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中文名称 英文名称 CAS号 化学式 结构式图片
—— (Z)-2-cyano-N-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-3-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]prop-2-enamide —— C20H23N5O2S
(Z)-2-cyano-N-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-3-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]prop-2-enamide
—— 1-(4-fluorophenyl)-N-[(2S)-2-(1H-indol-3-yl)-2-(4-methoxyphenyl)ethyl]-5-methyltriazole-4-carboxamide —— C27H24FN5O2
1-(4-fluorophenyl)-N-[(2S)-2-(1H-indol-3-yl)-2-(4-methoxyphenyl)ethyl]-5-methyltriazole-4-carboxamide
—— N-[(1S)-1-(2-chlorophenyl)-2-oxocyclohexyl]-N-methyl-2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)acetamide —— C23H23ClN2O3S
N-[(1S)-1-(2-chlorophenyl)-2-oxocyclohexyl]-N-methyl-2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)acetamide
—— 1-(4-fluorophenyl)-5-methyl-N-[(1S)-1-naphthalen-2-ylethyl]triazole-4-carboxamide —— C22H19FN4O
1-(4-fluorophenyl)-5-methyl-N-[(1S)-1-naphthalen-2-ylethyl]triazole-4-carboxamide
—— N-[2-[(5Z)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide —— C22H18FN5O3S
N-[2-[(5Z)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide
—— 1-(4-fluorophenyl)-5-methyl-N-[(1R)-1-naphthalen-2-ylethyl]triazole-4-carboxamide —— C22H19FN4O
1-(4-fluorophenyl)-5-methyl-N-[(1R)-1-naphthalen-2-ylethyl]triazole-4-carboxamide
—— N-[(1R)-1-(2-chlorophenyl)-2-oxocyclohexyl]-N-methyl-2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)acetamide —— C23H23ClN2O3S
N-[(1R)-1-(2-chlorophenyl)-2-oxocyclohexyl]-N-methyl-2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)acetamide
—— N-[(1S)-1-(2-chlorophenyl)-2-oxocyclohexyl]-1-(4-fluorophenyl)-N,5-dimethyl-1,2,4-triazole-3-carboxamide —— C23H22ClFN4O2
N-[(1S)-1-(2-chlorophenyl)-2-oxocyclohexyl]-1-(4-fluorophenyl)-N,5-dimethyl-1,2,4-triazole-3-carboxamide
—— 1-(4-fluorophenyl)-N-[(2R)-2-(1H-indol-3-yl)-2-(4-methoxyphenyl)ethyl]-5-methyltriazole-4-carboxamide —— C27H24FN5O2
1-(4-fluorophenyl)-N-[(2R)-2-(1H-indol-3-yl)-2-(4-methoxyphenyl)ethyl]-5-methyltriazole-4-carboxamide
—— N-[(2R)-2-(2-chlorophenyl)-2-(diethylamino)ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide —— C22H25ClFN5O
N-[(2R)-2-(2-chlorophenyl)-2-(diethylamino)ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide
—— (1-phenyltetrazol-5-yl)methyl 2-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]acetate —— C17H20N4O2
(1-phenyltetrazol-5-yl)methyl 2-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]acetate
—— 1-(4-fluorophenyl)-5-methyl-N'-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]triazole-4-carbohydrazide —— C20H20FN5O2S
1-(4-fluorophenyl)-5-methyl-N'-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]triazole-4-carbohydrazide
—— 1-[(1S)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]-3-[(1-phenylpyrazol-4-yl)methyl]urea —— C23H24N4O3
1-[(1S)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]-3-[(1-phenylpyrazol-4-yl)methyl]urea
—— 2-[(2S)-2-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-3-methyl-4-oxo-2H-quinazolin-1-yl]-N-methylacetamide —— C22H21ClFN5O2
2-[(2S)-2-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-3-methyl-4-oxo-2H-quinazolin-1-yl]-N-methylacetamide
—— N-[2-[(5E)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide —— C22H18FN5O3S
N-[2-[(5E)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide
—— ethyl 2-[[(2R)-2-(2-cyanophenoxy)propanoyl]amino]-4-phenyl-1,3-thiazole-5-carboxylate —— C22H19N3O4S
ethyl 2-[[(2R)-2-(2-cyanophenoxy)propanoyl]amino]-4-phenyl-1,3-thiazole-5-carboxylate
