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—— (6R)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one —— C20H30N4O
(6R)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H30N4O3
(6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[[3-[(3,5-dimethylpyrazol-1-yl)methyl]-4-methoxyphenyl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one —— C26H36N4O2
(6S)-6-[1-[[3-[(3,5-dimethylpyrazol-1-yl)methyl]-4-methoxyphenyl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-(2-methoxyethyl)-6-[1-[[2-(2-methylpropoxy)phenyl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C25H38N2O3
(6R)-1-(2-methoxyethyl)-6-[1-[[2-(2-methylpropoxy)phenyl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[[3-[(3,5-dimethylpyrazol-1-yl)methyl]-4-methoxyphenyl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one —— C26H36N4O2
(6R)-6-[1-[[3-[(3,5-dimethylpyrazol-1-yl)methyl]-4-methoxyphenyl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H34N2O2
(6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-(2-methoxyethyl)-6-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H31N3O2
(6R)-1-(2-methoxyethyl)-6-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one —— C20H30N4O
(6S)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-methyl-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(2-methylpyrazole-3-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H30N4O3
(6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(2-methylpyrazole-3-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H34N2O2
(6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(pyridine-2-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C25H29N3O3
(6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(pyridine-2-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-(5-methoxy-1-benzofuran-2-carbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C24H30N2O5
(6S)-6-[1-(5-methoxy-1-benzofuran-2-carbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-(1-benzylpiperidin-4-yl)-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H32N2O2
(6R)-6-(1-benzylpiperidin-4-yl)-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-(2-methoxyethyl)-6-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H31N3O2
(6S)-1-(2-methoxyethyl)-6-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[(4-fluorophenyl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H31FN2O2
(6S)-6-[1-[(4-fluorophenyl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H35N5O3
(6R)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C24H32N4O
(6S)-6-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[[2-(dimethylamino)quinolin-3-yl]methyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C26H36N4O2
(6S)-6-[1-[[2-(dimethylamino)quinolin-3-yl]methyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-(1-benzylpiperidin-4-yl)-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H32N2O2
(6S)-6-(1-benzylpiperidin-4-yl)-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H35N5O3
(6S)-1-(2-methoxyethyl)-6-[1-(2-piperidin-1-ylpyrimidine-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(pyridine-2-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C25H29N3O3
(6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(pyridine-2-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-(2-methoxyethyl)-6-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C22H32N2O2
(6R)-1-(2-methoxyethyl)-6-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-benzyl-6-[1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H34N2O3
(6S)-1-benzyl-6-[1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-[2-[2-(4-bromophenyl)-2-oxoethyl]-3-methyl-1H-1,2,4-triazol-5-ylidene]cyclohexa-2,4-dien-1-one —— C17H14BrN3O2
6-[2-[2-(4-bromophenyl)-2-oxoethyl]-3-methyl-1H-1,2,4-triazol-5-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-amine —— C14H25N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-amine
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine —— C16H29N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine —— C16H29N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-amine
