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—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 3-(4-methyl-2-oxo-1,3-thiazol-3-yl)propanoate —— C16H16ClNO5S
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 3-(4-methyl-2-oxo-1,3-thiazol-3-yl)propanoate
—— (6S)-4-[(5-fluoro-2-pyrazol-1-ylphenyl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C18H23FN4O2
(6S)-4-[(5-fluoro-2-pyrazol-1-ylphenyl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— 6-[(4S)-4-(dimethylamino)azepan-1-yl]pyridine-2-carbonitrile —— C14H20N4
6-[(4S)-4-(dimethylamino)azepan-1-yl]pyridine-2-carbonitrile
—— 6-[(4R)-4-(dimethylamino)azepan-1-yl]pyridine-2-carbonitrile —— C14H20N4
6-[(4R)-4-(dimethylamino)azepan-1-yl]pyridine-2-carbonitrile
—— 6-cyclopentyl-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C18H25N7O
6-cyclopentyl-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— (6-chloroimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C14H16ClN3O3
(6-chloroimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— 6-cyclopentyl-N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C18H25N7O
6-cyclopentyl-N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— (6-chloroimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C14H16ClN3O3
(6-chloroimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— 6-tert-butyl-1-methyl-N-[2-[(3S)-oxan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C17H27N5O
6-tert-butyl-1-methyl-N-[2-[(3S)-oxan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6R)-2-methyl-6-[(1-methyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]heptan-2-ol —— C19H26N6O
(6R)-2-methyl-6-[(1-methyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]heptan-2-ol
—— 6-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C18H21F2N3O2
6-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-Amino-5-[2-(3,4-dimethylanilino)-5-methyl-1,3-thiazol-4-yl]-1,3-dimethylpyrimidine-2,4-dione —— C18H21N5O2S
6-Amino-5-[2-(3,4-dimethylanilino)-5-methyl-1,3-thiazol-4-yl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[4-[(6S)-6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C19H26N4O2
6-[4-[(6S)-6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-methoxy-N-[[(6S)-1,4-oxazepan-6-yl]methyl]pyrimidin-4-amine —— C11H18N4O2
6-methoxy-N-[[(6S)-1,4-oxazepan-6-yl]methyl]pyrimidin-4-amine
—— (6S)-2-methyl-6-[(1-methyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]heptan-2-ol —— C19H26N6O
(6S)-2-methyl-6-[(1-methyl-6-pyridin-2-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]heptan-2-ol
—— 6-tert-butyl-1-methyl-N-[2-[(3R)-oxan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C17H27N5O
6-tert-butyl-1-methyl-N-[2-[(3R)-oxan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6R)-6-[(dimethylamino)methyl]-N-(2,3-dimethylphenyl)-1,4-oxazepane-4-carboxamide —— C17H27N3O2
(6R)-6-[(dimethylamino)methyl]-N-(2,3-dimethylphenyl)-1,4-oxazepane-4-carboxamide
—— 6-methoxy-N-[[(6R)-1,4-oxazepan-6-yl]methyl]pyrimidin-4-amine —— C11H18N4O2
6-methoxy-N-[[(6R)-1,4-oxazepan-6-yl]methyl]pyrimidin-4-amine
—— (6S)-6-[(dimethylamino)methyl]-N-(2,3-dimethylphenyl)-1,4-oxazepane-4-carboxamide —— C17H27N3O2
(6S)-6-[(dimethylamino)methyl]-N-(2,3-dimethylphenyl)-1,4-oxazepane-4-carboxamide
—— 6-[(3S)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl]pyridine-2-carbonitrile —— C22H27N5O
6-[(3S)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl]pyridine-2-carbonitrile
—— 6-[[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-N-(3-methylphenyl)-1,3,5-triazine-2,4-diamine —— C21H23FN6
6-[[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-N-(3-methylphenyl)-1,3,5-triazine-2,4-diamine
—— 6-(4-fluorobenzoyl)-5-hydroxy-3H-thieno[2,3-d][1,3]thiazol-2-one —— C12H6FNO3S2
6-(4-fluorobenzoyl)-5-hydroxy-3H-thieno[2,3-d][1,3]thiazol-2-one
—— 6-(4-chlorobenzoyl)-5-hydroxy-3H-thieno[2,3-d][1,3]thiazol-2-one —— C12H6ClNO3S2
6-(4-chlorobenzoyl)-5-hydroxy-3H-thieno[2,3-d][1,3]thiazol-2-one
—— 6-[(3R)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl]pyridine-2-carbonitrile —— C22H27N5O
6-[(3R)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl]pyridine-2-carbonitrile
—— 6-methyl-5-phenyl-3-[(Z)-(2,4,6-trimethylphenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-one —— C23H21N3OS
6-methyl-5-phenyl-3-[(Z)-(2,4,6-trimethylphenyl)methylideneamino]thieno[2,3-d]pyrimidin-4-one
