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—— 6-[(3S)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-4-one —— C22H24N4O3
6-[(3S)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-4-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[[2-(1-adamantyl)acetyl]amino]acetate —— C24H29N3O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[[2-(1-adamantyl)acetyl]amino]acetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(2-methylbenzoyl)piperidine-4-carboxylate —— C24H25N3O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(2-methylbenzoyl)piperidine-4-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate —— C22H20N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate
—— 6-(4-Fluorophenyl)-8-(piperidin-1-ylmethyl)tetrazolo[1,5-a]pyridine —— C17H18FN5
6-(4-Fluorophenyl)-8-(piperidin-1-ylmethyl)tetrazolo[1,5-a]pyridine
—— (6-Bromo-1,3-benzodioxol-5-yl)methyl quinoxaline-6-carboxylate —— C17H11BrN2O4
(6-Bromo-1,3-benzodioxol-5-yl)methyl quinoxaline-6-carboxylate
—— 6-(4-fluorophenyl)-8-[[(2S)-2-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine —— C18H20FN5
6-(4-fluorophenyl)-8-[[(2S)-2-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine
—— (6-Bromo-1,3-benzodioxol-5-yl)methyl 2-(2-fluorophenyl)sulfanylacetate —— C16H12BrFO4S
(6-Bromo-1,3-benzodioxol-5-yl)methyl 2-(2-fluorophenyl)sulfanylacetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2-fluorophenyl)sulfanylacetate —— C18H15FN2O3S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2-fluorophenyl)sulfanylacetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate —— C20H20N2O3S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl quinoxaline-6-carboxylate —— C19H14N4O3
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl quinoxaline-6-carboxylate
—— 6-Methyl-3-[[4-(5-methylsulfonylthiadiazol-4-yl)piperidin-1-yl]methyl]chromen-4-one —— C19H21N3O4S2
6-Methyl-3-[[4-(5-methylsulfonylthiadiazol-4-yl)piperidin-1-yl]methyl]chromen-4-one
—— 6-(4-Fluorophenyl)-8-[(4-methylpiperidin-1-yl)methyl]tetrazolo[1,5-a]pyridine —— C18H20FN5
6-(4-Fluorophenyl)-8-[(4-methylpiperidin-1-yl)methyl]tetrazolo[1,5-a]pyridine
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-methyl-4-oxophthalazine-1-carboxylate —— C20H16N4O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-methyl-4-oxophthalazine-1-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3,4,5-trichloropyridine-2-carboxylate —— C16H10Cl3N3O3
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3,4,5-trichloropyridine-2-carboxylate
—— 6-(4-Fluorophenyl)-8-(pyrrolidin-1-ylmethyl)tetrazolo[1,5-a]pyridine —— C16H16FN5
6-(4-Fluorophenyl)-8-(pyrrolidin-1-ylmethyl)tetrazolo[1,5-a]pyridine
—— 6-(4-Fluorophenyl)-8-[(4-prop-2-enylpiperazin-1-yl)methyl]tetrazolo[1,5-a]pyridine —— C19H21FN6
6-(4-Fluorophenyl)-8-[(4-prop-2-enylpiperazin-1-yl)methyl]tetrazolo[1,5-a]pyridine
—— 6-Methyl-2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C15H17N5OS
6-Methyl-2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— 6-(4-fluorophenyl)-8-[[(3S)-3-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine —— C18H20FN5
6-(4-fluorophenyl)-8-[[(3S)-3-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxylate —— C20H20N2O3S
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxylate
—— 6-(4-fluorophenyl)-8-[[(3R)-3-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine —— C18H20FN5
6-(4-fluorophenyl)-8-[[(3R)-3-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine
—— 6-Phenyl-8-[[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl]tetrazolo[1,5-a]pyridine —— C22H23N7
6-Phenyl-8-[[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl]tetrazolo[1,5-a]pyridine
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate —— C21H21N3O5
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate
—— 6-Methyl-2-[[1-(2-methylphenyl)tetrazol-5-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C18H16N6OS
6-Methyl-2-[[1-(2-methylphenyl)tetrazol-5-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— 6-Phenyl-8-(piperidin-1-ylmethyl)tetrazolo[1,5-a]pyridine —— C17H19N5
6-Phenyl-8-(piperidin-1-ylmethyl)tetrazolo[1,5-a]pyridine