—— 6-[3-methyl-2-(2-morpholin-4-yl-2-oxoethyl)-1H-1,2,4-triazol-5-ylidene]cyclohexa-2,4-dien-1-one —— C15H18N4O3
6-[3-methyl-2-(2-morpholin-4-yl-2-oxoethyl)-1H-1,2,4-triazol-5-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-amine —— C14H25N5
6-[(dimethylamino)methyl]-N-methyl-2-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-amine
—— 6-[5-[(E)-1-(4-methoxyphenyl)prop-1-en-2-yl]-2-(4-phenyl-1,3-thiazol-2-yl)-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C27H22N4O2S
6-[5-[(E)-1-(4-methoxyphenyl)prop-1-en-2-yl]-2-(4-phenyl-1,3-thiazol-2-yl)-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[5-methyl-2-(4-phenyl-1,3-thiazol-2-yl)-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C18H14N4OS
6-[5-methyl-2-(4-phenyl-1,3-thiazol-2-yl)-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H21N5O3
6-[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]quinoline —— C20H22N4
6-[[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]quinoline
—— 6-[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H21N5O3
6-[(3S)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]quinoline —— C20H22N4
6-[[(3R)-3-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]quinoline
—— [6-methyl-2-(1-methylpiperidin-4-yl)pyrimidin-4-yl]-[(3S)-3-methylpiperidin-1-yl]methanone —— C18H28N4O
[6-methyl-2-(1-methylpiperidin-4-yl)pyrimidin-4-yl]-[(3S)-3-methylpiperidin-1-yl]methanone
—— 6-methyl-2-(1-methylpiperidin-4-yl)-N-prop-2-enylpyrimidine-4-carboxamide —— C15H22N4O
6-methyl-2-(1-methylpiperidin-4-yl)-N-prop-2-enylpyrimidine-4-carboxamide
—— 6-[[(3R)-1-acetylpiperidin-3-yl]methyl]-N-ethylpyridazine-3-carboxamide —— C15H22N4O2
6-[[(3R)-1-acetylpiperidin-3-yl]methyl]-N-ethylpyridazine-3-carboxamide
—— 6-methyl-2-[(3R)-1-methylpiperidin-3-yl]-N-prop-2-enylpyrimidine-4-carboxamide —— C15H22N4O
6-methyl-2-[(3R)-1-methylpiperidin-3-yl]-N-prop-2-enylpyrimidine-4-carboxamide
—— [6-Methyl-2-(1-methylpiperidin-4-yl)pyrimidin-4-yl]-(4-propylpiperazin-1-yl)methanone —— C19H31N5O
[6-Methyl-2-(1-methylpiperidin-4-yl)pyrimidin-4-yl]-(4-propylpiperazin-1-yl)methanone
—— 6-methyl-2-[(3R)-1-methylpiperidin-3-yl]-N-(2-methylpropyl)pyrimidine-4-carboxamide —— C16H26N4O
6-methyl-2-[(3R)-1-methylpiperidin-3-yl]-N-(2-methylpropyl)pyrimidine-4-carboxamide
—— 6-methyl-2-[(3S)-1-methylpiperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidine-4-carboxamide —— C18H29N5O
6-methyl-2-[(3S)-1-methylpiperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidine-4-carboxamide
—— 6-[(2S)-2-(1H-pyrazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C13H14N4O2
6-[(2S)-2-(1H-pyrazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— [6-methyl-2-[(3R)-1-methylpiperidin-3-yl]pyrimidin-4-yl]-(4-methylpiperazin-1-yl)methanone —— C17H27N5O
[6-methyl-2-[(3R)-1-methylpiperidin-3-yl]pyrimidin-4-yl]-(4-methylpiperazin-1-yl)methanone
—— 6-methyl-2-[(3R)-1-methylpiperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidine-4-carboxamide —— C18H29N5O
6-methyl-2-[(3R)-1-methylpiperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidine-4-carboxamide
—— 6-[[(3-benzylsulfanyl-5-sulfanylidene-1H-1,2,4-triazol-4-yl)amino]methylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C17H16N4O2S2
6-[[(3-benzylsulfanyl-5-sulfanylidene-1H-1,2,4-triazol-4-yl)amino]methylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-methyl-2-(1-methylpiperidin-4-yl)-N-(2-methylpropyl)pyrimidine-4-carboxamide —— C16H26N4O
6-methyl-2-(1-methylpiperidin-4-yl)-N-(2-methylpropyl)pyrimidine-4-carboxamide
—— 6-[[(3-benzylsulfanyl-5-sulfanylidene-1H-1,2,4-triazol-4-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C16H14N4OS2
6-[[(3-benzylsulfanyl-5-sulfanylidene-1H-1,2,4-triazol-4-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]methyl]-N,N-dimethylpyridazin-3-amine —— C18H26N6O
6-[[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]methyl]-N,N-dimethylpyridazin-3-amine
—— 6-methyl-5-[[(3R)-3-(6-methylpyrazin-2-yl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C17H21N5S
6-methyl-5-[[(3R)-3-(6-methylpyrazin-2-yl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole