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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 1-[4-[[(2S)-3-methylbutan-2-yl]carbamoyl]phenyl]-5-(trifluoromethyl)pyrazole-4-carboxylate —— C19H22F3N3O3
ethyl 1-[4-[[(2S)-3-methylbutan-2-yl]carbamoyl]phenyl]-5-(trifluoromethyl)pyrazole-4-carboxylate
—— N-[(2R)-2-(dimethylamino)-3-phenylpropyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide —— C24H30N4O3
N-[(2R)-2-(dimethylamino)-3-phenylpropyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
—— 2-benzyl-N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C24H26FN3O2S
2-benzyl-N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— 4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]butanamide —— C26H32N4O4
4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]butanamide
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-phenyl-2-pyrrolidin-1-ylethyl]butanamide —— C24H27ClN4O2
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-phenyl-2-pyrrolidin-1-ylethyl]butanamide
—— 1-[1-[3-(3,4-Dichlorophenyl)-4-(3-phenyl-1,2,4-triazol-4-yl)butyl]piperidin-4-yl]-1,3-diazinan-2-one —— C27H32Cl2N6O
1-[1-[3-(3,4-Dichlorophenyl)-4-(3-phenyl-1,2,4-triazol-4-yl)butyl]piperidin-4-yl]-1,3-diazinan-2-one
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]butanamide —— C23H27ClN4O3
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-(dimethylamino)-2-(2-methoxyphenyl)ethyl]butanamide
—— ethyl 1-[4-[[(2R)-3-methylbutan-2-yl]carbamoyl]phenyl]-5-(trifluoromethyl)pyrazole-4-carboxylate —— C19H22F3N3O3
ethyl 1-[4-[[(2R)-3-methylbutan-2-yl]carbamoyl]phenyl]-5-(trifluoromethyl)pyrazole-4-carboxylate
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-(dimethylamino)-2-phenylethyl]butanamide —— C22H25ClN4O2
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-(dimethylamino)-2-phenylethyl]butanamide
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-(dimethylamino)-2-(4-ethylphenyl)ethyl]butanamide —— C24H29ClN4O2
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-(dimethylamino)-2-(4-ethylphenyl)ethyl]butanamide
—— ethyl 1-[4-[[(2R)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate —— C24H28N4O4
ethyl 1-[4-[[(2R)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]butanamide —— C22H25ClN4O2S
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]butanamide
—— 2-benzyl-N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C24H26FN3O2S
2-benzyl-N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]butanamide —— C22H25ClN4O2S
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]butanamide
—— N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide —— C22H27N5O3
N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-phenyl-2-pyrrolidin-1-ylethyl]butanamide —— C24H27ClN4O2
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-2-phenyl-2-pyrrolidin-1-ylethyl]butanamide
—— 1-[5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl]-3-[4-(3-morpholin-4-yl-propyl)naphthalen-1-yl]-urea —— C32H39N5O2
1-[5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl]-3-[4-(3-morpholin-4-yl-propyl)naphthalen-1-yl]-urea
—— ethyl 1-[4-[[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate —— C24H28N4O4
ethyl 1-[4-[[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate
—— N-[(2S)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-phenylpyrazole-3-carboxamide —— C23H26N4O2
N-[(2S)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-phenylpyrazole-3-carboxamide
—— N-[(2R)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide —— C21H25N5O3
N-[(2R)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide
—— N-[(2R)-2-(1H-indol-3-yl)-2-thiophen-2-ylethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide —— C27H26N4O3S
N-[(2R)-2-(1H-indol-3-yl)-2-thiophen-2-ylethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
—— N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide —— C22H27N5O3
N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide
—— (2R,5S)-2,5-dimethyl-4-[[3-(3-nitrophenyl)-1,2,4-triazol-1-yl]methyl]morpholine —— C15H19N5O3
(2R,5S)-2,5-dimethyl-4-[[3-(3-nitrophenyl)-1,2,4-triazol-1-yl]methyl]morpholine
—— N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide —— C24H30N4O4
N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
—— N-[(2S)-2-(dimethylamino)-3-phenylpropyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide —— C24H30N4O3
N-[(2S)-2-(dimethylamino)-3-phenylpropyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-(dimethylamino)-2-phenylethyl]butanamide —— C22H25ClN4O2
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-2-(dimethylamino)-2-phenylethyl]butanamide
—— 5-Amino-1-[2,6-dichloro-4-(pentafluoro-lambda6-sulfanyl)phenyl]-4-(trifluoromethylsulfonyl)pyrazole-3-carbonitrile —— C11H4Cl2F8N4O2S2
5-Amino-1-[2,6-dichloro-4-(pentafluoro-lambda6-sulfanyl)phenyl]-4-(trifluoromethylsulfonyl)pyrazole-3-carbonitrile
