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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-N-methyl-1-(2-phenylacetyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-3-carboxamide —— C25H29N5O2
(3S)-N-methyl-1-(2-phenylacetyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-3-carboxamide
—— N-[(R)-furan-2-yl(phenyl)methyl]-5-methyl-1-(2-methylphenyl)pyrazole-4-carboxamide —— C23H21N3O2
N-[(R)-furan-2-yl(phenyl)methyl]-5-methyl-1-(2-methylphenyl)pyrazole-4-carboxamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N',N',5-trimethyl-1-(2-methylphenyl)pyrazole-4-carbohydrazide —— C18H24N4O3S
N-[(3S)-1,1-dioxothiolan-3-yl]-N',N',5-trimethyl-1-(2-methylphenyl)pyrazole-4-carbohydrazide
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2R)-4-(furan-2-yl)butan-2-yl]benzamide —— C20H22BrN3O2
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2R)-4-(furan-2-yl)butan-2-yl]benzamide
—— [(1S)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl] 5-methyl-1-(2-methylphenyl)pyrazole-4-carboxylate —— C22H20F2N4O2
[(1S)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl] 5-methyl-1-(2-methylphenyl)pyrazole-4-carboxylate
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N',N',5-trimethyl-1-(2-methylphenyl)pyrazole-4-carbohydrazide —— C18H24N4O3S
N-[(3R)-1,1-dioxothiolan-3-yl]-N',N',5-trimethyl-1-(2-methylphenyl)pyrazole-4-carbohydrazide
—— 2-[(3aS)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)acetamide —— C28H25N5O3
2-[(3aS)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)acetamide
—— 5-[(E)-(2,6-dichlorophenyl)methylideneamino]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C18H11Cl2N5O
5-[(E)-(2,6-dichlorophenyl)methylideneamino]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— ethyl 5-methyl-2-[3-[(2S)-oxolan-2-yl]propanoyl-(2-phenylethyl)amino]-1,3-thiazole-4-carboxylate —— C22H28N2O4S
ethyl 5-methyl-2-[3-[(2S)-oxolan-2-yl]propanoyl-(2-phenylethyl)amino]-1,3-thiazole-4-carboxylate
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2S)-4-(furan-2-yl)butan-2-yl]benzamide —— C20H22BrN3O2
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2S)-4-(furan-2-yl)butan-2-yl]benzamide
—— (3S)-N-methyl-1-(2-phenylacetyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-3-carboxamide —— C25H29N5O2
(3S)-N-methyl-1-(2-phenylacetyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-3-carboxamide
—— (3S)-N-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazol-5-yl]-1-(2-phenylacetyl)piperidine-3-carboxamide —— C25H23FN4O2S
(3S)-N-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazol-5-yl]-1-(2-phenylacetyl)piperidine-3-carboxamide
—— (3R)-N-methyl-1-(2-phenylacetyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-3-carboxamide —— C25H29N5O2
(3R)-N-methyl-1-(2-phenylacetyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]piperidine-3-carboxamide
—— [(2S)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]methanone —— C24H27N3O3
[(2S)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]methanone
—— N-[(1R)-1-(2,5-dimethoxyphenyl)ethyl]-1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carboxamide —— C24H29N3O3
N-[(1R)-1-(2,5-dimethoxyphenyl)ethyl]-1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carboxamide
—— ethyl 5-methyl-2-[3-[(2R)-oxolan-2-yl]propanoyl-(2-phenylethyl)amino]-1,3-thiazole-4-carboxylate —— C22H28N2O4S
ethyl 5-methyl-2-[3-[(2R)-oxolan-2-yl]propanoyl-(2-phenylethyl)amino]-1,3-thiazole-4-carboxylate
—— (3R)-N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-methyl-5-oxo-1-propan-2-ylpyrrolidine-3-carboxamide —— C25H28N4O2
(3R)-N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-methyl-5-oxo-1-propan-2-ylpyrrolidine-3-carboxamide
—— 3,5-dichloro-N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]pyridin-2-amine —— C17H15Cl2N5
3,5-dichloro-N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]pyridin-2-amine
—— [(2R)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]methanone —— C24H27N3O3
[(2R)-2-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]methanone
—— 1,3-Dihydroisoindol-2-yl-[1-(3-fluorophenyl)pyrazol-3-yl]methanone —— C18H14FN3O
1,3-Dihydroisoindol-2-yl-[1-(3-fluorophenyl)pyrazol-3-yl]methanone
—— N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C23H25F3N4O2
N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— 5-cyclopropyl-N-[(2R)-2-phenylpropyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C23H22F3N3O
5-cyclopropyl-N-[(2R)-2-phenylpropyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 5-[(E)-(3-nitrophenyl)methylideneamino]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C18H12N6O3
5-[(E)-(3-nitrophenyl)methylideneamino]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— 2-(5-phenyltetrazol-2-yl)-N-[(E)-1-(3,4,5-trimethoxyphenyl)ethylideneamino]acetamide —— C20H22N6O4
2-(5-phenyltetrazol-2-yl)-N-[(E)-1-(3,4,5-trimethoxyphenyl)ethylideneamino]acetamide
—— 5-cyclopropyl-N-[(2S)-2-phenylpropyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C23H22F3N3O
5-cyclopropyl-N-[(2S)-2-phenylpropyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 4-[(3aR)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)butanamide —— C29H27N5O3
4-[(3aR)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)butanamide
—— (3S)-N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-methyl-5-oxo-1-propan-2-ylpyrrolidine-3-carboxamide —— C25H28N4O2
(3S)-N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-methyl-5-oxo-1-propan-2-ylpyrrolidine-3-carboxamide
—— N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C23H25F3N4O2
N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— [(1R)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl] 5-methyl-1-(2-methylphenyl)pyrazole-4-carboxylate —— C22H20F2N4O2
[(1R)-1-[1-(difluoromethyl)benzimidazol-2-yl]ethyl] 5-methyl-1-(2-methylphenyl)pyrazole-4-carboxylate
—— 5-cyclopropyl-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C24H25F3N4OS
5-cyclopropyl-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]benzamide —— C22H22BrN3O3
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]benzamide
—— 4-[(3aS)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)butanamide —— C29H27N5O3
4-[(3aS)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)butanamide
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]benzamide —— C22H22BrN3O3
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]benzamide
—— (3S)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-5-oxo-1-(2,2,2-trifluoroethyl)pyrrolidine-3-carboxamide —— C17H15F4N3O2S
(3S)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-5-oxo-1-(2,2,2-trifluoroethyl)pyrrolidine-3-carboxamide
—— N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C23H25F3N4O2
N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— N-[(2S)-2-(4-methoxyphenyl)-2-morpholin-4-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C25H27F3N4O3
N-[(2S)-2-(4-methoxyphenyl)-2-morpholin-4-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— 5-cyclopropyl-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C25H27F3N4O2
5-cyclopropyl-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 2-(4-ethoxyphenyl)-N-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C23H27N3O3S
2-(4-ethoxyphenyl)-N-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— N-[(1S)-1-(2-chlorophenyl)ethyl]-5-methyl-1-(2-methylphenyl)pyrazole-4-carboxamide —— C20H20ClN3O
N-[(1S)-1-(2-chlorophenyl)ethyl]-5-methyl-1-(2-methylphenyl)pyrazole-4-carboxamide
—— 5-cyclopropyl-1-(2,4-dichlorophenyl)-N-[(2R)-1-methoxypropan-2-yl]pyrazole-4-carboxamide —— C17H19Cl2N3O2
5-cyclopropyl-1-(2,4-dichlorophenyl)-N-[(2R)-1-methoxypropan-2-yl]pyrazole-4-carboxamide
—— 6-[(2Z)-2-[[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]pyridine-3-sulfonamide —— C23H18N6O3S
6-[(2Z)-2-[[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]pyridine-3-sulfonamide
—— 1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]pyrazole-4-carboxamide —— C25H29ClN4O2
1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(2S)-2-(furan-2-yl)-2-piperidin-1-ylethyl]pyrazole-4-carboxamide
—— 3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[3-[5-amino-4-cyano-1-(4-fluorophenyl)pyrazol-3-yl]propyl]propanamide —— C24H27FN6O3
3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[3-[5-amino-4-cyano-1-(4-fluorophenyl)pyrazol-3-yl]propyl]propanamide
—— 5-cyclopropyl-N-[(2R)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C27H29F3N4O2
5-cyclopropyl-N-[(2R)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 5-cyclopropyl-N-[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C27H29F3N4O2
5-cyclopropyl-N-[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— N-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C23H25F3N4O2
N-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— N'-[(2R)-2-(4-ethoxyphenoxy)propanoyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carbohydrazide —— C23H23F3N4O4
N'-[(2R)-2-(4-ethoxyphenoxy)propanoyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carbohydrazide
—— [4-[5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazole-4-carbonyl]piperazin-1-yl]-[(2R)-oxolan-2-yl]methanone —— C22H24Cl2N4O3
[4-[5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazole-4-carbonyl]piperazin-1-yl]-[(2R)-oxolan-2-yl]methanone
—— 5-cyclopropyl-N-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C25H27F3N4O2
5-cyclopropyl-N-[(2R)-2-(furan-2-yl)-2-piperidin-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— [(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]methanone —— C23H22N4OS
[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]methanone