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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide —— C23H21F3N4O3
3-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]propanamide
—— [(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone —— C22H23FN4OS
[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone
—— [(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone —— C22H23FN4OS
[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[1-(4-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone
—— (2R)-2-[5-(4-bromophenyl)tetrazol-2-yl]-N-pyrimidin-2-ylpropanamide —— C14H12BrN7O
(2R)-2-[5-(4-bromophenyl)tetrazol-2-yl]-N-pyrimidin-2-ylpropanamide
—— 1-(4-fluorophenyl)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C18H17FN4O3S2
1-(4-fluorophenyl)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— 2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-2-methyl-4-oxopentan-3-yl]acetamide —— C21H27FN4O3S
2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-2-methyl-4-oxopentan-3-yl]acetamide
—— (E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C27H29FN4O
(E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— N-[(3S)-2-methyl-4-oxopentan-3-yl]-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C20H27N3O2S
N-[(3S)-2-methyl-4-oxopentan-3-yl]-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— (Z,1R,4S)-N-[(Z)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C21H24ClFN4
(Z,1R,4S)-N-[(Z)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide —— C28H26N4O3
N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide
—— 2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-2-methyl-4-oxopentan-3-yl]acetamide —— C21H27FN4O3S
2-[[5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-2-methyl-4-oxopentan-3-yl]acetamide
—— (Z,1S,4R)-N-[(Z)-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C27H30N4O
(Z,1S,4R)-N-[(Z)-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— (4S)-6-amino-4-(4-bromophenyl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C21H17BrN4O
(4S)-6-amino-4-(4-bromophenyl)-3-(2,4-dimethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (3S)-1-cyclopentyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide —— C21H23F3N4O2
(3S)-1-cyclopentyl-N-[5-methyl-2-[3-(trifluoromethyl)phenyl]pyrazol-3-yl]-5-oxopyrrolidine-3-carboxamide
—— [4-[(4R)-6-amino-5-cyano-3-(3,4,5-trimethoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]phenyl] furan-2-carboxylate —— C27H22N4O7
[4-[(4R)-6-amino-5-cyano-3-(3,4,5-trimethoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]phenyl] furan-2-carboxylate
—— [2-[[(1S,2S)-2-methylcyclohexyl]amino]-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate —— C20H24FN3O3S
[2-[[(1S,2S)-2-methylcyclohexyl]amino]-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate
—— [4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]-[(1S,2R)-2-(2-fluorophenyl)cyclopropyl]methanone —— C23H22ClFN4O2
[4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]-[(1S,2R)-2-(2-fluorophenyl)cyclopropyl]methanone
—— ethyl N-[2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetyl]carbamate —— C17H21N3O3S
ethyl N-[2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetyl]carbamate
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-quinolin-8-ylacetate —— C25H24N4O4
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-quinolin-8-ylacetate
—— N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-methylacetamide —— C22H24N4O3S
N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[4-(3,4-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-methylacetamide
—— (2R)-N-cyclopentyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylpropanamide —— C20H27N3OS
(2R)-N-cyclopentyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylpropanamide
—— N-(2,6-dimethylphenyl)-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C22H25N3OS
N-(2,6-dimethylphenyl)-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— N-(1,3-benzodioxol-5-yl)-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C21H21N3O3S
N-(1,3-benzodioxol-5-yl)-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— [4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]-[(1S,2S)-2-(2-fluorophenyl)cyclopropyl]methanone —— C23H22ClFN4O2
[4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]-[(1S,2S)-2-(2-fluorophenyl)cyclopropyl]methanone
—— N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide —— C28H26N4O3
N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide
—— (1R,2R)-N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-(2-fluorophenyl)cyclopropane-1-carboxamide —— C27H24FN3O
(1R,2R)-N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-(2-fluorophenyl)cyclopropane-1-carboxamide
