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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-2-ethyl-8-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6R)-2-ethyl-8-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-acetylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6S)-8-(5-acetylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-chloropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H27ClN4O
(6R)-8-(5-chloropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-amino-5-[2-(2,3-dihydro-1H-inden-5-ylsulfanyl)acetyl]-1-propylpyrimidine-2,4-dione —— C18H21N3O3S
6-amino-5-[2-(2,3-dihydro-1H-inden-5-ylsulfanyl)acetyl]-1-propylpyrimidine-2,4-dione
—— 6-(2-fluoro-4-methoxyphenyl)-2-[(3R)-3-(hydroxymethyl)piperidine-1-carbonyl]-7-methylimidazo[1,2-a]pyrazin-8-one —— C21H23FN4O4
6-(2-fluoro-4-methoxyphenyl)-2-[(3R)-3-(hydroxymethyl)piperidine-1-carbonyl]-7-methylimidazo[1,2-a]pyrazin-8-one
—— (6R)-8-(3-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23ClN4O
(6R)-8-(3-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O3
(6S)-2-ethyl-8-(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H18FN3O4
6-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-(2-chlorophenyl)-2-[(2R)-2-ethylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O2
6-(2-chlorophenyl)-2-[(2R)-2-ethylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-(2-fluorophenoxy)acetate —— C18H16ClFO5
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-(2-fluorophenoxy)acetate
—— (6S)-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O3
(6S)-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2S)-1-morpholin-4-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile —— C16H21N3O2
6-[(2S)-1-morpholin-4-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(2-phenoxyacetyl)amino]acetate —— C20H20ClNO6
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(2-phenoxyacetyl)amino]acetate
—— (6R)-8-(3-methylbutyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N3O
(6R)-8-(3-methylbutyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2R)-1-[(3aS,7aR)-1,3,3a,4,7,7a-hexahydroisoindol-2-yl]hex-5-en-2-yl]oxy-N,N-dimethylpyridazin-3-amine —— C20H30N4O
6-[(2R)-1-[(3aS,7aR)-1,3,3a,4,7,7a-hexahydroisoindol-2-yl]hex-5-en-2-yl]oxy-N,N-dimethylpyridazin-3-amine
—— 6-[(3S)-3-[(4-methoxyphenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H21N3O5
6-[(3S)-3-[(4-methoxyphenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (6R)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H35N5O
(6R)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(3S)-3-(2-methyl-6-morpholin-4-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C21H26N6O
6-methyl-2-[(3S)-3-(2-methyl-6-morpholin-4-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[(3R)-3-[(4-methoxyphenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H21N3O5
6-[(3R)-3-[(4-methoxyphenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H18FN3O4
6-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-[(6S)-2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C19H26N4O2
6-[(6S)-2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— 6-[(6R)-2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C19H26N4O2
6-[(6R)-2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— (6S)-8-(3-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23ClN4O
(6S)-8-(3-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-acetylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6R)-8-(5-acetylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(4-aminopiperidine-4-carbonyl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N4O2
(6S)-8-(4-aminopiperidine-4-carbonyl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O3
(6R)-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2S)-1-[(3aS,7aR)-1,3,3a,4,7,7a-hexahydroisoindol-2-yl]hex-5-en-2-yl]oxy-N,N-dimethylpyridazin-3-amine —— C20H30N4O
6-[(2S)-1-[(3aS,7aR)-1,3,3a,4,7,7a-hexahydroisoindol-2-yl]hex-5-en-2-yl]oxy-N,N-dimethylpyridazin-3-amine
—— 6-(2-chlorophenyl)-2-[(2S)-2-ethylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O2
6-(2-chlorophenyl)-2-[(2S)-2-ethylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6R)-8-(4-aminopiperidine-4-carbonyl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N4O2
(6R)-8-(4-aminopiperidine-4-carbonyl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(3-fluoropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23FN4O
(6S)-8-(3-fluoropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(3R)-3-(2-methyl-6-morpholin-4-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C21H26N6O
6-methyl-2-[(3R)-3-(2-methyl-6-morpholin-4-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— (6R)-2-ethyl-8-(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O3
(6R)-2-ethyl-8-(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[2-(4-ethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O2
(6S)-2-ethyl-8-[2-(4-ethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[2-(4-ethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O2
(6R)-2-ethyl-8-[2-(4-ethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]-(5-ethyl-1H-pyrazol-4-yl)methanone —— C22H30N4O
[(6S)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]-(5-ethyl-1H-pyrazol-4-yl)methanone
—— 6-cyclopentyl-1-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C16H23N5O
6-cyclopentyl-1-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6S)-8-(3-methylbutyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N3O
(6S)-8-(3-methylbutyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(4-methylpentanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6R)-8-(4-methylpentanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]pyridine-2-carbonitrile —— C21H26N4O
6-[(3S)-3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]pyridine-2-carbonitrile
—— (6S)-8-(4-aminobutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6S)-8-(4-aminobutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-aminopyridin-3-yl)-[(3R)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]methanone —— C19H23N3O3
(6-aminopyridin-3-yl)-[(3R)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]methanone
—— 6-methyl-5-[[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]methyl]quinoline —— C22H31N3
6-methyl-5-[[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]methyl]quinoline
—— 6-(2-chlorophenyl)-2-[(3R)-3-hydroxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C21H21ClN4O3
6-(2-chlorophenyl)-2-[(3R)-3-hydroxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6R)-8-(6-oxo-1H-pyrimidine-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23N5O3
(6R)-8-(6-oxo-1H-pyrimidine-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-2-[(3S)-3-hydroxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C21H21ClN4O3
6-(2-chlorophenyl)-2-[(3S)-3-hydroxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6R)-8-(5-methylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O
(6R)-8-(5-methylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(pyridin-4-ylmethyl)-8-(2,2,3-trimethylbut-3-enoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H31N3O2
(6R)-2-(pyridin-4-ylmethyl)-8-(2,2,3-trimethylbut-3-enoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(5-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O2
(6S)-2-ethyl-8-(5-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-8-oxo-N-[(3R)-2-oxopyrrolidin-3-yl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C20H18ClN5O3
6-(2-chlorophenyl)-8-oxo-N-[(3R)-2-oxopyrrolidin-3-yl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(2-methyl-6-propan-2-ylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H35N5O
(6S)-2-[2-(dimethylamino)ethyl]-8-(2-methyl-6-propan-2-ylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one