—— 1-(4-fluorophenyl)-5-methyl-N'-[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]triazole-4-carbohydrazide —— C20H20FN5O2S
1-(4-fluorophenyl)-5-methyl-N'-[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]triazole-4-carbohydrazide
—— 2-[(2R)-2-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-3-methyl-4-oxo-2H-quinazolin-1-yl]-N-methylacetamide —— C22H21ClFN5O2
2-[(2R)-2-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-3-methyl-4-oxo-2H-quinazolin-1-yl]-N-methylacetamide
—— (1-phenyltetrazol-5-yl)methyl 2-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetate —— C17H20N4O2
(1-phenyltetrazol-5-yl)methyl 2-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetate
—— 3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-imidazol-1-ylphenyl)propanamide —— C20H22N4O3
3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-imidazol-1-ylphenyl)propanamide
—— (1-phenyltetrazol-5-yl)methyl 2-[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetate —— C17H20N4O2
(1-phenyltetrazol-5-yl)methyl 2-[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetate
—— N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-2-methylaniline —— C19H20N4
N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-2-methylaniline
—— 3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-imidazol-1-ylphenyl)propanamide —— C20H22N4O3
3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-(2-imidazol-1-ylphenyl)propanamide
—— N-[(1R)-1-(2-chlorophenyl)-2-oxocyclohexyl]-1-(4-fluorophenyl)-N,5-dimethyl-1,2,4-triazole-3-carboxamide —— C23H22ClFN4O2
N-[(1R)-1-(2-chlorophenyl)-2-oxocyclohexyl]-1-(4-fluorophenyl)-N,5-dimethyl-1,2,4-triazole-3-carboxamide
—— 1-[(1R)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]-3-[(1-phenylpyrazol-4-yl)methyl]urea —— C23H24N4O3
1-[(1R)-1-(7-ethoxy-1-benzofuran-2-yl)ethyl]-3-[(1-phenylpyrazol-4-yl)methyl]urea
—— 1-(4-fluorophenyl)-5-methyl-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide —— C20H20FN7OS
1-(4-fluorophenyl)-5-methyl-N-[(1R)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide
—— N-[(2S)-2-[4-(dimethylamino)phenyl]-2-(1H-indol-3-yl)ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide —— C28H27FN6O
N-[(2S)-2-[4-(dimethylamino)phenyl]-2-(1H-indol-3-yl)ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide
—— 1-(4-fluorophenyl)-N-[(2S)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-5-methyltriazole-4-carboxamide —— C23H26FN5O2
1-(4-fluorophenyl)-N-[(2S)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-5-methyltriazole-4-carboxamide
—— 1-(4-fluorophenyl)-5-methyl-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide —— C20H20FN7OS
1-(4-fluorophenyl)-5-methyl-N-[(1S)-3-methylsulfanyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide
—— 1-(4-fluorophenyl)-N-[(2R)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-5-methyltriazole-4-carboxamide —— C23H26FN5O2
1-(4-fluorophenyl)-N-[(2R)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-5-methyltriazole-4-carboxamide
—— 3-[(3aS)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)propanamide —— C28H25N5O3
3-[(3aS)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)propanamide
—— 3-[(3aR)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)propanamide —— C28H25N5O3
3-[(3aR)-3a-methyl-1,5-dioxo-2,3-dihydropyrrolo[1,2-a]quinazolin-4-yl]-N-(2-phenylimidazo[1,2-a]pyridin-3-yl)propanamide
—— (2R)-N-[4-[5-(acetamidomethyl)thiophen-2-yl]-5-methyl-1,3-thiazol-2-yl]-2-(2-cyanophenoxy)propanamide —— C21H20N4O3S2
(2R)-N-[4-[5-(acetamidomethyl)thiophen-2-yl]-5-methyl-1,3-thiazol-2-yl]-2-(2-cyanophenoxy)propanamide
