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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(2,3-Diethoxyphenoxy)methyl]-4-methyl-5-(4-methylsulfonylphenyl)-1,3-oxazole —— C22H25NO6S
2-[(2,3-Diethoxyphenoxy)methyl]-4-methyl-5-(4-methylsulfonylphenyl)-1,3-oxazole
—— 4-(2-amino-2-oxoethoxy)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methoxybenzamide —— C22H23FN4O4
4-(2-amino-2-oxoethoxy)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methoxybenzamide
—— 2-[2-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)acetamide —— C20H22FN5O3S
2-[2-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)acetamide
—— 4-(2-amino-2-oxoethoxy)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methoxybenzamide —— C22H23FN4O4
4-(2-amino-2-oxoethoxy)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methoxybenzamide
—— N,N-diethyl-4-(4-fluorophenyl)-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]-1,3-oxazol-2-amine —— C25H26FN5O
N,N-diethyl-4-(4-fluorophenyl)-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]-1,3-oxazol-2-amine
—— 1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-(2,4-dichlorophenyl)urea —— C21H22Cl2N4O
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-(2,4-dichlorophenyl)urea
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-(5-methylpyrazol-1-yl)benzamide —— C23H22FN5O
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-(5-methylpyrazol-1-yl)benzamide
—— N-isobutyryl-N-(1-(1-(4-methoxyphenyl)-5(4-methylphenyl)pyrazol-3-yl)-1-butyn-3-yl)hydroxylamine —— C25H27N3O3
N-isobutyryl-N-(1-(1-(4-methoxyphenyl)-5(4-methylphenyl)pyrazol-3-yl)-1-butyn-3-yl)hydroxylamine
—— 3-(4-methoxyphenyl)-5-(3-morpholin-4-yl-2-oxopropyl)-1H-indeno[1,2-c]pyrazol-4-one —— C24H23N3O4
3-(4-methoxyphenyl)-5-(3-morpholin-4-yl-2-oxopropyl)-1H-indeno[1,2-c]pyrazol-4-one
—— 5-(4-methylsulfonylphenyl)-3-(4-thiophen-3-ylphenyl)-4-(trifluoromethyl)-1H-pyrazole —— C21H15F3N2O2S2
5-(4-methylsulfonylphenyl)-3-(4-thiophen-3-ylphenyl)-4-(trifluoromethyl)-1H-pyrazole
—— 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-oxobutanamide —— C24H24FN3O4
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-oxobutanamide
—— N'-[(2R)-2-(4-fluorophenoxy)propanoyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carbohydrazide —— C21H18F4N4O3
N'-[(2R)-2-(4-fluorophenoxy)propanoyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carbohydrazide
—— 2-[2-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)acetamide —— C20H22FN5O3S
2-[2-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)acetamide
—— 6-[4-[5-(4-Methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]butyl-propylamino]-5,6,7,8-tetrahydronaphthalene-1-carbonitrile —— C28H35N5O
6-[4-[5-(4-Methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]butyl-propylamino]-5,6,7,8-tetrahydronaphthalene-1-carbonitrile
—— 3-[4-(cyclopropylsulfamoyl)phenyl]-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C24H27FN4O3S
3-[4-(cyclopropylsulfamoyl)phenyl]-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C24H31N5O3S
N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— N-[4-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-1-cyclohexene-1-carboxamide —— C18H15F6N3O
