
—— (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]prop-2-enamide —— C21H17ClF4N4O2
(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]prop-2-enamide
—— (Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]prop-2-enamide —— C21H17ClF4N4O2
(Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]prop-2-enamide
—— (Z)-N-(3-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide —— C25H26FN3O3S
(Z)-N-(3-cyclopentylsulfonylphenyl)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enamide
—— methyl 5-[[[(Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]amino]methyl]-2-methylfuran-3-carboxylate —— C21H19ClFN3O4
methyl 5-[[[(Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]amino]methyl]-2-methylfuran-3-carboxylate
—— methyl 3-[1-[4-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methylcarbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C25H27N3O4
methyl 3-[1-[4-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methylcarbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— (3R)-N-[(2R)-2-morpholin-4-ylpropyl]-2,3-diphenyl-3,4-dihydropyrazole-5-carboxamide —— C23H28N4O2
(3R)-N-[(2R)-2-morpholin-4-ylpropyl]-2,3-diphenyl-3,4-dihydropyrazole-5-carboxamide
—— N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-4-(3,4-dimethoxyphenyl)-1-phenylpyrazole-3-carboxamide —— C27H25N3O4
N-[[(2R)-2,3-dihydro-1-benzofuran-2-yl]methyl]-4-(3,4-dimethoxyphenyl)-1-phenylpyrazole-3-carboxamide
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)butanamide —— C20H19ClN6O2
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)butanamide