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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[2-(4-fluorophenyl)pyrazolo[1,5-a]pyridin-3-yl]-2-pyrimidinamine —— C17H12FN5
4-[2-(4-fluorophenyl)pyrazolo[1,5-a]pyridin-3-yl]-2-pyrimidinamine
—— 3-(6-Aminopyridin-3-yl)-2-(1-hexylimidazol-4-yl)propanoic acid —— C17H24N4O2
3-(6-Aminopyridin-3-yl)-2-(1-hexylimidazol-4-yl)propanoic acid
—— N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C24H31N5O2S
N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— N-[(3R,4S)-1-azabicyclo[2.2.1]heptan-3-yl]-5-phenyl-1,3-oxazole-2-carboxamide —— C16H17N3O2
N-[(3R,4S)-1-azabicyclo[2.2.1]heptan-3-yl]-5-phenyl-1,3-oxazole-2-carboxamide
—— [(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl] (3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carboxylate —— C19H20F3N3O4
[(1R)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl] (3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carboxylate
—— N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C24H31N5O2S
N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-2-[[4-(4-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(1R)-1-naphthalen-2-ylethyl]pyrazole-4-carboxamide —— C24H21F2N3O
1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(1R)-1-naphthalen-2-ylethyl]pyrazole-4-carboxamide
—— 2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]acetamide —— C24H28ClN5O2S
2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]acetamide
—— 3-(4-aminophenyl)-4-(4-fluorophenyl)-1H-1,2,4-triazole-5-thione —— C14H11FN4S
3-(4-aminophenyl)-4-(4-fluorophenyl)-1H-1,2,4-triazole-5-thione
—— 2-(3,4-dimethyl-phenyl)-imidazo[1,2-a]pyridine hydrochloride —— C15H14N2*ClH
2-(3,4-dimethyl-phenyl)-imidazo[1,2-a]pyridine hydrochloride
—— 1-(2,4-difluorophenyl)-N-[(2R)-2-(4-methoxyphenyl)-2-piperidin-1-ylethyl]-3,5-dimethylpyrazole-4-carboxamide —— C26H30F2N4O2
1-(2,4-difluorophenyl)-N-[(2R)-2-(4-methoxyphenyl)-2-piperidin-1-ylethyl]-3,5-dimethylpyrazole-4-carboxamide
—— N-[(1R)-1-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide —— C20H18ClF2N3O
N-[(1R)-1-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide
—— [(1S)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl] (3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carboxylate —— C19H20F3N3O4
[(1S)-1-[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]ethyl] (3R)-5-oxo-1-propan-2-ylpyrrolidine-3-carboxylate
—— (2R)-N-[(1S)-1-(2,4-dichlorophenyl)ethyl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide —— C19H25Cl2N3O2S
(2R)-N-[(1S)-1-(2,4-dichlorophenyl)ethyl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide
—— 1-(2,4-difluorophenyl)-N'-[(2R)-2-(2-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide —— C21H19F3N4O3
1-(2,4-difluorophenyl)-N'-[(2R)-2-(2-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(3-propan-2-ylphenoxy)acetamide —— C23H26FN3O2
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(3-propan-2-ylphenoxy)acetamide
—— N-[[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide —— C27H34N4O2
N-[[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(3-propan-2-ylphenoxy)acetamide —— C23H26FN3O2
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(3-propan-2-ylphenoxy)acetamide
—— 2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanyl-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]acetamide —— C22H33N3O2S
2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanyl-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]acetamide
—— 1-[(1S,2S)-2-methylcyclohexyl]-3-[(1R)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]urea —— C13H23N5O
1-[(1S,2S)-2-methylcyclohexyl]-3-[(1R)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]urea
—— (2R)-N-benzyl-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanyl-N-methylpropanamide —— C19H27N3O2S
(2R)-N-benzyl-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanyl-N-methylpropanamide
—— 1-(2,4-difluorophenyl)-N'-[(2R)-2-(4-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide —— C21H19F3N4O3
1-(2,4-difluorophenyl)-N'-[(2R)-2-(4-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide
—— N-[(1R)-1-(4-bromophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide —— C20H18BrF2N3O
N-[(1R)-1-(4-bromophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide
—— (2S)-N-[(1R)-1-(2,4-dichlorophenyl)ethyl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide —— C19H25Cl2N3O2S
(2S)-N-[(1R)-1-(2,4-dichlorophenyl)ethyl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide
—— (2S)-N-[(1S)-1-(2,4-dichlorophenyl)ethyl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide —— C19H25Cl2N3O2S