N-[4-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-1-cyclohexene-1-carboxamide
—— 1,5-bis-(3-indolyl)-4-phenyl-1,3-dihydroimidazol-2-one —— C25H18N4O
1,5-bis-(3-indolyl)-4-phenyl-1,3-dihydroimidazol-2-one
—— 8-(4-fluorophenyl)-2-(2-methyl-2H-[1,2,4]triazol-3-ylmethoxy)-3-phenyl-imidazo[1,2-d][1,2,4]triazine 327985-41-1 C21H16FN7O
8-(4-fluorophenyl)-2-(2-methyl-2H-[1,2,4]triazol-3-ylmethoxy)-3-phenyl-imidazo[1,2-d][1,2,4]triazine
—— 2-[[5-[3-(Benzimidazol-1-ylmethyl)phenyl]tetrazol-2-yl]methyl]benzoic acid —— C23H18N6O2
2-[[5-[3-(Benzimidazol-1-ylmethyl)phenyl]tetrazol-2-yl]methyl]benzoic acid
—— 5-(2-methylsulfanylethyl)-8-(3,4,5-trimethoxyphenyl)-7H-[1,2,4]triazolo[5,1-f]purine —— C18H20N6O3S
5-(2-methylsulfanylethyl)-8-(3,4,5-trimethoxyphenyl)-7H-[1,2,4]triazolo[5,1-f]purine
—— 2-(4-chlorophenyl)-N-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propyl]-1,3-thiazole-4-carboxamide —— C19H24ClN3O2S
2-(4-chlorophenyl)-N-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propyl]-1,3-thiazole-4-carboxamide
—— 4-[2-(4-Fluorophenyl)pyrazolo[1,5-a]pyridin-3-yl]-N-[2-(1H-imidazol-5-yl)ethyl]-2-pyrimidinamine 401816-71-5 C22H18FN7
4-[2-(4-Fluorophenyl)pyrazolo[1,5-a]pyridin-3-yl]-N-[2-(1H-imidazol-5-yl)ethyl]-2-pyrimidinamine
—— 4-(3-methoxyphenyl)-3-tridecyl-1H-1,2,4-triazole-5-thione —— C22H35N3OS
4-(3-methoxyphenyl)-3-tridecyl-1H-1,2,4-triazole-5-thione
—— 5-(4-fluorophenyl)-2-[(1S)-1-(oxan-2-yloxy)ethyl]-4-(1H-pyrazol-5-yl)-1,3-thiazole —— C19H20FN3O2S
5-(4-fluorophenyl)-2-[(1S)-1-(oxan-2-yloxy)ethyl]-4-(1H-pyrazol-5-yl)-1,3-thiazole
—— 2-(4-chlorophenyl)-N-[3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propyl]-1,3-thiazole-4-carboxamide —— C19H24ClN3O2S
2-(4-chlorophenyl)-N-[3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propyl]-1,3-thiazole-4-carboxamide
—— 3-[1-(3,5-Difluorophenyl)pyrazol-4-yl]-1-methyl-1-[1-(2-methylpropanoyl)piperidin-4-yl]urea —— C20H25F2N5O2
3-[1-(3,5-Difluorophenyl)pyrazol-4-yl]-1-methyl-1-[1-(2-methylpropanoyl)piperidin-4-yl]urea
—— 2-(4-chlorophenyl)-N-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propyl]-1,3-thiazole-4-carboxamide —— C19H24ClN3O2S
2-(4-chlorophenyl)-N-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propyl]-1,3-thiazole-4-carboxamide
—— 5-(2-methoxyethyl)-8-(3,4,5-trimethoxyphenyl)-7H-[1,2,4]triazolo[5,1-f]purine —— C18H20N6O4
5-(2-methoxyethyl)-8-(3,4,5-trimethoxyphenyl)-7H-[1,2,4]triazolo[5,1-f]purine
—— 4-[4-(2,3-dihydro-1-benzofuran-6-yl)-5-pyridin-2-yl-1H-imidazol-2-yl]benzoic acid —— C23H17N3O3
4-[4-(2,3-dihydro-1-benzofuran-6-yl)-5-pyridin-2-yl-1H-imidazol-2-yl]benzoic acid
—— 2-[2-(4-chlorophenyl)-5,6-dihydro-4H-imidazo[1,2-a][1]benzazepin-1-yl]-N,N-dimethylacetamide —— C22H22ClN3O
2-[2-(4-chlorophenyl)-5,6-dihydro-4H-imidazo[1,2-a][1]benzazepin-1-yl]-N,N-dimethylacetamide
—— [(3S)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-[5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]methanone —— C26H24F3N5O
[(3S)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-[5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]methanone
—— 6-Cyclobutyl-3-(4-fluorophenyl)-5-[(1-methyl-1,2,4-triazol-3-yl)methoxy]triazolo[1,5-a]pyrimidine —— C19H18FN7O
6-Cyclobutyl-3-(4-fluorophenyl)-5-[(1-methyl-1,2,4-triazol-3-yl)methoxy]triazolo[1,5-a]pyrimidine