—— 7-Chloro-2-((E)-2-{3-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)-phenoxymethyl]-phenyl}-vinyl)-quinoline —— C31H23ClN4O
7-Chloro-2-((E)-2-{3-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)-phenoxymethyl]-phenyl}-vinyl)-quinoline
—— N-[(2R)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-phenylpyrazole-3-carboxamide —— C23H26N4O2
N-[(2R)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-phenylpyrazole-3-carboxamide
—— 6-[(E)-2-[7-[(4-tert-butylphenyl)methyl]-2-(4-fluorophenyl)-4,5,6,7-tetrahydroindazol-3-yl]ethenyl]-4-hydroxyoxan-2-one —— C31H35FN2O3
6-[(E)-2-[7-[(4-tert-butylphenyl)methyl]-2-(4-fluorophenyl)-4,5,6,7-tetrahydroindazol-3-yl]ethenyl]-4-hydroxyoxan-2-one
—— N-[(1S)-1-(2,4-dichlorophenyl)ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide —— C21H21Cl2N3O3
N-[(1S)-1-(2,4-dichlorophenyl)ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
—— N-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide —— C21H25N5O3
N-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-1-(3-methoxyphenyl)-5-methyltriazole-4-carboxamide
—— 1-[(3,4-dichlorophenyl)methyl]-5-(4-methylphenyl)-N-[(1S,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]pyrazole-3-carboxamide —— C28H31Cl2N3O
1-[(3,4-dichlorophenyl)methyl]-5-(4-methylphenyl)-N-[(1S,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]pyrazole-3-carboxamide
—— 2-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[5-tert-butyl-2-(3-methylphenyl)pyrazol-3-yl]acetamide —— C24H30N4O3
2-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[5-tert-butyl-2-(3-methylphenyl)pyrazol-3-yl]acetamide
—— 1-[(E)-2-phenylethenyl]sulfonyl-N-(2-pyrazol-1-ylphenyl)piperidine-4-carboxamide —— C23H24N4O3S
1-[(E)-2-phenylethenyl]sulfonyl-N-(2-pyrazol-1-ylphenyl)piperidine-4-carboxamide
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[4-(3-cyanopyridin-2-yl)oxy-2-methylphenyl]butanamide —— C24H20ClN7O2
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[4-(3-cyanopyridin-2-yl)oxy-2-methylphenyl]butanamide
—— (3S)-N-[4-fluoro-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-1-propylsulfonylpiperidine-3-carboxamide —— C22H30FN5O3S
(3S)-N-[4-fluoro-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-1-propylsulfonylpiperidine-3-carboxamide
—— (4R,7R,8S,9S,10E,13Z,16S)-4,8-dihydroxy-5,5,7,9,13-pentamethyl-16-[(E)-1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-6-oxo-1-oxa-6lambda4-thiacyclohexadeca-10,13-dien-2-one —— C26H39NO5S2
(4R,7R,8S,9S,10E,13Z,16S)-4,8-dihydroxy-5,5,7,9,13-pentamethyl-16-[(E)-1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-6-oxo-1-oxa-6lambda4-thiacyclohexadeca-10,13-dien-2-one
—— 2-(2-benzyl-1,3-thiazol-4-yl)-N-[(1R)-1-(4-bromophenyl)ethyl]acetamide —— C20H19BrN2OS
2-(2-benzyl-1,3-thiazol-4-yl)-N-[(1R)-1-(4-bromophenyl)ethyl]acetamide
—— (3R)-1-(4-ethylphenyl)-5-oxo-N-(2-pyrazol-1-ylphenyl)pyrrolidine-3-carboxamide —— C22H22N4O2
(3R)-1-(4-ethylphenyl)-5-oxo-N-(2-pyrazol-1-ylphenyl)pyrrolidine-3-carboxamide
—— (3R)-1-(1,1-dioxo-1,2-benzothiazol-3-yl)-N-(2-pyrazol-1-ylphenyl)piperidine-3-carboxamide —— C22H21N5O3S
(3R)-1-(1,1-dioxo-1,2-benzothiazol-3-yl)-N-(2-pyrazol-1-ylphenyl)piperidine-3-carboxamide
—— (2S)-2-(2,4-dichlorophenoxy)-N-(2-pyrazol-1-ylphenyl)propanamide —— C18H15Cl2N3O2
(2S)-2-(2,4-dichlorophenoxy)-N-(2-pyrazol-1-ylphenyl)propanamide
—— 3-(5-aminopentyl)-1-(1H-indol-3-ylmethyl)-5-[(5-phenyl-1H-imidazol-2-yl)methyl]-2-sulfanylideneimidazolidin-4-one —— C27H30N6OS
3-(5-aminopentyl)-1-(1H-indol-3-ylmethyl)-5-[(5-phenyl-1H-imidazol-2-yl)methyl]-2-sulfanylideneimidazolidin-4-one
—— 2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-pyrazol-1-ylphenyl)acetamide —— C19H20N4O3
2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-pyrazol-1-ylphenyl)acetamide
—— (2S,5S)-2,5-dimethyl-4-[[3-(3-nitrophenyl)-1,2,4-triazol-1-yl]methyl]morpholine —— C15H19N5O3
(2S,5S)-2,5-dimethyl-4-[[3-(3-nitrophenyl)-1,2,4-triazol-1-yl]methyl]morpholine
—— 2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-pyrazol-1-ylphenyl)acetamide —— C19H20N4O3
2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-pyrazol-1-ylphenyl)acetamide
—— (3S)-1-(3-bromophenyl)-5-oxo-N-(2-pyrazol-1-ylphenyl)pyrrolidine-3-carboxamide —— C20H17BrN4O2
(3S)-1-(3-bromophenyl)-5-oxo-N-(2-pyrazol-1-ylphenyl)pyrrolidine-3-carboxamide
—— N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide —— C24H30N4O4
N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
—— (3R)-1-(3-bromophenyl)-5-oxo-N-(2-pyrazol-1-ylphenyl)pyrrolidine-3-carboxamide —— C20H17BrN4O2
(3R)-1-(3-bromophenyl)-5-oxo-N-(2-pyrazol-1-ylphenyl)pyrrolidine-3-carboxamide
—— N-[[1-(2,4-dichlorophenyl)-7-fluoro-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]piperidin-1-amine —— C22H21Cl2FN4S
N-[[1-(2,4-dichlorophenyl)-7-fluoro-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]piperidin-1-amine