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-acetamido-4,5-dimethylthiophene-3-carboxylate —— C19H19N3O4S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-acetamido-4,5-dimethylthiophene-3-carboxylate
—— 6-ethyl-5-methyl-N-[3-(2-morpholin-4-ylethoxy)phenyl]-2-oxo-1H-pyridine-3-carboxamide —— C21H27N3O4
6-ethyl-5-methyl-N-[3-(2-morpholin-4-ylethoxy)phenyl]-2-oxo-1H-pyridine-3-carboxamide
—— 6-methyl-N-[3-(2-morpholin-4-ylethoxy)phenyl]imidazo[1,2-a]pyridine-2-carboxamide —— C21H24N4O3
6-methyl-N-[3-(2-morpholin-4-ylethoxy)phenyl]imidazo[1,2-a]pyridine-2-carboxamide
—— 6-Phenyl-8-[(4-pyridin-2-ylpiperazin-1-yl)methyl]tetrazolo[1,5-a]pyridine —— C21H21N7
6-Phenyl-8-[(4-pyridin-2-ylpiperazin-1-yl)methyl]tetrazolo[1,5-a]pyridine
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5-chloro-2-methoxybenzoate —— C18H15ClN2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5-chloro-2-methoxybenzoate
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate —— C21H23N3O5
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate
—— 6-[(4-pyridin-2-yl-1,4-diazepan-1-yl)sulfonyl]-3H-1,3-benzoxazol-2-one —— C17H18N4O4S
6-[(4-pyridin-2-yl-1,4-diazepan-1-yl)sulfonyl]-3H-1,3-benzoxazol-2-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetate —— C20H17N3O4S
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetate
—— 6-oxo-1-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-N-[3-(pyrazol-1-ylmethyl)phenyl]pyridine-3-carboxamide —— C21H18N6O3S
6-oxo-1-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-N-[3-(pyrazol-1-ylmethyl)phenyl]pyridine-3-carboxamide
—— 6-(4-fluorophenyl)-8-[[(2R)-2-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine —— C18H20FN5
6-(4-fluorophenyl)-8-[[(2R)-2-methylpiperidin-1-yl]methyl]tetrazolo[1,5-a]pyridine
—— 6-[[2-(3-fluorophenyl)-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one —— C21H18FN3O3S2
6-[[2-(3-fluorophenyl)-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate —— C21H21N3O5
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetate —— C20H17N3O4S
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(5-chlorothiophen-2-yl)-4-oxobutanoate —— C18H15ClN2O4S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(5-chlorothiophen-2-yl)-4-oxobutanoate
—— 6-[[2-(4-fluorophenyl)-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one —— C21H18FN3O3S2
6-[[2-(4-fluorophenyl)-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C19H16N4O4S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— 6-Methyl-2-[[5-[(3-methylphenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C20H18N4O3S
6-Methyl-2-[[5-[(3-methylphenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— (6-fluoro-1H-indol-2-yl)-[2-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]methanone —— C22H15F4N3OS
(6-fluoro-1H-indol-2-yl)-[2-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]methanone
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4,5-dimethoxy-2-nitrobenzoate —— C19H17N3O7
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4,5-dimethoxy-2-nitrobenzoate
—— 6-(2-indazol-1-ylethyl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-2-methylpyrimidin-4-amine —— C23H25N5O
6-(2-indazol-1-ylethyl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-2-methylpyrimidin-4-amine
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylate —— C18H16N2O3S
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-phenylmethoxybenzoate —— C24H20N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-phenylmethoxybenzoate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4,5,6,7-tetrahydro-1-benzothiophene-2-carboxylate —— C19H18N2O3S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4,5,6,7-tetrahydro-1-benzothiophene-2-carboxylate
—— 6-(2-indazol-1-ylethyl)-N-[(1R)-1-(2-methoxyphenyl)ethyl]-2-methylpyrimidin-4-amine —— C23H25N5O
6-(2-indazol-1-ylethyl)-N-[(1R)-1-(2-methoxyphenyl)ethyl]-2-methylpyrimidin-4-amine
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(difluoromethoxy)benzoate —— C18H14F2N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(difluoromethoxy)benzoate