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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]butanamide —— C17H22ClN5O2
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]butanamide
—— N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide —— C23H24ClN3O2S
N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
—— N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C21H22ClN3O2S2
N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— 5-[(E)-[(3-chloro-4-methylphenyl)hydrazinylidene]methyl]-1,4-dimethyl-2-phenylpyrazol-3-one —— C19H19ClN4O
5-[(E)-[(3-chloro-4-methylphenyl)hydrazinylidene]methyl]-1,4-dimethyl-2-phenylpyrazol-3-one
—— N-[(E)-[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]methylideneamino]acetamide —— C18H15BrN4O
N-[(E)-[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]methylideneamino]acetamide
—— (2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]butanamide —— C17H22ClN5O2
(2S)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]butanamide
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]butanamide —— C17H22ClN5O2
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]butanamide
—— 5-cyclopropyl-1-(2,4-dichlorophenyl)-N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide —— C23H23Cl2N3O3
5-cyclopropyl-1-(2,4-dichlorophenyl)-N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide
—— 2-[(E)-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methylideneamino]guanidine —— C11H10ClN5S
2-[(E)-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methylideneamino]guanidine
—— 2-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]acetamide —— C18H18ClN5O3
2-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]acetamide
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]benzamide —— C20H23BrN4OS
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]benzamide
—— (3S)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide —— C26H29FN4O2
(3S)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide
—— (E)-1-[5-chloro-1-(2,5-dimethylphenyl)-3-methylpyrazol-4-yl]-N-(4-methylpiperazin-1-yl)methanimine —— C18H24ClN5
(E)-1-[5-chloro-1-(2,5-dimethylphenyl)-3-methylpyrazol-4-yl]-N-(4-methylpiperazin-1-yl)methanimine
—— 2-(4-ethoxyphenyl)-4-methyl-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide —— C19H24N2O3S
2-(4-ethoxyphenyl)-4-methyl-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide
—— (3S)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide —— C26H29FN4O2
(3S)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide
—— (3R)-1-(2-fluoro-4-methylphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-oxopyrrolidine-3-carboxamide —— C24H24F2N4O2
(3R)-1-(2-fluoro-4-methylphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-oxopyrrolidine-3-carboxamide
—— 5-cyclopropyl-1-(2,4-dichlorophenyl)-N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide —— C23H23Cl2N3O3
5-cyclopropyl-1-(2,4-dichlorophenyl)-N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide
—— N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]acetamide —— C21H21ClN2O2S
N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]acetamide
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]benzamide —— C20H23BrN4OS
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]benzamide
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-N-methylbenzamide —— C22H24BrN3O2
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-N-methylbenzamide
—— (2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]butanamide —— C17H22ClN5O2
(2R)-2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]butanamide
—— 1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide —— C24H26ClN3O3
1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide
—— 2-(4-ethoxyphenyl)-4-methyl-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide —— C19H24N2O3S
2-(4-ethoxyphenyl)-4-methyl-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide
—— (3R)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide —— C26H29FN4O2
(3R)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide
—— (3R)-5-oxo-N-[2-(1,2,4-triazol-1-yl)phenyl]-1-(2,2,2-trifluoroethyl)pyrrolidine-3-carboxamide —— C15H14F3N5O2
(3R)-5-oxo-N-[2-(1,2,4-triazol-1-yl)phenyl]-1-(2,2,2-trifluoroethyl)pyrrolidine-3-carboxamide
—— N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]acetamide —— C21H21ClN2O2S
N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]acetamide
—— 2-[(3aR,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]acetamide —— C18H18ClN5O3
2-[(3aR,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-N-[3-chloro-2-(1,2,4-triazol-1-yl)phenyl]acetamide