—— 6-[2-[3-Chloro-2-oxo-5-(trifluoromethyl)pyridin-1-yl]acetyl]-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one —— C19H14ClF3N2O3
6-[2-[3-Chloro-2-oxo-5-(trifluoromethyl)pyridin-1-yl]acetyl]-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
—— 6-[2-[[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one —— C19H15N3O4S
6-[2-[[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
—— 6-[[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-N-(3-methylphenyl)-1,3,5-triazine-2,4-diamine —— C21H23FN6
6-[[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-N-(3-methylphenyl)-1,3,5-triazine-2,4-diamine
—— 6-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one —— C16H22N4O3S
6-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one
—— (6-chloro-2-methylquinolin-4-yl)-[(4R)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methanone —— C18H21ClN2O3
(6-chloro-2-methylquinolin-4-yl)-[(4R)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methanone
—— 6-cyclopentyl-1-methyl-N-[2-[(3R)-oxolan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C17H25N5O
6-cyclopentyl-1-methyl-N-[2-[(3R)-oxolan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-cyclopentyl-1-methyl-N-[2-[(3S)-oxolan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C17H25N5O
6-cyclopentyl-1-methyl-N-[2-[(3S)-oxolan-3-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6-chloro-2-methylquinolin-4-yl)-[(4S)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methanone —— C18H21ClN2O3
(6-chloro-2-methylquinolin-4-yl)-[(4S)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methanone
—— 6-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C18H21F2N3O2
6-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one —— C16H22N4O3S
6-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one
—— (6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone —— C14H18ClN5O2
(6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone
—— 6-[[(3R)-1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]amino]pyridine-3-carbonitrile —— C17H15FN4O
6-[[(3R)-1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]amino]pyridine-3-carbonitrile
—— 6-ethyl-1-methyl-N-[(1S)-1-(1-methylpyrazol-4-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C15H21N7
6-ethyl-1-methyl-N-[(1S)-1-(1-methylpyrazol-4-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone —— C14H18ClN5O2
(6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone
—— 6-cyclopentyl-1-methyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H26N6
6-cyclopentyl-1-methyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-2-N-(2-methylphenyl)-1,3,5-triazine-2,4-diamine —— C19H19N7S2
6-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-2-N-(2-methylphenyl)-1,3,5-triazine-2,4-diamine
—— 6-cyclopentyl-1-methyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H26N6
6-cyclopentyl-1-methyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-ethyl-1-methyl-N-[(1R)-1-(1-methylpyrazol-4-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C15H21N7
6-ethyl-1-methyl-N-[(1R)-1-(1-methylpyrazol-4-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-(methoxymethyl)-1-methyl-N-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H26N6O
6-(methoxymethyl)-1-methyl-N-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6R)-5-acetyl-3-ethyl-6-(3-fluorophenyl)-4-methyl-1,6-dihydropyrimidin-2-one —— C15H17FN2O2
(6R)-5-acetyl-3-ethyl-6-(3-fluorophenyl)-4-methyl-1,6-dihydropyrimidin-2-one
—— 6-(methoxymethyl)-1-methyl-N-[2-[(3S)-3-phenylpyrrolidin-1-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H26N6O
6-(methoxymethyl)-1-methyl-N-[2-[(3S)-3-phenylpyrrolidin-1-yl]ethyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— [(6R)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone —— C18H21FN4O3
[(6R)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone
—— 6,7-Dimethyl-4-[[2-oxo-2-(5-phenyl-3,4-dihydropyrazol-2-yl)ethyl]sulfanylmethyl]chromen-2-one —— C23H22N2O3S
6,7-Dimethyl-4-[[2-oxo-2-(5-phenyl-3,4-dihydropyrazol-2-yl)ethyl]sulfanylmethyl]chromen-2-one
—— (6S)-4-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C16H26N4O2
(6S)-4-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— 6-cyclopentyl-1-methyl-N-[[(3R)-1-propylpiperidin-3-yl]methyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H32N6
6-cyclopentyl-1-methyl-N-[[(3R)-1-propylpiperidin-3-yl]methyl]pyrazolo[3,4-d]pyrimidin-4-amine