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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(1,3-benzothiazol-2-yl)-3-[5-(4-methylphenyl)-1,3-oxazol-2-yl]-N-[[(2S)-oxolan-2-yl]methyl]propanamide —— C25H25N3O3S
N-(1,3-benzothiazol-2-yl)-3-[5-(4-methylphenyl)-1,3-oxazol-2-yl]-N-[[(2S)-oxolan-2-yl]methyl]propanamide
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylphenyl]-2-oxoacetamide —— C26H30N4O4S
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylphenyl]-2-oxoacetamide
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylphenyl]-2-oxoacetamide —— C26H30N4O4S
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylphenyl]-2-oxoacetamide
—— 2-chloro-N-[5-(5,7-dimethyl-1,3-benzoxazol-2-yl)-2-methylphenyl]-5-nitrobenzenesulfonamide —— C22H18ClN3O5S
2-chloro-N-[5-(5,7-dimethyl-1,3-benzoxazol-2-yl)-2-methylphenyl]-5-nitrobenzenesulfonamide
—— [(1R)-2-amino-2-oxo-1-phenylethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate —— C19H16FN3O3S
[(1R)-2-amino-2-oxo-1-phenylethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate
—— [(3S)-1-ethylpiperidin-3-yl] 3-[5-(2,4-dichlorophenyl)-1,3-oxazol-2-yl]propanoate —— C19H22Cl2N2O3
[(3S)-1-ethylpiperidin-3-yl] 3-[5-(2,4-dichlorophenyl)-1,3-oxazol-2-yl]propanoate
—— (3-methyl-1-phenylthieno[2,3-c]pyrazol-5-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone —— C24H26N6OS
(3-methyl-1-phenylthieno[2,3-c]pyrazol-5-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone
—— 3-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]propanamide —— C22H27FN2O2
3-[5-(4-fluorophenyl)-1,3-oxazol-2-yl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]propanamide
—— 4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)(4-ethoxy-2-hydroxyphenyl)methyl]-1,5-dimethyl-2-phenyl-1,2-dihydro-3H-pyrazol-3-one —— C31H32N4O4
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)(4-ethoxy-2-hydroxyphenyl)methyl]-1,5-dimethyl-2-phenyl-1,2-dihydro-3H-pyrazol-3-one
—— (3aR)-3a-[(E)-2-[(3S)-2,3-diphenyl-3,4-dihydropyrazol-5-yl]ethenyl]-4,4-dimethyl-1,2-dihydro-[1,3]oxazolo[3,2-a]indole —— C29H29N3O
(3aR)-3a-[(E)-2-[(3S)-2,3-diphenyl-3,4-dihydropyrazol-5-yl]ethenyl]-4,4-dimethyl-1,2-dihydro-[1,3]oxazolo[3,2-a]indole
—— [(2S)-1-oxo-1-(pyrimidin-2-ylamino)propan-2-yl] (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enoate —— C21H20FN5O3
[(2S)-1-oxo-1-(pyrimidin-2-ylamino)propan-2-yl] (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enoate
—— [(2R)-1-oxo-1-(pyrimidin-2-ylamino)propan-2-yl] (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enoate —— C21H20FN5O3
[(2R)-1-oxo-1-(pyrimidin-2-ylamino)propan-2-yl] (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enoate
—— 3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propan-1-one —— C18H20F2N2O3
3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propan-1-one
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]propanamide —— C21H25ClN2O2
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]propanamide
—— [(1S)-2-amino-2-oxo-1-phenylethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate —— C19H16FN3O3S
[(1S)-2-amino-2-oxo-1-phenylethyl] 3-(4-fluorophenyl)-2-methylsulfanylimidazole-4-carboxylate
—— 1-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-2-[(1-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethanone —— C20H24N4O2S
1-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-2-[(1-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethanone
—— (2S)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide —— C25H28FN3O2S
(2S)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide
—— 1-[(2S)-2-ethylpiperidin-1-yl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylethanone —— C23H31N3O2S
1-[(2S)-2-ethylpiperidin-1-yl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylethanone
—— 2-(4-chlorophenyl)-5-[[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylmethyl]-1,3,4-oxadiazole —— C23H21ClN4O2S
2-(4-chlorophenyl)-5-[[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylmethyl]-1,3,4-oxadiazole
—— 3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-1-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propan-1-one —— C18H20F2N2O3
3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-1-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propan-1-one
—— (2R)-2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-phenylacetamide —— C16H14BrN5OS
(2R)-2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-phenylacetamide
—— (3-methyl-1-phenylthieno[2,3-c]pyrazol-5-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone —— C24H26N6OS
(3-methyl-1-phenylthieno[2,3-c]pyrazol-5-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone
—— 3,3-dimethyl-1-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylbutan-2-one —— C20H26N2O2S
3,3-dimethyl-1-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylbutan-2-one
—— (5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl 2-[(Z)-1-(1,3-benzodioxol-5-yl)ethylideneamino]oxyacetate —— C22H20N2O6
(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl 2-[(Z)-1-(1,3-benzodioxol-5-yl)ethylideneamino]oxyacetate