—— (E)-1-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]-N-(4-methylpiperazin-1-yl)methanimine —— C16H19Cl2N5
(E)-1-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]-N-(4-methylpiperazin-1-yl)methanimine
—— N-[(1R)-1-(7-methoxy-1-benzofuran-2-yl)ethyl]-2-(5-phenyltetrazol-2-yl)acetamide —— C20H19N5O3
N-[(1R)-1-(7-methoxy-1-benzofuran-2-yl)ethyl]-2-(5-phenyltetrazol-2-yl)acetamide
—— N-[(1S)-1-(3-acetamidophenyl)ethyl]-5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C24H23F3N4O2
N-[(1S)-1-(3-acetamidophenyl)ethyl]-5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 1-[4-[(1R)-1-(2-chlorophenyl)ethyl]piperazin-1-yl]-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]ethanone —— C22H24ClN3O2S
1-[4-[(1R)-1-(2-chlorophenyl)ethyl]piperazin-1-yl]-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]ethanone
—— N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C20H21F3N4OS
N-[(2S)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— (3S)-1-(2-fluoro-4-methylphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-oxopyrrolidine-3-carboxamide —— C24H24F2N4O2
(3S)-1-(2-fluoro-4-methylphenyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-5-oxopyrrolidine-3-carboxamide
—— (3R)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide —— C26H29FN4O2
(3R)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-1-(2-phenylacetyl)piperidine-3-carboxamide
—— 2-(4-ethoxyphenyl)-4-methyl-N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide —— C19H24N2O3S
2-(4-ethoxyphenyl)-4-methyl-N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide
—— 2-[2-[(2S)-butan-2-yl]phenoxy]-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]acetamide —— C20H23N5O2S
2-[2-[(2S)-butan-2-yl]phenoxy]-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]acetamide
—— 2-(4-ethoxyphenyl)-4-methyl-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide —— C19H24N2O3S
2-(4-ethoxyphenyl)-4-methyl-N-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]-1,3-thiazole-5-carboxamide
—— 4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1R,2S)-2-(trifluoromethyl)cyclohexyl]benzamide —— C19H21BrF3N3O
4-(4-bromo-3,5-dimethylpyrazol-1-yl)-N-[(1R,2S)-2-(trifluoromethyl)cyclohexyl]benzamide
—— 1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide —— C24H26ClN3O3
1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]pyrazole-4-carboxamide
—— (2R)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]propanamide —— C19H19FN6O2S2
(2R)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]propanamide
—— N-[(1S)-1-(7-methoxy-1-benzofuran-2-yl)ethyl]-2-(5-phenyltetrazol-2-yl)acetamide —— C20H19N5O3
N-[(1S)-1-(7-methoxy-1-benzofuran-2-yl)ethyl]-2-(5-phenyltetrazol-2-yl)acetamide
—— N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C20H21F3N4OS
N-[(2R)-2-(dimethylamino)-2-thiophen-3-ylethyl]-1-(2-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— 2-[2-[(2R)-butan-2-yl]phenoxy]-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]acetamide —— C20H23N5O2S
2-[2-[(2R)-butan-2-yl]phenoxy]-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]acetamide
—— 1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(2S)-4-methyl-2-morpholin-4-ylpentyl]pyrazole-4-carboxamide —— C24H33ClN4O2
1-(3-chloro-4-methylphenyl)-5-cyclopropyl-N-[(2S)-4-methyl-2-morpholin-4-ylpentyl]pyrazole-4-carboxamide
—— N-[(1R)-1-(1,3-benzodioxol-5-yl)ethyl]-5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C23H20F3N3O3
N-[(1R)-1-(1,3-benzodioxol-5-yl)ethyl]-5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 2-(4-ethoxyphenyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide —— C23H26N2O3S
2-(4-ethoxyphenyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide
—— N-[(1R)-1-(3-acetamidophenyl)ethyl]-5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C24H23F3N4O2
N-[(1R)-1-(3-acetamidophenyl)ethyl]-5-cyclopropyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— 1-[4-[(1S)-1-(2-chlorophenyl)ethyl]piperazin-1-yl]-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]ethanone —— C22H24ClN3O2S
1-[4-[(1S)-1-(2-chlorophenyl)ethyl]piperazin-1-yl]-2-[2-(5-methylfuran-2-yl)-1,3-thiazol-4-yl]ethanone
—— (2S)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]propanamide —— C19H19FN6O2S2
(2S)-2-[2-(4-fluoroanilino)-2-oxoethyl]sulfanyl-N-[3-(5-methylsulfanyltetrazol-1-yl)phenyl]propanamide
—— N-[(2R)-4-methyl-2-morpholin-4-ylpentyl]-1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carboxamide —— C24H36N4O2
N-[(2R)-4-methyl-2-morpholin-4-ylpentyl]-1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carboxamide