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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-6-[[2-(furan-2-yl)ethylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C14H19N5O2
(6R)-6-[[2-(furan-2-yl)ethylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[(2-propan-2-yloxypyridin-3-yl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H24N6O2
(6S)-6-[[(2-propan-2-yloxypyridin-3-yl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[1-(4-fluorophenyl)cyclopropyl]methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H22FN5O
(6R)-6-[[[1-(4-fluorophenyl)cyclopropyl]methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H22N6OS
(6S)-6-[[[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[(2-thiophen-2-ylethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C14H19N5OS
(6R)-6-[(2-thiophen-2-ylethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H22N6OS
(6S)-6-[[[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(2S)-1-(2-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6R)-6-[[[(2S)-1-(2-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H22N6OS
(6R)-6-[[[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[(2-propan-2-yloxypyridin-3-yl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H24N6O2
(6R)-6-[[(2-propan-2-yloxypyridin-3-yl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H22N6OS
(6R)-6-[[[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[(2-thiophen-2-ylethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C14H19N5OS
(6S)-6-[(2-thiophen-2-ylethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[3-(cyclohexylamino)-3-oxopropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H28N6O2
(6R)-6-[[[3-(cyclohexylamino)-3-oxopropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-Amino-5-[2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetyl]-3-methyl-1-propylpyrimidine-2,4-dione —— C18H21N5O3S2
6-Amino-5-[2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetyl]-3-methyl-1-propylpyrimidine-2,4-dione
—— (6S)-6-[[[3-(cyclohexylamino)-3-oxopropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H28N6O2
(6S)-6-[[[3-(cyclohexylamino)-3-oxopropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[1-(4-fluorophenyl)cyclopropyl]methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H22FN5O
(6S)-6-[[[1-(4-fluorophenyl)cyclopropyl]methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(2R)-1-(2-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6R)-6-[[[(2R)-1-(2-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[(2-quinolin-8-ylethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H22N6O
(6R)-6-[(2-quinolin-8-ylethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6-chloropyridin-3-yl)-[4-[(R)-(4-fluorophenyl)-hydroxymethyl]piperidin-1-yl]methanone —— C18H18ClFN2O2
(6-chloropyridin-3-yl)-[4-[(R)-(4-fluorophenyl)-hydroxymethyl]piperidin-1-yl]methanone
—— (6-chloropyridin-3-yl)-[4-[(S)-(4-fluorophenyl)-hydroxymethyl]piperidin-1-yl]methanone —— C18H18ClFN2O2
(6-chloropyridin-3-yl)-[4-[(S)-(4-fluorophenyl)-hydroxymethyl]piperidin-1-yl]methanone
—— 6-Bromo-3-[2-oxo-2-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]quinazolin-4-one —— C20H17BrN2O2
6-Bromo-3-[2-oxo-2-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]quinazolin-4-one
—— 6-Bromo-3-[2-(4-methoxyphenoxy)ethyl]quinazolin-4-one —— C17H15BrN2O3
6-Bromo-3-[2-(4-methoxyphenoxy)ethyl]quinazolin-4-one
—— 6-Bromo-3-[2-(4-ethoxyphenyl)-2-oxoethyl]quinazolin-4-one —— C18H15BrN2O3
6-Bromo-3-[2-(4-ethoxyphenyl)-2-oxoethyl]quinazolin-4-one
—— 6-bromo-3-[2-oxo-2-(1H-pyrrol-2-yl)ethyl]quinazolin-4-one —— C14H10BrN3O2
6-bromo-3-[2-oxo-2-(1H-pyrrol-2-yl)ethyl]quinazolin-4-one
—— 6-bromo-3-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one —— C17H20BrN3O2
6-bromo-3-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one
—— 6-Bromo-3-[2-(4-chlorophenoxy)ethyl]quinazolin-4-one —— C16H12BrClN2O2
6-Bromo-3-[2-(4-chlorophenoxy)ethyl]quinazolin-4-one
—— 6-bromo-3-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]quinazolin-4-one —— C19H16BrN3O2
6-bromo-3-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]quinazolin-4-one
—— 6-[(2S)-2-methylmorpholine-4-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one —— C16H19N3O3
6-[(2S)-2-methylmorpholine-4-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one
—— 6-chloro-N-[(2R)-6-methylheptan-2-yl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C16H23ClN2O4S
6-chloro-N-[(2R)-6-methylheptan-2-yl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 6-Bromo-3-[2-(4-ethoxyphenoxy)ethyl]quinazolin-4-one —— C18H17BrN2O3
6-Bromo-3-[2-(4-ethoxyphenoxy)ethyl]quinazolin-4-one
—— 6-Bromo-3-[(7-methyl-2-oxochromen-4-yl)methyl]quinazolin-4-one —— C19H13BrN2O3
6-Bromo-3-[(7-methyl-2-oxochromen-4-yl)methyl]quinazolin-4-one
—— 6-bromo-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one —— C16H18BrN3O2
6-bromo-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one
—— 6-bromo-3-[2-(1H-indol-3-yl)-2-oxoethyl]quinazolin-4-one —— C18H12BrN3O2
6-bromo-3-[2-(1H-indol-3-yl)-2-oxoethyl]quinazolin-4-one
—— 6-bromo-3-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one —— C17H20BrN3O2
6-bromo-3-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one
—— 6-Bromo-3-(2-oxo-2-piperidin-1-ylethyl)quinazolin-4-one —— C15H16BrN3O2
6-Bromo-3-(2-oxo-2-piperidin-1-ylethyl)quinazolin-4-one
—— 6-chloro-N-[(2S)-6-methylheptan-2-yl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C16H23ClN2O4S
6-chloro-N-[(2S)-6-methylheptan-2-yl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 6-[(2R)-2-methylmorpholine-4-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one —— C16H19N3O3
6-[(2R)-2-methylmorpholine-4-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one
—— 6-Bromo-3-[2-(4-methylphenoxy)ethyl]quinazolin-4-one —— C17H15BrN2O2
6-Bromo-3-[2-(4-methylphenoxy)ethyl]quinazolin-4-one
—— 6-Bromo-3-[2-(4-ethylphenyl)-2-oxoethyl]quinazolin-4-one —— C18H15BrN2O2
6-Bromo-3-[2-(4-ethylphenyl)-2-oxoethyl]quinazolin-4-one
—— 6-bromo-3-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one —— C17H20BrN3O2
6-bromo-3-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one
—— 6-Bromo-3-[2-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]-2-oxoethyl]quinazolin-4-one —— C19H20BrN3O3
6-Bromo-3-[2-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]-2-oxoethyl]quinazolin-4-one
—— 6-Bromo-3-[2-(4-fluorophenoxy)ethyl]quinazolin-4-one —— C16H12BrFN2O2
6-Bromo-3-[2-(4-fluorophenoxy)ethyl]quinazolin-4-one
—— 6-Bromo-3-[(3-chlorophenyl)methyl]quinazolin-4-one —— C15H10BrClN2O
6-Bromo-3-[(3-chlorophenyl)methyl]quinazolin-4-one
—— 6-bromo-3-[2-(2,3-dihydro-1H-inden-5-yl)-2-oxoethyl]quinazolin-4-one —— C19H15BrN2O2
6-bromo-3-[2-(2,3-dihydro-1H-inden-5-yl)-2-oxoethyl]quinazolin-4-one
—— 6-bromo-3-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one —— C17H20BrN3O2
6-bromo-3-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]quinazolin-4-one
—— 6-methyl-2-oxo-N-[(1R)-2-phenoxy-1-phenylethyl]-1H-pyridine-3-carboxamide —— C21H20N2O3
6-methyl-2-oxo-N-[(1R)-2-phenoxy-1-phenylethyl]-1H-pyridine-3-carboxamide
—— 6-[(4S)-4-methyl-2-oxo-3,4-dihydro-1H-1,5-benzodiazepine-5-carbonyl]pyridine-3-carbonitrile —— C17H14N4O2
6-[(4S)-4-methyl-2-oxo-3,4-dihydro-1H-1,5-benzodiazepine-5-carbonyl]pyridine-3-carbonitrile
—— 6-methyl-2-oxo-N-[(1S)-2-phenoxy-1-phenylethyl]-1H-pyridine-3-carboxamide —— C21H20N2O3
6-methyl-2-oxo-N-[(1S)-2-phenoxy-1-phenylethyl]-1H-pyridine-3-carboxamide
—— [6-[[(3R)-1-methylpiperidin-3-yl]methylsulfanyl]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C17H25N3OS
[6-[[(3R)-1-methylpiperidin-3-yl]methylsulfanyl]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— [6-[[(3S)-1-methylpiperidin-3-yl]methylsulfanyl]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C17H25N3OS
[6-[[(3S)-1-methylpiperidin-3-yl]methylsulfanyl]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— [(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-(5-nitro-1H-indazol-3-yl)methanone —— C24H24N4O5
[(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-(5-nitro-1H-indazol-3-yl)methanone