—— (Z)-1,1,1-trifluoro-4-[(5-methyl-2-phenylpyrazol-3-yl)amino]but-3-en-2-one —— C14H12F3N3O
(Z)-1,1,1-trifluoro-4-[(5-methyl-2-phenylpyrazol-3-yl)amino]but-3-en-2-one
—— N-[(2S)-2-(2-chlorophenyl)-2-(diethylamino)ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide —— C22H25ClFN5O
N-[(2S)-2-(2-chlorophenyl)-2-(diethylamino)ethyl]-1-(4-fluorophenyl)-5-methyltriazole-4-carboxamide
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(4-fluorophenoxy)ethyl]butanamide —— C19H19ClFN5O2
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(4-fluorophenoxy)ethyl]butanamide
—— 1-(3-chlorophenyl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-5-ethylpyrazole-4-carboxamide —— C22H24ClN3O3
1-(3-chlorophenyl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-5-ethylpyrazole-4-carboxamide
—— 1-(4-fluorophenyl)-N-[4-[[(3S)-3-methylpiperidin-1-yl]methyl]-1,3-thiazol-2-yl]-5-propan-2-ylpyrazole-4-carboxamide —— C23H28FN5OS
1-(4-fluorophenyl)-N-[4-[[(3S)-3-methylpiperidin-1-yl]methyl]-1,3-thiazol-2-yl]-5-propan-2-ylpyrazole-4-carboxamide
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(ethoxymethyl)phenyl]methyl]butanamide —— C21H24ClN5O2
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[[4-(ethoxymethyl)phenyl]methyl]butanamide
—— N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-1-(3-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C23H21FN4O3S
N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-1-(3-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(4-fluorophenoxy)ethyl]butanamide —— C19H19ClFN5O2
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[2-(4-fluorophenoxy)ethyl]butanamide
—— N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]-2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-2-oxoacetamide —— C24H24F3N3O4
N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]-2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-2-oxoacetamide
—— N-[(2R)-2-anilino-3-methylbutyl]-1-(4-fluorophenyl)-5-propan-2-ylpyrazole-4-carboxamide —— C24H29FN4O
N-[(2R)-2-anilino-3-methylbutyl]-1-(4-fluorophenyl)-5-propan-2-ylpyrazole-4-carboxamide
—— [(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[5-ethyl-1-(4-fluorophenyl)pyrazol-4-yl]methanone —— C21H26FN3O
[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-[5-ethyl-1-(4-fluorophenyl)pyrazol-4-yl]methanone
—— (E)-1-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine —— C13H10ClFN6
(E)-1-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine
—— 1-(3-chlorophenyl)-N-[(1S)-2,3-dihydro-1H-inden-1-yl]-5-methylpyrazole-4-carboxamide —— C20H18ClN3O
1-(3-chlorophenyl)-N-[(1S)-2,3-dihydro-1H-inden-1-yl]-5-methylpyrazole-4-carboxamide
—— 1-(4-fluorophenyl)-N-[4-[[(3R)-3-methylpiperidin-1-yl]methyl]-1,3-thiazol-2-yl]-5-propan-2-ylpyrazole-4-carboxamide —— C23H28FN5OS
1-(4-fluorophenyl)-N-[4-[[(3R)-3-methylpiperidin-1-yl]methyl]-1,3-thiazol-2-yl]-5-propan-2-ylpyrazole-4-carboxamide
—— N-[4-[4-[(1S)-1-acetamidoethyl]phenyl]-1,3-thiazol-2-yl]-1-(3-chlorophenyl)-5-methylpyrazole-4-carboxamide —— C24H22ClN5O2S
N-[4-[4-[(1S)-1-acetamidoethyl]phenyl]-1,3-thiazol-2-yl]-1-(3-chlorophenyl)-5-methylpyrazole-4-carboxamide
—— 1-(3-chlorophenyl)-N-[(1R)-2,3-dihydro-1H-inden-1-yl]-5-methylpyrazole-4-carboxamide —— C20H18ClN3O
1-(3-chlorophenyl)-N-[(1R)-2,3-dihydro-1H-inden-1-yl]-5-methylpyrazole-4-carboxamide
—— [(2R)-2-(1H-benzimidazol-2-yl)pyrrolidin-1-yl]-[1-(3-chlorophenyl)-5-methylpyrazol-4-yl]methanone —— C22H20ClN5O
[(2R)-2-(1H-benzimidazol-2-yl)pyrrolidin-1-yl]-[1-(3-chlorophenyl)-5-methylpyrazol-4-yl]methanone