(2S)-N-[(1S)-1-(2,4-dichlorophenyl)ethyl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide
—— N-[(1S)-1-(4-bromophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide —— C20H18BrF2N3O
N-[(1S)-1-(4-bromophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide
—— (2R)-N-[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]-2-[(4,5-dimethyl-1,3-oxazol-2-yl)sulfanyl]propanamide —— C17H15F2N3O2S2
(2R)-N-[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]-2-[(4,5-dimethyl-1,3-oxazol-2-yl)sulfanyl]propanamide
—— [1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone —— C24H28F2N6O
[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone
—— (2R)-N-[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide —— C20H22F2N4O2S2
(2R)-N-[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]-2-[1-(2-methoxyethyl)-4,5-dimethylimidazol-2-yl]sulfanylpropanamide
—— 1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(1S)-1-naphthalen-2-ylethyl]pyrazole-4-carboxamide —— C24H21F2N3O
1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(1S)-1-naphthalen-2-ylethyl]pyrazole-4-carboxamide
—— 1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(2R)-6-methylheptan-2-yl]pyrazole-4-carboxamide —— C20H27F2N3O
1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(2R)-6-methylheptan-2-yl]pyrazole-4-carboxamide
—— (E)-N-[[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C28H34N4O2
(E)-N-[[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— 1-(2,4-difluorophenyl)-N-[(2S)-2-(4-methoxyphenyl)-2-piperidin-1-ylethyl]-3,5-dimethylpyrazole-4-carboxamide —— C26H30F2N4O2
1-(2,4-difluorophenyl)-N-[(2S)-2-(4-methoxyphenyl)-2-piperidin-1-ylethyl]-3,5-dimethylpyrazole-4-carboxamide
—— N-[(1S)-1-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide —— C20H18ClF2N3O
N-[(1S)-1-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide
—— 1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazole-4-carboxamide —— C22H21F2N3O
1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazole-4-carboxamide
—— N-[2-[(5E)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide —— C24H20F2N4O3S
N-[2-[(5E)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide
—— 1-(2,4-difluorophenyl)-N'-[(2R)-2-(4-ethoxyphenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide —— C23H24F2N4O4
1-(2,4-difluorophenyl)-N'-[(2R)-2-(4-ethoxyphenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide
—— 1-[(2R)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C16H28N4O2S
1-[(2R)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— N-[[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide —— C27H34N4O2
N-[[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetamide
—— [(3S)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methanone —— C24H23F2N5O
[(3S)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methanone
—— N-[2-[(5Z)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide —— C24H20F2N4O3S
N-[2-[(5Z)-5-benzylidene-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-1-(2,4-difluorophenyl)-3,5-dimethylpyrazole-4-carboxamide
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(1S)-1-[3-methoxy-4-(2-methylpropoxy)phenyl]ethyl]acetamide —— C26H33N3O3
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(1S)-1-[3-methoxy-4-(2-methylpropoxy)phenyl]ethyl]acetamide
—— (E)-N-[[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C28H34N4O2
(E)-N-[[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— 1-(2,4-difluorophenyl)-N'-[(2S)-2-(4-ethoxyphenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide —— C23H24F2N4O4
1-(2,4-difluorophenyl)-N'-[(2S)-2-(4-ethoxyphenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide
—— 1-(2,4-difluorophenyl)-N'-[(2S)-2-(2-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide —— C21H19F3N4O3
1-(2,4-difluorophenyl)-N'-[(2S)-2-(2-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide
—— 1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(2S)-6-methylheptan-2-yl]pyrazole-4-carboxamide —— C20H27F2N3O
1-(2,4-difluorophenyl)-3,5-dimethyl-N-[(2S)-6-methylheptan-2-yl]pyrazole-4-carboxamide
—— 2-[4-(2-Methylimidazol-1-yl)phenoxy]ethanamine —— C12H15N3O
2-[4-(2-Methylimidazol-1-yl)phenoxy]ethanamine
—— 3-(6-Amino-5-chloro-pyridin-3-yl)-2-(1H-imidazol-4-yl)-propionic acid —— C11H11ClN4O2
3-(6-Amino-5-chloro-pyridin-3-yl)-2-(1H-imidazol-4-yl)-propionic acid
—— 1-(2,4-difluorophenyl)-N'-[(2S)-2-(4-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide —— C21H19F3N4O3
1-(2,4-difluorophenyl)-N'-[(2S)-2-(4-fluorophenoxy)propanoyl]-3,5-dimethylpyrazole-4-carbohydrazide
—— [(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methanone —— C24H23F2N5O
[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methanone