—— (3-Phenyl-[1,2,4]triazolo[3,4-a]isoquinolin-6-yl)-pyrrolidin-1-ylmethanone —— C21H18N4O
(3-Phenyl-[1,2,4]triazolo[3,4-a]isoquinolin-6-yl)-pyrrolidin-1-ylmethanone
—— N-methyl-2-[2-(4-methylphenyl)-5,6-dihydro-4H-imidazo[1,2-a][1]benzazepin-1-yl]acetamide —— C22H23N3O
N-methyl-2-[2-(4-methylphenyl)-5,6-dihydro-4H-imidazo[1,2-a][1]benzazepin-1-yl]acetamide
—— 3-methyl-N-[(1S)-1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-4-(tetrazol-1-yl)benzamide —— C21H23N5O
3-methyl-N-[(1S)-1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-4-(tetrazol-1-yl)benzamide
—— (3Z)-3-[[2-(3,4-dimethylphenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-4-oxocyclohexa-1,5-diene-1-carboxylic acid —— C19H18N4O4
(3Z)-3-[[2-(3,4-dimethylphenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-4-oxocyclohexa-1,5-diene-1-carboxylic acid
—— 5-(2-Chloro-6-methoxy-3-pyridyl)-1-(4-methylsulfonylphenyl)imidazole(30 % yield) —— C16H14ClN3O3S
5-(2-Chloro-6-methoxy-3-pyridyl)-1-(4-methylsulfonylphenyl)imidazole(30 % yield)
—— N-[2-[4-[3-(1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]phenyl]ethyl]propanamide —— C20H19N3O4
N-[2-[4-[3-(1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]phenyl]ethyl]propanamide
—— N-(diaminomethylidene)-4-imidazol-1-yl-3-(trifluoromethyl)benzamide —— C12H10F3N5O
N-(diaminomethylidene)-4-imidazol-1-yl-3-(trifluoromethyl)benzamide
—— 3-methyl-N-[(1R)-1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-4-(tetrazol-1-yl)benzamide —— C21H23N5O
3-methyl-N-[(1R)-1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-4-(tetrazol-1-yl)benzamide
—— N'-[(3R)-5-oxo-1-phenylpyrrolidine-3-carbonyl]-1,3-diphenylpyrazole-4-carbohydrazide —— C27H23N5O3
N'-[(3R)-5-oxo-1-phenylpyrrolidine-3-carbonyl]-1,3-diphenylpyrazole-4-carbohydrazide
—— 3-[4-(2-propoxy-1H-imidazol-5-yl)phenyl]-5-(trifluoromethyl)-1,2,4-oxadiazole —— C15H13F3N4O2
3-[4-(2-propoxy-1H-imidazol-5-yl)phenyl]-5-(trifluoromethyl)-1,2,4-oxadiazole
—— 5-methyl-1-(2-methylphenyl)-N-[3-[(1S)-1-phenylethoxy]propyl]pyrazole-4-carboxamide —— C23H27N3O2
5-methyl-1-(2-methylphenyl)-N-[3-[(1S)-1-phenylethoxy]propyl]pyrazole-4-carboxamide
—— [4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]phenyl]methanamine —— C17H17N3O
[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]phenyl]methanamine
—— 2-[[4-(3-chloro-4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]acetamide —— C22H26ClN5O3S
2-[[4-(3-chloro-4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]acetamide
—— 5-methyl-1-(2-methylphenyl)-N-[3-[(1R)-1-phenylethoxy]propyl]pyrazole-4-carboxamide —— C23H27N3O2
5-methyl-1-(2-methylphenyl)-N-[3-[(1R)-1-phenylethoxy]propyl]pyrazole-4-carboxamide
—— 1-Benzyl-5-(4-methylsulfanylphenyl)pyrazol-3-amine —— C17H17N3S
1-Benzyl-5-(4-methylsulfanylphenyl)pyrazol-3-amine
—— 2-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]-N-[(2R)-1-(furan-2-yl)propan-2-yl]acetamide —— C24H22ClN3O2
2-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]-N-[(2R)-1-(furan-2-yl)propan-2-yl]acetamide
—— 2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-1-(furan-2-yl)propan-2-yl]acetamide —— C20H24N4O2S
2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-1-(furan-2-yl)propan-2-yl]acetamide