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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-cyclopropyl-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C26H29N3O
N-cyclopropyl-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-triene-5-carboxamide —— C23H22FN5O2S
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-triene-5-carboxamide
—— 3-(tert-butylsulfamoyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methoxybenzamide —— C24H29FN4O4S
3-(tert-butylsulfamoyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methoxybenzamide
—— 4-(3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide —— C24H24FN5O
4-(3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide
—— 2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C25H27FN6OS
2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide
—— (2R)-2-[2-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)propanamide —— C21H24FN5O3S
(2R)-2-[2-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)propanamide
—— 5-(cyclopenta-2,4-dien-1-ylidenemethyl)-3-prop-2-enyl-2-sulfanylidene-1,3-thiazol-4-olate —— C12H10NOS2-
5-(cyclopenta-2,4-dien-1-ylidenemethyl)-3-prop-2-enyl-2-sulfanylidene-1,3-thiazol-4-olate
—— 4-(3,5-dimethylpyrazol-1-yl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide —— C24H24FN5O
4-(3,5-dimethylpyrazol-1-yl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]benzamide
—— 2-[2-(2-ethoxyphenyl)-1,3-thiazol-4-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C25H25FN4O2S
2-[2-(2-ethoxyphenyl)-1,3-thiazol-4-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide
—— 2-chloro-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-(propan-2-ylsulfamoyl)benzamide —— C22H24ClFN4O3S
2-chloro-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-(propan-2-ylsulfamoyl)benzamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-[methyl(propan-2-yl)sulfamoyl]benzamide —— C23H27FN4O3S
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-[methyl(propan-2-yl)sulfamoyl]benzamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2,2-dioxo-3,4-dihydropyrido[2,1-c][1,2,4]thiadiazine-7-carboxamide —— C20H20FN5O3S
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2,2-dioxo-3,4-dihydropyrido[2,1-c][1,2,4]thiadiazine-7-carboxamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methoxy-1-[3-(trifluoromethyl)phenyl]pyrazole-3-carboxamide —— C24H21F4N5O2
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methoxy-1-[3-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2,2-dioxo-3,4-dihydropyrido[2,1-c][1,2,4]thiadiazine-7-carboxamide —— C20H20FN5O3S
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2,2-dioxo-3,4-dihydropyrido[2,1-c][1,2,4]thiadiazine-7-carboxamide
—— methyl 3-[1-[4-[[(1R)-1-(3-chlorophenyl)ethyl]-methylcarbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C25H28ClN3O3
methyl 3-[1-[4-[[(1R)-1-(3-chlorophenyl)ethyl]-methylcarbamoyl]phenyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— 2-(3,4-dimethylphenoxy)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C22H24FN3O2
2-(3,4-dimethylphenoxy)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide
—— (2S)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C23H24F2N4O2S
(2S)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— 2-cyclopropyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide —— C24H24FN5OS
2-cyclopropyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
—— N-[(1R)-1-(3-chlorophenyl)ethyl]-N-methyl-3-nitro-4-(1,2,4-triazol-1-yl)benzamide —— C18H16ClN5O3
N-[(1R)-1-(3-chlorophenyl)ethyl]-N-methyl-3-nitro-4-(1,2,4-triazol-1-yl)benzamide
—— (2R)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C23H24F2N4O2S
(2R)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— 3-(4-fluorophenyl)-4-[(E)-(2,4,6-trimethoxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C18H17FN4O3S
3-(4-fluorophenyl)-4-[(E)-(2,4,6-trimethoxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 4-(2-amino-2-oxoethoxy)-3-chloro-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-methoxybenzamide —— C22H22ClFN4O4
4-(2-amino-2-oxoethoxy)-3-chloro-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-methoxybenzamide
—— (2R)-2-[2-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)propanamide —— C21H24FN5O3S
(2R)-2-[2-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)propanamide
—— 3-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C24H22ClFN4O2
3-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— (2S)-2-[2-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)propanamide —— C21H24FN5O3S