—— [2-(1-Ethyl-2,5-dimethylpyrrol-3-yl)-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate —— C21H22FN3O3S
[2-(1-Ethyl-2,5-dimethylpyrrol-3-yl)-2-oxoethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate
—— N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C19H25N3O3S2
N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— (3-Fluoro-4-methoxyphenyl)methyl 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate —— C19H16F2N2O3S
(3-Fluoro-4-methoxyphenyl)methyl 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate
—— N-[(1R)-1-(1,3-benzodioxol-5-yl)ethyl]-3-(1-phenylpyrazol-4-yl)propanamide —— C21H21N3O3
N-[(1R)-1-(1,3-benzodioxol-5-yl)ethyl]-3-(1-phenylpyrazol-4-yl)propanamide
—— N-[(1S)-1-(1,3-benzodioxol-5-yl)ethyl]-3-(1-phenylpyrazol-4-yl)propanamide —— C21H21N3O3
N-[(1S)-1-(1,3-benzodioxol-5-yl)ethyl]-3-(1-phenylpyrazol-4-yl)propanamide
—— [(1S,2R)-2-(4-fluorophenyl)cyclopropyl]-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methanone —— C24H25FN4O2
[(1S,2R)-2-(4-fluorophenyl)cyclopropyl]-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methanone
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-methyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C19H25N3O3S2
N-[(3S)-1,1-dioxothiolan-3-yl]-N-methyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— (2S)-1-(2-tert-butylphenoxy)-3-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]propan-2-ol —— C24H32N4O2
(2S)-1-(2-tert-butylphenoxy)-3-[methyl-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]propan-2-ol
—— [4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]-[(1R,2R)-2-(2-fluorophenyl)cyclopropyl]methanone —— C23H22ClFN4O2
[4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]-[(1R,2R)-2-(2-fluorophenyl)cyclopropyl]methanone
—— 2-[1-(4-Propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C14H17N3OS
2-[1-(4-Propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— [2-Oxo-2-(propylamino)ethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate —— C16H18FN3O3S
[2-Oxo-2-(propylamino)ethyl] 2-[1-(3-fluorophenyl)imidazol-2-yl]sulfanylacetate
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C20H27N3O3S2
N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— (2R)-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylpropanamide —— C15H19N3OS
(2R)-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylpropanamide
—— (1S,2R)-N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-(2-fluorophenyl)cyclopropane-1-carboxamide —— C27H24FN3O
(1S,2R)-N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-(2-fluorophenyl)cyclopropane-1-carboxamide
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 4-(5-methylthiophen-2-yl)-4-oxobutanoate —— C19H16ClNO4S
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 4-(5-methylthiophen-2-yl)-4-oxobutanoate
—— [3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(5-methylthiophen-2-yl)-4-oxobutanoate —— C18H15FN2O4S
[3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(5-methylthiophen-2-yl)-4-oxobutanoate
—— [(1R,2S)-2-(4-fluorophenyl)cyclopropyl]-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methanone —— C24H25FN4O2
[(1R,2S)-2-(4-fluorophenyl)cyclopropyl]-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methanone
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]butanamide —— C21H21ClF3N5O2
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]butanamide
—— [(1S,2S)-2-(4-fluorophenyl)cyclopropyl]-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methanone —— C24H25FN4O2
[(1S,2S)-2-(4-fluorophenyl)cyclopropyl]-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methanone
—— N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-[(1R,2S,6R,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide —— C28H26N4O3
N-[(1-benzyl-3-phenylpyrazol-4-yl)methyl]-2-[(1R,2S,6R,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide
—— (2S)-1-(2-tert-butylphenoxy)-3-[methyl-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]propan-2-ol —— C24H32N4O2
(2S)-1-(2-tert-butylphenoxy)-3-[methyl-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]amino]propan-2-ol
—— 2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-1-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]ethanone —— C23H30N4O2
2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-1-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]ethanone
—— 2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-1-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]ethanone —— C23H30N4O2
2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-1-[4-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]ethanone
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]butanamide —— C21H21ClF3N5O2
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]butanamide