—— (2R)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide —— C25H28FN3O2S
(2R)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]propanamide —— C21H25ClN2O2
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]propanamide
—— (2R)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide —— C25H28FN3O2S
(2R)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide
—— 3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-1-[(2S,6R)-2,6-dimethylmorpholin-4-yl]propan-1-one —— C18H20F2N2O3
3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-1-[(2S,6R)-2,6-dimethylmorpholin-4-yl]propan-1-one
—— (2S)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide —— C25H28FN3O2S
(2S)-N-[(3-fluorophenyl)methyl]-N-methyl-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide
—— 1-[(2R)-2-ethylpiperidin-1-yl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylethanone —— C23H31N3O2S
1-[(2R)-2-ethylpiperidin-1-yl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylethanone
—— (2R)-2-[[4-benzyl-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-pyrimidin-2-ylpropanamide —— C22H19ClN6OS
(2R)-2-[[4-benzyl-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-pyrimidin-2-ylpropanamide
—— (2S)-2-[[4-benzyl-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-pyrimidin-2-ylpropanamide —— C22H19ClN6OS
(2S)-2-[[4-benzyl-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-pyrimidin-2-ylpropanamide
—— 3,3-dimethyl-1-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylbutan-2-one —— C20H26N2O2S
3,3-dimethyl-1-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylbutan-2-one
—— 1-[(2R)-2-ethylpiperidin-1-yl]-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylethanone —— C23H31N3O2S
1-[(2R)-2-ethylpiperidin-1-yl]-2-[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylethanone
—— 5-(3-amino-4,6-dimethylthieno[2,3-b]pyridin-2-yl)-4-phenyl-2,4-dihydro-3H-1,2,4-triazole-3-thione —— C17H15N5S2
5-(3-amino-4,6-dimethylthieno[2,3-b]pyridin-2-yl)-4-phenyl-2,4-dihydro-3H-1,2,4-triazole-3-thione
—— (4R)-6-amino-4-(3,5-dimethoxyphenyl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C22H20N4O4
(4R)-6-amino-4-(3,5-dimethoxyphenyl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4R)-6-amino-3-(2-chlorophenyl)-4-(4-cyclopentyloxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C25H23ClN4O3
(4R)-6-amino-3-(2-chlorophenyl)-4-(4-cyclopentyloxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4R)-6-amino-3-(2-chlorophenyl)-4-(4-hydroxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C20H15ClN4O3
(4R)-6-amino-3-(2-chlorophenyl)-4-(4-hydroxy-3-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4R)-6-amino-3-(4-fluorophenyl)-4-quinolin-4-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C22H14FN5O
(4R)-6-amino-3-(4-fluorophenyl)-4-quinolin-4-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (4S)-6-amino-4-(4-cyclopentyloxy-3-methoxyphenyl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C25H23FN4O3
(4S)-6-amino-4-(4-cyclopentyloxy-3-methoxyphenyl)-3-(4-fluorophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (3R,3aR)-3-(1,3-diphenylpyrazol-4-yl)-2-phenyl-3,3a,4,5-tetrahydrobenzo[g]indazole —— C32H26N4
(3R,3aR)-3-(1,3-diphenylpyrazol-4-yl)-2-phenyl-3,3a,4,5-tetrahydrobenzo[g]indazole
—— 2-[bis(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)methyl]benzoate —— C28H23N4O4-
2-[bis(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)methyl]benzoate
—— (4S)-6-amino-3-(2,4-dimethylphenyl)-4-(2-propan-2-yloxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C24H24N4O2
(4S)-6-amino-3-(2,4-dimethylphenyl)-4-(2-propan-2-yloxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (5E)-2-(3-butyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)-3-ethyl-5-[(2Z)-2-(3-ethyl-4-methyl-6-phenylimidazo[4,5-d][1,3]thiazol-4-ium-2-ylidene)ethylidene]-1,3-thiazolidin-4-one —— C27H30N5O2S4+
(5E)-2-(3-butyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)-3-ethyl-5-[(2Z)-2-(3-ethyl-4-methyl-6-phenylimidazo[4,5-d][1,3]thiazol-4-ium-2-ylidene)ethylidene]-1,3-thiazolidin-4-one
—— (4S)-6-amino-4-(6-chloro-1,3-benzodioxol-5-yl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C21H15ClN4O4
(4S)-6-amino-4-(6-chloro-1,3-benzodioxol-5-yl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]methyl]acetamide —— C21H23FN4O3
2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]methyl]acetamide
—— (4S)-6-amino-3-(4-fluorophenyl)-4-naphthalen-1-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C23H15FN4O
(4S)-6-amino-3-(4-fluorophenyl)-4-naphthalen-1-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 2-[1-(3-methoxyphenyl)imidazol-2-yl]sulfanyl-N-[(3S)-2-methyl-4-oxopentan-3-yl]acetamide —— C18H23N3O3S
2-[1-(3-methoxyphenyl)imidazol-2-yl]sulfanyl-N-[(3S)-2-methyl-4-oxopentan-3-yl]acetamide
—— N-[(1S)-1-(4-ethoxyphenyl)ethyl]-3-[5-(4-methylphenyl)-1,3-oxazol-2-yl]propanamide —— C23H26N2O3
N-[(1S)-1-(4-ethoxyphenyl)ethyl]-3-[5-(4-methylphenyl)-1,3-oxazol-2-yl]propanamide
—— N-[(1S)-1-(1,3-benzodioxol-5-yl)ethyl]-1-benzyl-3-phenylpyrazole-4-carboxamide —— C26H23N3O3
N-[(1S)-1-(1,3-benzodioxol-5-yl)ethyl]-1-benzyl-3-phenylpyrazole-4-carboxamide