(2S)-2-[2-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-oxoethyl]sulfanyl-N-(5-methyl-1,2-oxazol-3-yl)propanamide
—— N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-2-(2-phenyl-1,3-thiazol-4-yl)acetamide —— C22H21ClN2OS
N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
—— (3R)-3-acetamido-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(4-methylphenyl)propanamide —— C24H27FN4O2
(3R)-3-acetamido-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(4-methylphenyl)propanamide
—— N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]-5-ethyl-1-(4-methylphenyl)pyrazole-4-carboxamide —— C23H27N3O3
N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]-5-ethyl-1-(4-methylphenyl)pyrazole-4-carboxamide
—— N-[(1S)-1-(4-cyanophenyl)ethyl]-N-ethyl-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide —— C22H21FN4OS
N-[(1S)-1-(4-cyanophenyl)ethyl]-N-ethyl-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-triene-5-carboxamide —— C23H22FN5O2S
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-triene-5-carboxamide
—— N-ethyl-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C24H24N4O2S
N-ethyl-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— 2-[2-(2-ethoxyphenyl)-1,3-thiazol-4-yl]-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C25H25FN4O2S
2-[2-(2-ethoxyphenyl)-1,3-thiazol-4-yl]-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide
—— 1-(3-chlorophenyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-methylpyrazole-4-carboxamide —— C23H21ClFN5O
1-(3-chlorophenyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-methylpyrazole-4-carboxamide
—— N-[(1R)-1-(4-cyanophenyl)ethyl]-N-ethyl-1-(3-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C24H20FN5OS
N-[(1R)-1-(4-cyanophenyl)ethyl]-N-ethyl-1-(3-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)acetamide —— C23H27FN4O3S2
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)acetamide
—— (3S)-1-(3,4-dimethoxyphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-oxopyrrolidine-3-carboxamide —— C25H27FN4O4
(3S)-1-(3,4-dimethoxyphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-oxopyrrolidine-3-carboxamide
—— 4-fluoro-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(prop-2-enylsulfamoyl)benzamide —— C22H22F2N4O3S
4-fluoro-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(prop-2-enylsulfamoyl)benzamide
—— N-[(E)-1-(2-fluorophenyl)ethylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide —— C17H15FN6O
N-[(E)-1-(2-fluorophenyl)ethylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)propanamide —— C24H28FN3O4
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)propanamide
—— 5-(2,2-dimethylpropanoylamino)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methylthiophene-2-carboxamide —— C23H27FN4O2S
5-(2,2-dimethylpropanoylamino)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methylthiophene-2-carboxamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-(trifluoromethoxy)benzamide —— C20H17F4N3O2
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-(trifluoromethoxy)benzamide
—— 2-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C22H23FN6O2S
2-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methoxy-5-methylbenzamide —— C21H22FN3O2
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methoxy-5-methylbenzamide
—— 5-chloro-1-[(4-fluorophenyl)methyl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methylpyrazole-4-carboxamide —— C24H22ClF2N5O
5-chloro-1-[(4-fluorophenyl)methyl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methylpyrazole-4-carboxamide
—— 3-cyclohexyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C21H28FN3O
3-cyclohexyl-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— N-[(1R)-1-(4-cyanophenyl)ethyl]-N-ethyl-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide —— C22H21FN4OS
N-[(1R)-1-(4-cyanophenyl)ethyl]-N-ethyl-3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxamide
—— 3-(3-bromo-4-methoxyphenyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C22H23BrFN3O2
3-(3-bromo-4-methoxyphenyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(5-methyl-1,2,4-oxadiazol-3-yl)methylsulfanyl]benzamide —— C23H22FN5O2S
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-[(5-methyl-1,2,4-oxadiazol-3-yl)methylsulfanyl]benzamide
—— 3-(3-bromo-4-methoxyphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C22H23BrFN3O2
3-(3-bromo-4-methoxyphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— 2-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide —— C22H23FN6O2S
2-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]acetamide